Herbicidal sulfonamides

ABSTRACT

Tetrazole-substituted benzenesulfonamides are useful as agricultural chemicals and, in particular, as growth regulants and herbicides.

RELATED APPLICATION

This application is a continuation-in-part of copending application U.S. Ser. No. 849,618, filed Apr. 11, 1986, now abandoned, which is a continuation-in-part of copending application U.S. Ser. No. 739,214, filed May 30, 1985, now abandoned.

BACKGROUND OF THE INVENTION

This invention relates to tetrazole-substituted benzene sulfonamides which are useful as agricultural chemicals such as growth regulants and herbicides.

U.S. Pat. No. 4,127,405 and U.S. Pat. No. 4,169,719 disclose herbicidal benzenesulfonylureas.

No. EP-A-165,753, published Dec. 27, 1985, discloses herbicidal thiophenesulfonamides of formula ##STR1## wherein Q is optionally substituted phenyl or an optionally substituted saturated or unsaturated 5- or 6-membered heterocyclic ring containing one to three heteroatoms.

No. EP-A-83,975 (published July 20, 1983) discloses herbicidal benzenesulfonamides of formula ##STR2## wherein Q is selected from various five or six-membered aromatic or partially unsaturated heterocyclic rings containing 2 or 3 heteroatoms selected from O, S or NR.

No. EP-A-85,476 (published Aug. 10, 1983) discloses herbicidal benzenesulfonamides of formulae ##STR3## wherein Q is selected from various 5-membered aromatic heterocycles, and their dihydro and tetrahydro analogs, which contain one heteroatom selected from O, S or NR, or Q is a saturated or partially unsaturated 6-membered ring containing one heteroatom selected from O or S; and

Q¹ is a 6-membered aromatic heterocycle containing one to three N atoms.

South African Patent Application No. 83/8416 (published May 12, 1984) discloses herbicidal benzenesulfonamides of formula ##STR4## wherein A is an unsaturated or only partially saturated 5- or 6-membered heterocyclic ring system which is bonded through a carbon atom and contains 1, 2 or 3 heteroatoms.

No. EP-A-116,518, published Aug. 22, 1984, discloses herbicidal sulfonamides of formula ##STR5## wherein X is NR₆ R₇, N(SO₂ R₉)₂ or ##STR6## A is CO, SO₂, CONR₂₃ or CO₂ ; B is C₁ -C₄ alkyl or C₂ -C₄ alkenyl; and

C is CO, CR₂₁ R₂₂ or SO₂.

U.S. Pat. No. 4,475,944 discloses herbicidal sulfamates, possessing an ortho-heterocyclic ring, such as those of formula ##STR7## wherein W is O, S or NR₁.

No. EP-A-164,268, published Dec. 11, 1985, discloses herbicidal benzylsulfonamides of formula ##STR8## wherein Q is a saturated, 5- or 6-membered ring containing 1 to 2 heteroatoms selected from 0-2S or 0-2O or an unsaturated 5- or 6-membered ring containing 1 to 3 heteroatoms selected from 0-1S, 0-1O or 0-3N and Q may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₁ -C₂ haloalkoxy, C₃ -C₄ alkenylthio, C₁ -C₂ haloalkylthio or SCH₂ CN.

No. EP-A-165,753, published Dec. 27, 1985, discloses herbicidal pyridinesulfonamides of formula ##STR9## wherein Q is phenyl optionally substituted with Cl, CH₃ O or CH₃, a saturated 5-membered ring containing 1 heteroatom selected from O or S, or an unsaturated 5- or 6-membered ring containing 1 to 3 heteroatoms selected from 0-1S, 0-1O or 0-3N and when Q is an unsaturated 5- or 6-membered ring, it may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₃ -C₄ alkenylthio, C₁ -C₂ haloalkoxy or C₁ -C₂ haloalkylthio.

No. EP-A-176,304, published Apr. 11, 1986, discloses herbicidal pyrazolesulfonamides such as those of formula ##STR10## wherein Q is a saturated 5- or 6-membered ring containing 1 heteroatom selected from 0-1S or 0-1O or an unsaturated 5- or 6-membered ring containing 1-3 heteroatoms selected from 0-1S, 0-1O or 0-3N and Q may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₃ -C₄ alkenylthio, C₃ -C₄ alkenyloxy, C₁ -C₂ haloalkoxy, C₁ -C₂ haloalkylthio, C₂ -C₄ cyanoalkylthio or C₁ -C₂ alkoxycarbonylmethylthio.

No. EP-A-141,777, published May 15, 1985, discloses ortho-benzyl-substituted sulfonylureas of the formula ##STR11## wherein Y is O or S; and

R¹⁷ is a 5- to 6-membered unsaturated heterocyclic radical including ##STR12## U.S. Pat. No. 4,602,936 carrying part of this disclosure, issued July 29, 1986.

South African Patent Application No. 83/0441, published July 25, 1983, discloses herbicidal benzenesulfonamides of formula ##STR13## wherein R₁ is H, halogen, NO₂, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₅ alkenyl or C₁ -C₄ alkoxycarbonyl;

R₂ is C₁ -C₃ alkyl or C₁ -C₃ alkoxy, each unsubstituted or substituted by 1 to 3 halogen atoms;

R₃ is halogen, H, NR₄ R₅, C₁ -C₃ alkyl, unsubstituted or substituted by 1 to 3 alkoxy, unsubstituted or substituted by methoxy, ethoxy, or 1 to 3 halogen atoms;

A is C₁ -C₄ alkylene or C₂ -C₄ alkenylene, each unsubstituted or substituted by C₁ -C₄ alkyl;

m is 0 or 1;

E is N or CH;

X is oxygen, sulfur, SO or SO₂ ; and

Q is, in part, a 5- or 6-membered heterocyclic ring bound through carbon or nitrogen, such heterocycles including furan, pyrane, thiophene, triazole, pyridine, pyrroline, oxaxole, isooxazole, thiazole, isothiazole, thiadiaxole, oxathiole, pyrrole, imidazole, pyrazole, pyrazine, pyrimidine, pyridazine, symmetrical and assymetrical triazines, oxdiazole, oxazine, furazane, pyridine-N-oxide, thiophene-S-oxide, benzthiophene, benzofuran, isobenzofuran, chromene, chromane, indole, isoindole, indazole, quinoline, isoquinoline, phthalazine, quinoxaline, quinazoline, quinoline, benzthiazole and benzimidiazole, and partially or completely hydrogenated and fused homoglogues thereof.

South African Patent Application No. 85/2646, published Oct. 11, 1985, discloses herbicidal benzenesulfonamides of formula ##STR14## wherein R₁ is H, halogen, NO₂, alkyl, alkoxy, alkoxycarbonyl or haloalkyl;

X is O, S, SO or SO₂ ;

Y is O or S;

E is CH or N;

R₂ and R₃ are independently alkyl, alkoxy or alkoxyalkyl;

A is alkylene or alkenylene;

m is 0 or 1;

Q is, in part, ##STR15## each of which is optionally substituted and/or optionally partially hydrogenated; and

X' is O, S or NR.

The presence of undesired vegetation causes substantial damage to useful crops, especially agricultural products that satisfy man's basic food needs, such as corn, soybeans, wheat and the like. The current population explosion and concomitant world food shortage demand improvements in the efficiency of producing these crops. Prevention or minimization of the loss of a portion of valuable crops by killing or inhibiting the growth of undesired vegetation is one way of improving this efficiency.

A wide variety of materials, useful for killing, or inhibiting (controlling) the growth of undesired vegetation is available. Such materials are commonly referred to as herbicides. The need exists, however, for still more effective herbicides that destroy or retard weeds without causing significant damage to useful crops.

SUMMARY OF THE INVENTION

This invention relates to novel compounds of Formula I, agriculturally suitable compositions containing them, and their method-of-use as preemergent or postemergent herbicides or as plant growth regulants. ##STR16## wherein J is ##STR17## W is O, S or NR_(X) ; R_(X) is H, OH, C₁ -C₃ alkyl, C₁ -C₃ alkoxy, allyloxy, propargyloxy, C₁ -C₃ haloalkyl, C₁ -C₃ haloalkoxy or NR_(Y) R_(Z) ;

R_(Y) is H or C₁ -C₃ alkyl;

R_(Z) is C₁ -C₃ alkyl;

G is O, S, SO or SO₂ ;

m is 0 or 1;

n is 0, 1 or 2;

R is H or CH₃ ;

E is a single bond, CH₂ or O;

Q is ##STR18## R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(a) R_(b), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, SCN, CO₂ R_(c), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio or CN;

R₂ is H, C₁ -C₃ alkyl, allyl or phenyl;

R₃ is H, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, CH₂ --(C₂ -C₅ alkenyl), CH₂ (C₂ -C₅ haloalkenyl), CH₂ (C₂ -C₅ alkynyl), CH₂ (C₂ -C₅ haloalkynyl), C₆ H₅ or C₁ -C₄ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, C₁ -C₂ alkylsulfinyl or C₁ -C₂ alkylsulfonyl;

R₄ is H, halogen, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, C₂ -C₆ alkenyl, C₂ -C₆ haloalkenyl, C₂ -C₆ alkynyl, C₃ -C₆ haloalkynyl, C₆ H₅, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, OCH₂ CH₂ O--(C₁ -C₂ alkyl) or di(C₁ -C₃ alkyl)amino;

R₅ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, allyl or propargyl;

R_(a) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy;

R_(b) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or

R_(a) and R_(b) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --;

R_(c) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl;

A is ##STR19## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₃ -C₅ cycloalkyl;

Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, C₁ -C₄ haloalkyl, C₂ -C₄ alkynyl, azido, cyano, ##STR20## or --N(OCH₃)CH₃ ; p is 2 or 3;

L₁ and L₂ are independently O or S;

R₆ is H or CH₃ ;

R₇ and R₈ are independently C₁ -C₃ alkyl;

Z is CH, N, CCH₃, CC₂ H₅, CCl or CBr;

Y₁ is O or CH₂ ;

X₁ is CH₃, OCH₃, OC₂ H₅ or OCF₂ H;

X₂ is CH₃, C₂ H₅ or CH₂ CF₃ ;

Y₂ is OCH₃, OC₂ H₅, SCH₃, SC₂ H₅, CH₃ or CH₂ CH₃ ;

X₃ is CH₃ or OCH₃ ;

Y₃ is H or CH₃ ;

X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl;

Y₄ is CH₃, OCH₃, OC₂ H₅ or Cl; and

Z¹ is CH or N;

and their agriculturally suitable salts; provided that

(a) when X is Cl, F, Br or I, then Z is CH and Y is OCH₃, OC₂ H₅, N(OCH₃)CH₃, NHCH₃, N(CH₃)₂ or OCF₂ H;

(b) when X or Y is C₁ haloalkoxy, then Z is CH;

(c) when J is J-9 and n is O, then Q is Q-1 or Q-2;

(d) when E is O, then J is J-1;

(e) when W is S, then A is A-1, R is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂ or ##STR21## (f) when the total number of carbon atoms in X and Y is greater than 4, then the carbon content of R₁, R₃, R₄ and R₅ must each be less than or equal to 2;

(g) X₄ and Y₄ cannot simultaneously be Cl;

(h) when J is J-1 and m is 0, then n is 0; and

(i) when n is 0 and m is 1, then Q is Q-1 or Q-2.

In the above definitions, the term "alkyl" used either alone or in compound words such as "alkylthio" or "haloalkyl", denotes straight chain or branched alkyl, e.g., methyl, ethyl, n-propyl, isopropyl or the different butyl, pentyl or hexyl isomers.

Alkoxy denotes methoxy, ethoxy, n-propoxy, isopropoxy and the different butyl isomers.

Alkenyl denotes straight chain or branched alkenes, e.g., vinyl, 1-propenyl, 2-propenyl, 3-propenyl and the different butenyl, pentenyl or hexenyl isomers.

Alkynyl denotes straight chain or branched alkynes, e.g., ethynyl, 1-propynyl, 2-propynyl and the different butynyl, pentynyl and hexynyl isomers.

Alkylsulfonyl denotes methylsulfonyl, ethylsulfonyl or the different propylsulfonyl isomers.

Alkylthio, alkylsulfinyl, alkylamino, etc. are defined in an analogous manner.

Cycloalkyl denotes cyclopropyl, cyclobutyl, cyclopentyl and cyclohexyl.

The term "halogen", either alone or in compound words such as "haloalkyl", denotes fluorine, chlorine, bromine or iodine.

In terms such as C₂ -C₃ alkylthioalkyl, the specified number of carbon atoms is meant to define the total number of carbon atoms in that substituent group. For example, C₂ -C₃ alkylthioalkyl would designate CH₂ SCH₃, CH₂ SC₂ H₅, CH₂ CH₂ SCH₃ or CH(CH₃)SCH₃, and C₂ -C₅ alkoxyalkoxy would represent OCH₂ OCH₃ through O(CH₂)₄ OCH₃ or OCH₂ O(CH₂)₃ CH₃ and the various structural isomers embraced therein.

Preferred for reasons of increased ease of synthesis and/or greater herbicidal efficacy are:

(1) Compounds of Formula I where E is a single bond.

(2) Compounds of Formula I where E is CH₂.

(3) Compounds of Formula I where E is O.

(4) Compounds of Preferred 1 where

m is 0; and

W is O.

(5) Compounds of Preferred 4 where

X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, cyclopropyl, Cl, F, Br, I, OCF₂ H, CH₂ F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and

Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR22## OCF₂ H, SCF₂ H, OCF₂ Br, C.tbd.CH or C.tbd.CCH₃.

(6) Compounds of Preferred 5 where

R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; and

n is 0.

(7) Compounds of Preferred 6 where

R₃ is H, C₁ -C₃ alkyl, C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; and

R₄ is H, C₁ -C₃ alkyl, C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, N(CH₃)₂, alkyl, propargyl or C₁ -C₂ alkyl substituted with 1-3 atoms of F, Cl or Br.

(8) Compounds of Preferred 7 where J is J-1.

(9) Compounds of Preferred 8 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(10) Compounds of Preferred 9 where Q is Q₁.

(11) Compounds of Preferred 9 where Q is Q₂.

(12) Compounds of Preferred 9 where Q is Q₃.

(13) Compounds of Preferred 9 where Q is Q₄.

(14) Compounds of Preferred 9 where Q is Q₅.

(15) Compounds of Preferred 9 where Q is Q₆.

(16) Compounds of Preferred 9 where Q is Q₇.

(17) Compounds of Preferred 7 where J is J₂.

(18) Compounds of Preferred 17 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(19) Compounds of Preferred 18 where Q is Q₁.

(20) Compounds of Preferred 18 where Q is Q₂.

(21) Compounds of Preferred 18 where Q is Q₃.

(22) Compounds of Preferred 18 where Q is Q₄.

(23) Compounds of Preferred 18 where Q is Q₅.

(24) Compounds of Preferred 18 where Q is Q₆.

(25) Compounds of Preferred 18 where Q is Q₇.

(26) Compounds of Preferred 7 where J is J₃.

(27) Compounds of Preferred 26 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(28) Compounds of Preferred 27 where Q is Q₁.

(29) Compounds of Preferred 27 where Q is Q₂.

(30) Compounds of Preferred 27 where Q is Q₃.

(31) Compounds of Preferred 27 where Q is Q₄.

(32) Compounds of Preferred 27 where Q is Q₅.

(33) Compounds of Preferred 27 where Q is Q₆.

(34) Compounds of Preferred 27 where Q is Q₇.

(35) Compounds of Preferred 7 where J is J₄.

(36) Compounds of Preferred 35 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(37) Compounds of Preferred 36 where Q is Q₁.

(38) Compounds of Preferred 36 where Q is Q₂.

(39) Compounds of Preferred 36 where Q is Q₃.

(40) Compounds of Preferred 36 where Q is Q₄.

(41) Compounds of Preferred 36 where Q is Q₅.

(42) Compounds of Preferred 36 where Q is Q₆.

(43) Compounds of Preferred 36 where Q is Q₇.

(44) Compounds of Preferred 7 where J is J₅.

(45) Compounds of Preferred 44 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(46) Compounds of Preferred 45 where Q is Q₁.

(47) Compounds of Preferred 45 where Q is Q₂.

(48) Compounds of Preferred 45 where Q is Q₃.

(49) Compounds of Preferred 45 where Q is Q₄.

(50) Compounds of Preferred 45 where Q is Q₅.

(51) Compounds of Preferred 45 where Q is Q₆.

(52) Compounds of Preferred 45 where Q is Q₇.

(53) Compounds of Preferred 7 where J is J₆.

(54) Compounds of Preferred 53 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(55) Compounds of Preferred 54 where Q is Q₁.

(56) Compounds of Preferred 54 where Q is Q₂.

(57) Compounds of Preferred 54 where Q is Q₃.

(58) Compounds of Preferred 54 where Q is Q₄.

(59) Compounds of Preferred 54 where Q is Q₅.

(60) Compounds of Preferred 54 where Q is Q₆.

(61) Compounds of Preferred 54 where Q is Q₇.

(62) Compounds of Preferred 7 where J is J₇.

(63) Compounds of Preferred 62 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(64) Compounds of Preferred 63 where Q is Q₁.

(65) Compounds of Preferred 63 where Q is Q₂.

(66) Compounds of Preferred 63 where Q is Q₃.

(67) Compounds of Preferred 63 where Q is Q₄.

(68) Compounds of Preferred 63 where Q is Q₅.

(69) Compounds of Preferred 63 where Q is Q₆.

(70) Compounds of Preferred 63 where Q is Q₇.

(71) Compounds of Preferred 7 where J is J₈.

(72) Compounds of Preferred 71 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(73) Compounds of Preferred 72 where Q is Q₁.

(74) Compounds of Preferred 72 where Q is Q₂.

(75) Compounds of Preferred 72 where Q is Q₃.

(76) Compounds of Preferred 72 where Q is Q₄.

(77) Compounds of Preferred 72 where Q is Q₅.

(78) Compounds of Preferred 72 where Q is Q₆.

(79) Compounds of Preferred 72 where Q is Q₇.

(80) Compounds of Preferred 7 where J is J₉.

(81) Compounds of Preferred 80 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(82) Compounds of Preferred 81 where Q is Q₁.

(83) Compounds of Preferred 81 where Q is Q₂.

(84) Compounds of Preferred 81 where Q is Q₃.

(85) Compounds of Preferred 81 where Q is Q₄.

(86) Compounds of Preferred 81 where Q is Q₅.

(87) Compounds of Preferred 81 where Q is Q₆.

(88) Compounds of Preferred 81 where Q is Q₇.

(89) Compounds of Preferred 7 where J is J₁₀.

(90) Compounds of Preferred 89 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(91) Compounds of Preferred 90 where Q is Q₁.

(92) Compounds of Preferred 90 where Q is Q₂.

(93) Compounds of Preferred 90 where Q is Q₃.

(94) Compounds of Preferred 90 where Q is Q₄.

(95) Compounds of Preferred 90 where Q is Q₅.

(96) Compounds of Preferred 90 where Q is Q₆.

(97) Compounds of Preferred 90 where Q is Q₇.

(98) Compounds of Preferred 7 where J is J₁₁.

(99) Compounds of Preferred 98 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(100) Compounds of Preferred 99 where Q is Q₁.

(101) Compounds of Preferred 99 where Q is Q₂.

(102) Compounds of Preferred 99 where Q is Q₃.

(103) Compounds of Preferred 99 where Q is Q₄.

(104) Compounds of Preferred 99 where Q is Q₅.

(105) Compounds of Preferred 99 where Q is Q₆.

(106) Compounds of Preferred 99 where Q is Q₇.

(107) Compounds of Preferred 7 where J is J₁₂.

(108) Compounds of Preferred 107 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(109) Compounds of Preferred 108 where Q is Q₁.

(110) Compounds of Preferred 108 where Q is Q₂.

(111) Compounds of Preferred 108 where Q is Q₃.

(112) Compounds of Preferred 108 where Q is Q₄.

(113) Compounds of Preferred 108 where Q is Q₅.

(114) Compounds of Preferred 108 where Q is Q₆.

(115) Compounds of Preferred 108 where Q is Q₇.

(116) Compounds of Preferred 7 where J is J₁₃.

(117) Compounds of Preferred 116 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(118) Compounds of Preferred 117 where Q is Q₁.

(119) Compounds of Preferred 117 where Q is Q₂.

(120) Compounds of Preferred 117 where Q is Q₃.

(121) Compounds of Preferred 117 where Q is Q₄.

(122) Compounds of Preferred 117 where Q is Q₅.

(123) Compounds of Preferred 117 where Q is Q₆.

(124) Compounds of Preferred 117 where Q is Q₇.

(125) Compounds of Preferred 2 where

m is 0;

n is 0;

J is J-1, J-2, J-3, J-8, J-10 or J-11;

W is O;

R is H;

R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H;

R₃ is H, C₁ -C₃ alkyl, CH₂ CH₂ OCH₃, CH₂ CH₂ Cl, Ch₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl;

R₄ is H or C₁ -C₃ alkyl;

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(126) Compounds of Preferred 3 where

m is 0;

R is H;

R₁ is H;

R₃ is H or C₁ -C₃ alkyl;

R₄ is H or C₁ -C₃ alkyl;

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

Specifically preferred for reasons of greatest ease of synthesis and/or greatest herbicidal efficacy are:

N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-ethyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 223°-225° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-methyl-6-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 178°-189° C.;

N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 225°-227° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 207°-210° C.;

N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 224°-226° C.;

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole-5-sulfonamide, m.p. 181°-183° C.; and

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole-5-sulfonamide, m.p. 171°-173° C.

DETAILED DESCRIPTION OF THE INVENTION Synthesis

Compounds of Formula I can be synthesized by one or both of the methods shown below in Equation 1 and 2.

Equation 1 illustrates the reaction of sulfonyl isocyanates and isothiocyanates of Formula II with the appropriate heterocyclic amines of Formula III to give the desired sulfonylureas and sulfonylthioureas of Formula I. ##STR23## wherein J, W, R, and A are as previously defined.

The reaction of Equation 1 is best carried out in an inert aprotic solvent such as methylene chloride, tetrahydrofuran or acetonitrile at a temperature between 0° and 82° C. A catalytic amount of 1,4-diazabicyclo[2,2,2]octane (DABCO®) may be used to accelerate the reaction. In cases in which the products are insoluble in the reaction solvent, they may be isolated by simple filtration. When the products are soluble, they can be isolated by evaporation of the solvent and trituration of the residue with solvents such as 1-chlorobutane, diethyl ether or ethyl acetate, and filtration.

Compounds of Formula I can be prepared as shown below in Equation 2 by the reaction of sulfonamides IV with the phenyl ester of the appropriate carbamic acid or thiocarbamic acid of Formula V, in the presence of an equimolar quantity of a tertiary amine base such as 1,8-diazabicyclo[5,4,0]undec-7-ene (DBU). ##STR24## wherein J, R, W and A are as previously defined.

The reaction shown in Equation 2 is best carried out at 25° C. in a solvent such as dioxane or acetonitrile for 1-2 hours under an inert atmosphere as described in European Patent Application No. 70,804 (published Jan. 26, 1983). The desired products of Formula I can be conveniently isolated by acidifying the reaction solution with aqueous hydrochloric acid. Alternatively, the aqueous layer can be extracted with a solvent such as methylene chloride or ethyl acetate. Drying and evaporation of the solvent affords the desired products.

The phenylcarbamates and phenylthiocarbamates of Formula V can be prepared by methods, or modifications thereof known to those skilled in the art, described in South African Patent Application No. 82/5671 and South African Patent Application No. 82/5045.

A judicious choice of the appropriate methods for preparing compounds of Formula I must take into account the nature of the substituents contained within the J values (J₁ -J₆), namely Q and R₁, and their chemical compatibility with the reaction conditions of Equations 1 and 2.

Sulfonyl isocyanates of Formula II can be prepared as shown in Equation 3 by the reaction of sulfonamides of the general structure IV with phosgene in the presence of n-butyl isocyanate and a catalytic amount of 1,4-diazabicyclo[2.2.2]octane (DABCO). ##STR25## wherein J is as previously defined, provided E is not oxygen.

The reaction depicted in Equation 3 is best carried out according to the procedure described in U.S. Pat. No. 4,238,621.

Alternatively, sulfonyl isocyanates II can be prepared via phosgenation of the preformed n-butylureas of Formula VI as represented in Equation 4. ##STR26## wherein J is as previously defined, provided E is not oxygen.

The compounds of Formula VI are conveniently prepared by stirring a mixture of the appropriate sulfonamide IV, anhydrous potassium carbonate, and n-butyl isocyanate in a suitable solvent such as acetone or methyl ethyl ketone at 25° to 80° C. until all of the isocyanate has reacted. The products are isolated by quenching in dilute aqueous acid and recrystallizing the insoluble solid. The n-butylureas VI are then treated with phosgene and a catalytic amount of DABCO in refluxing xylenes or chlorobenzene in a manner analogous to that described in the reference cited for Equation 3.

Alternatively, treatment of the sulfonamides of Formula IV with thionyl chloride gives intermediate N-sulfinylsulfonamides VII, which afford sulfonylisocyanates II (where W is O) upon exposure to phosgene in the presence of a catalytic amount of pyridine. ##STR27##

The reaction of Equation 5 can best be performed according to the procedure of H. Ulrich, B. Tucker and A. Sayigh, J. Org. Chem., 34, 3200 (1969).

Sulfonyl isothiocyanates II (where W is S) are known in the art and are prepared from the corresponding sulfonamides (IV) by reaction with carbon disulfide and potassium hydroxide followed by treatment of the resulting dipotassium salt with phosgene. Such a procedure is described in Arch. Pharm. 299, 174 (1966).

A judicious choice of the appropriate method for preparing compounds of Formula II must take into account the nature of the substituents contained within the J values (J₁ -J₆), namely Q and R₁, and their chemical compatability with reaction conditions of Equations 3-5.

The required sulfonamides of Formula IV can be synthesized by one or more of the methods shown below.

Equation 6 depicts the reaction of sulfonyl chlorides of Formula VIII with ammonia to give sulfonamides of Formula IVa. ##STR28## wherein J is as previously defined, provided E is not oxygen.

The amination of Equation 6 can be effected by adding at least two molar equivalents of either anhydrous ammonia or concentrated ammonium hydroxide to a solution of the sulfonyl chloride VIII in a solvent such as diethyl ether, methylene chloride, or tetrahydrofuran at temperatures between -30° and 25° C. The sulfonamides of Formula IVa are isolated either by filtration, in which case the ammonium chloride by-product is removed by washing with water, or extraction into an organic solvent such as methylene chloride. Drying and evaporation of the solvent affords the sulfonamides IVa, which are usually sufficiently pure to be carried directly on to the next step.

Sulfonyl chlorides of Formula VIII can be prepared by one or more of the methods shown below in Equations 7, 8 and 9.

The reaction of an appropriately substituted N-arylhydroxylamine of Formula IX, as shown in Equation 7, and subsequent displacement with sulfur dioxide in the presence of cupric or cuprous chloride yields the desired sulfonyl chloride of Formula VIII. ##STR29##

The reaction of Equation 7 can be carried out by combining the appropriate arylhydroxylamine with aqueous concentrated hydrochloric acid and acetic acid and adding an aqueous solution of sodium nitrite at -10° to 10° C. After being stirred for 10 minutes to two hours the reaction mixture is added to a mixture of acetic acid, a catalytic amount of cuprous or cupric chloride and excess sulfur dioxide at -5° to 20° C. After being stirred for 0.5 to 24 hours the mixture is diluted with cold water and the product is extracted into a solvent such as methylene chloride or ethyl ether.

The solution of sulfonyl chloride thus obtained can be treated as in Equation 6 to prepare the desired sulfonamide IVa.

Diazotization of appropriately substituted amine derivatives of Formula X, as shown in Equation 8, and subsequent reaction with sulfur dioxide in the presence of either cupric or cuprous chloride gives the desired products of Formula VIII. ##STR30##

The reaction of Equation 8 can be effected by methods analogous to those described in EP-A Nos. 83,975 and 85,476 (published Aug. 10, 1983). In Equation 8, a substituted amine X, in concentrated hydrochloric acid is treated with a solution of sodium nitrite in water at -5° to 5° C. After being stirred for 10 minutes to one hour at about 0° C., the solution is added to a mixture of excess sulfur dioxide and a catalytic amount of cupric or cuprous chloride in acetic acid at about 10° C. After being stirred for 0.25 to 24 hours at temperatures between 10° to 25° C., the solution is poured into a large excess of ice water. The sulfonyl chloride VIII can be isolated by filtration, or by extraction into a solvent such as methylene chloride or ether, followed by drying and evaporation of the solvent.

Alternatively, diazotization of appropriately substituted amine hydrochloride salts of Formula Xa can be effected under anhydrous conditions, as shown in Equation 8a, and subsequent reaction with sulfur dioxide and cupric chloride gives the desired products of Formula VIII. ##STR31##

The amine hydrochloride salts Xa are diazotized with an alklnitrite in a suitable solvent such as acetonitrile or acetone, and the resulting diazonium salts are reacted with sulfur dioxide and cupric chloride to give sulfonyl chlorides VIII. M. Doyle, in J. Org. Chem. 42, 2426, 2431 (1977), describes conditions for conducting similar Meerwein reactions.

Sulfonyl chlorides can also be prepared as shown below in Equation 9 by metal halogen exchange or directed lithiation of appropriately substituted aryl or heterocyclic substrates XI, and trapping with sulfuryl chloride. ##STR32## wherein J is as previously described provided that R₁ is not CO₂ R_(c), C₁ -C₃ haloalkyl, Br, nitro, C₁ -C₃ alkylsulfonyl or CN.

The lithiation shown in Equation 9 can be performed according to the procedure of S. H. Bhattacharyl, et al., J. Chem. Soc. (C), 1265 (1968) or by procedures reviewed by H. Gschwind and H. Rodriquez in Organic Reactions, Vol. 26, Wiley, N.Y., 1979, and references cited within.

Compounds of Formula VIII can be prepared via oxidative chlorination of the appropriate thioethers or mercaptans of Formula XII as represented in Equation 10. ##STR33## wherein J is as previously defined, R₁₅ is H, C₂ -C₄ alkyl or benzyl, R₁ is not C₁ -C₃ alkylthio or C₁ -C₃ alkylsulfinyl, and R₄ is not C₁ -C₄ alkylthio or C₁ -C₄ alkylsulfinyl.

The reaction of Equation 10 can be carried out by treating a solution of the thioether XII in a solvent such as acetic acid in the presence of at least 2.5 equivalents of water and at least 3.0 equivalents of chlorine at 0°-30° C. for 0.25 to 5 hours. The reaction is poured into ice-water and the product is isolated by extraction with a suitable solvent such as methylene chloride, dried, and the solvent evaporated to yield a product sufficiently pure to be carried directly on to the next step.

Arylmethanesulfonyl chlorides of Formula VIIIb can be prepared from appropriately substituted benzyl chlorides or bromides of Formula XIII by a simple two-step procedure outlined in Equation 11. ##STR34## wherein J'CH₂ is defined as for J-1 through J-6 where E is CH₂ ;

R₁, R₄ and Q are as previously defined except R₁ is not C₁ -C₃ l alkylthio or C₁ -C₃ alkylsulfinyl, and R₄ is not C₁ -C₄ alkylthio or C₁ -C₄ alkylsulfinyl; and

M is Cl or Br.

The conversion of alkyl halides of Formula XIII to isothiouronium salts of Formula XIV can be carried out by the procedure or T. B. Johnson and J. M. Sprague, J. Am. Chem. Soc., 58, 1348 (1936); 59 1837 and 2439 (1937); 61 176 (1939). Oxidative chlorination of isothouronium salts such as XIV to afford sulfonyl chlorides of Formula VIIIb is best carried out according to the procedure of Johnson as described in J. Am. Chem. Soc., 61 2548 (1939).

The requisite tetrazole substituted intermediates can be prepared by various methods depending on the nature of the aromatic ring in J (J-1 to J-6) systems on which the tetrazole is substituted and the nature of the other substituents present on J (J-1 to J-6). These intermediates can be prepared by one skilled in the art by the methods referred to in the following reviews on tetrazole chemistry: F. R. Benson, "Heterocyclic Compounds" (R. C. Elderfield, Ed.) 8, 1-104, John Wiley and Sons, New York, (1967); R. N. Butler. "Advances in Heterocyclic Chem.", 21, 323-436, Academic Press (1977); R. N. Butler, "Comprehensive Heterocyclic Chem.", (K. T. Potts, Ed.) 5, 791-838, Pergamon Press (1984) and F. R. Benson, "High Nitrogen Compounds", John Wiley and Sons, New York (1983).

The heterocyclic amines of Formula III in Equation 1 above can be prepared by methods known in the literature, or simple modifications thereof, by those skilled in the art. For instance, EP-A NO. 84,224 (published July 27, 1983) and W. Braker et al., J. Am. Chem. Soc., 69, 3072 (1947) describes method for preparing aminopyridines and triazines substituted by acetal groups such as dialkoxymethyl or 1,3-dioxolan-2-yl, among other groups. Also, for example, South African patent applications Nos. 82/5045 and 82/5671 describe methods for preparing aminopyrimidines and triazines substituted by haloalkyl or haloalkylthio groups such as OCH₂ CH₂ F, OCH₂ CF₃, SCF₂ H, or OCF₂ H, among other groups. South African patent application No. 83/7434 (published Oct. 5, 1983) describes methods for the synthesis of cyclopropylpyrimidines and triazines substituted by such groups as alkyl, haloalkyl, alkoxy, haloalkoxy, alkylamino, dialkylamino or alkoxyalkyl.

The 5,6-dihydrofuro[2,3-d]pyrimidine-2-amines, the cyclopenta[d]pyrimidin-2-amines (III, A is A-2) and the 6,7-dihydro-5H-pyrano[2,3-d]pyrimidin-2-amines (III, A is A-3) can be prepared as described in EP-A No. 15,683. The furo[2,3-d]pyrimidin-2-amines (III, A is A-4) are described in EP-A No. 46,677.

Compounds of Formula III, where A is A-5, are described in No. EP-A-73,562. Compound of Formula III, where A is A-6 are described in No. EP-A-94,260.

In addition, general methods for preparing aminopyrimidines and triazines have been reviewed in the following publications:

"The Chemistry of Heterocyclic Compounds", a series published by Interscience Publishers, Inc., New York and London;

"Pyrimidines", Vol. 16 of the same series by D. J. Brown;

"s-Triazines and Derivatives", Vol. 13 of the same series by E. M. Smolin and L. Rappoport; and

F. C. Schaefer, U.S. Pat. No. 3,154,547 and K. R. Huffman and F. C. Schaefer, J. Org. Chem., 28, 1812 (1963), which describes the synthesis of triazines.

Agriculturally suitable salts of compounds of Formula I are also useful herbicides and can be prepared in a number of ways known to the art. For example, metal salts can be made by contacting compounds of Formula I with a solution of an alkali or alkaline earth metal salt having a sufficiently basic anion (e.g., hydroxide, alkoxide or carbonate). Quaternary amine salts can be made by similar techniques.

Salts of compounds of Formula I can also be prepared by exchange of one cation for another. Cationic exchange can be effected by direct contact of an aqueous solution of a salt of a compound of Formula I (e.g. alkali or quaternary amine salt) with a solution containing the cation to be exchanged. This method is most effective when the desired salt containing the exchange cation is insoluble in water and can be separated by filtration.

Exchange may also be effected by passing an aqueous solution of a salt of a compound of Formula I (e.g., an alkali metal or quaternary amine salt) through a column packed with a cation exchange resin containing the cation to be exchanged for that of the original salt and the desired product is eluted from the column. This method is particularly useful when the desired salt is water-soluble, e.g., a potassium, sodium or calcium salt.

Acid addition salts, useful in this invention, can be obtained by reacting a compound of Formula I with a suitable acid, e.g., p-toluenesulfonic acid, trichloroacetic acid or the like.

The preparation of the compounds of this invention is further illustrated by the following specific examples.

EXAMPLE 1 1-(2-Chlorosulfonylphenyl)-5-methyl-1H-tetrazole

To 5 g of 1-(2-hydroxylaminophenyl)-5-methyl-1H-tetrazole in 12 mL of 37% hydrochloric acid and 5 mL of acetic acid at 0°-5° C. was added 2.3 g of sodium nitrite in 10 mL of water. The resultant solution was stirred at -5° to +5° C. for one hour and then added portionwise, with stirring, to a mixture of 25 mL of acetic acid, 0.5 g of cupric chloride and 5 mL of liquified sulfur dioxide at below 5° C. After stirring for two hours, during which time the mixture was allowed to warm to room temperature, it was poured into 150 mL of ice and water and extracted twice with 150 mL of methylene chloride. The methylene chloride solution was washed three times with 100 mL portions of water, two times with 100 mL of saturated aqeuous sodium bicarbonate followed by single washes with 100 mL of saturated aqueous sodium chloride and 100 mL of water. The methylene chloride solution was then dried over magnesium sulfate and filtered to yield a solution containing the desired sulfonylchloride. This solution was used without further work-up to prepare the sulfonamide of Example 2.

EXAMPLE 2 1-(2-Aminosulfonylphenyl)-5-methyl-1H-tetrazole

Twenty-five mL of 28% ammonium hydroxide was added to the methylene chloride solution obtained from Example 2 and the mixture was stirred for two hours and concentrated in vacuo to yield a mixture of an oil and a solid. The solid product was separated by filtration and washed with water to yield 2.2 g of the desired product, which melted at 141°-148° C. Infrared absorption peaks at 3260 and 3360 cm⁻¹ were consistent for NH₂ and 1160 and 1350 cm⁻¹ consistent for the SO₂ of the desired product. Elem. anal. calc'd for C₈ H₉ N₅ O₂ S:C, 40.15; H, 3.79; N, 29.26, S, 13.39. Found: C, 40.43; H, 3.84; N, 29.61; S, 13.04.

EXAMPLE 3 5-(2-Chlorosulfonylphenyl)-2-methyl-2H-tetrazole and 5-(2-chlorosulfonylphenyl)-1-methyl-1H-tetrazole

To 5 g of a mixture of 5-(2-hydroxylaminophenyl)-2-methyl-2H-tetrazole and 5-(2-hydroxyaminophenyl)-1-methyl-1H-tetrazole dissolved in 12 mL of 37% hydrochloric acid and 5 mL of acetic acid was added with stirring 2.3 g of sodium nitrite dissolved in 10 mL of water at -5° to 5° C. After one hour this solution was added, at 0°-5° C., portionwise to a mixture of 25 mL of acetic acid, 0.5 g of cupric chloride and 5 mL of liquified sulfur dioxide. After the addition was completed the cooling bath was removed and the reaction mixture was allowed to warm to 31° C. whereupon the cooling bath was reapplied and the stirring was continued until two and one half hours after completion of the addition. The mixture was then poured into ice and worked up as described in Example 1 except that the desired methylene chloride solution was concentrated in vacuo to yield an oil which solidified. This product, (3.28 g) which was a mixture of the desired sulfonylchlorides, was of sufficient purity for the preparation of the sulfonamides of Example 4.

EXAMPLE 4 5-(2-Aminosulfonylphenyl)-2-methyl-2H-tetrazole and 5-(2-aminosulfonylphenyl)-1-methyl-1H-tetrazole

The solid product obtained in Example 3 was dissolved in 50 mL of tetrahydrofuran and added portionwise to 20 mL of 28% ammonium hydroxide. The mixture was stirred for one hour and concentrated in vacuo. Water was added to the residue, the mixture filtered and the solid washed with a small amount of cold water to yield 1.3 g of the isomer mixture. Infrared absorption spectra showed peaks at 3260 and 3360 cm⁻¹ consistent for NH₂ and 1160 and 1330 consistent for the SO₂ group of the desired product. Elem. anal. calc'd for C₈ H₉ N₅ O₂ S:C, 40.15; H, 3.79; N, 29.26; S, 13.39. Found: C, 40.49; H, 3.86; N, 29.99; S, 13.75.

EXAMPLE 5 5-(2-Aminosulfonylphenyl)-1-methyl-1H-tetrazole

To 4.4 g of 5-(2-ethylthiophenyl)-1-methyl-1H-tetrazole in 40 mL of propionic acid and 1.08 g of waer at -10° C. was added slowly, dropwise, 5.2 mL, of liquid chlorine (1.367 g/mL). After the addition the mixture was allowed to warm to room temperature, and was then poured into approximately 100 g of ice. The resultant sulfonyl chloride was extracted with methylene chloride, washed with water and the methylene chloride solution added to 45 mL of concentrated aqueous ammonium hydroxide while maintaining the reaction temperature below 25° C. with ice bath cooling. Evaporation of the methylene chloride yielded a solid product which was removed by filtration from the aqueous residue and washed with water. The product, 3.72 g, melted at 176°-179° C. and showed absorption peaks by infrared spectroscopy at 3210 and 3300 cm⁻¹, consistent for the desired sulfonamide.

EXAMPLE 6 5-(2-Aminosulfonyl-4-methylphenyl)-1-methyl-1H-tetrazole

To a mixture of 4.68 g of 5-(4-methyl-2-propylthiophenyl)-1-methyl-1H-tetrazole, 40 mL of propionic acid and 1.08 g of water cooled to -10° C. was added dropwise 5.2 mL (liquified) of chlorine while maintaining the reaction temperature at -10° to 0° C. After one-half hour the reaction mixture was allowed to warm to room temperature and stirred for one hour. It was then poured into 200 mL of ice and water and extracted with methylene chloride. The methylene chloride solution was added to 45 mL of concentrated ammonium hydroxide at 10° C. and stirred overnight. The mixture was concentrated in vacuo to an oil residue which was taken up in 100 mL of methylene chloride washed with three 100 mL portions of water and 100 mL of saturated aqueous sodium hydroxide. The methylene chloride solution was then dried over magnesium sulfate, filtered, and the filtrate evaporated to yield 4.1 g of the desired product melting at 161°-171° C.

NMR (CDCl₃): δ2.56 (s, CH₃ on phenyl); 3.99 (s, CH₃ on tetrazole); 5.6 (s, w, NH₂); and 7.3-8.1 (m, 3CH on phenyl).

EXAMPLE 7 5-(2-Aminosulfonyl-3-methylphenyl)-1-methyl-1H-tetrazole

To a mixture of 14.6 mL of concentrated (12M) hydrochloric acid, 6.1 mL of acetic acid, 25 mL of ethyl ether and 6.91 g of 5-(2-amino-3-methylphenyl)-1-methyl-1H-tetrazole at 0° C. was added dropwise 2.8 g of sodium nitrite dissolved in 12.2 mL of water while maintaining the reaction temperature at below 10° C. Stirring was continued for one hour after the addition was completed. This mixture was then added slowly too 30.5 mL of acetic acid containing 0.6 g of cupric chloride and 6.1 mL of liquified sulfur dioxide. After stirring for two hours at ambient temperature, the mixture was poured into 200 mL of ice-water and extracted twice with 125 mL of methylene chloride. The organic phase was then washed twice with 200 ml of water, once with 200 mL saturated aqueous sodium chloride, once with 200 mL aqueous sodium bicarbonate followed by 200 mL of water and 200 mL saturated aqueous sodium chloride. The organic phase was then added dropwise to 25 mL of concentrated aqueous ammonium hydroxide and the mixture stirred overnight and evaporated to a solid, which was washed with water and dried. The crude product thus obtained melted at 140°-161° C., yield 6.26 g. Mass spectral analysis showed a molecular weight of 253 (calc. 253) for the product.

EXAMPLE 8 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(2-methyl-2H-tetrazol-5-yl)benzenesulfonamide

To 25 mL of acetonitrile was added at ambient temperature and pressure 0.48 g of 5-(2-aminosulfonylphenyl)-2-methyl-2H-tetrazole and 0.54 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate followed by 0.3 mL of DBU. After being stirred for three hours the reaction mixture was added to 25 g of ice and acidified to pH 3 with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried to yield 0.66 g of the desired product, m.p. 214°-222° C. Infrared absorptions at 1720, 1600 and 1580 cm⁻¹ were consistent with the desired structure.

NMR(CDCl₃): δ3.91 (s, 2XCH₃ O) 5.82 (s, CH, pyrimidin) 4.43 (s, CH₃ on N-2 of tetrazole) 4.38 (s, CH₃ on N-1 of tetrazole).

Integration of the peaks at 4.43 d and 4.38 d total one CH₃ indicating a ratio of 2-methyl-2H-tetrazole to 1-methyl-1H-tetrazole of 2:1. This mixture is suitable for purposes of this invention. If desired, the isomer mixture obtained in Example 6 can be separated by chromatography into its component parts.

EXAMPLE 9 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide

To 0.48 g of 1-(2-aminosulfonylphenyl)-5-methyl 1H-tetrazole in 25 mL of acetonitrile was added at ambient temperature and pressure 0.54 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate and 0.3 mL of DBU. The reaction mixture was stirred for three hours, added to 25 g of ice and acidified to pH 3 with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried to yield 0.74 g of the desired product, melting point at 213°-216° C. Infrared absorption spectra showed peaks at 1710, 1605 and 1570 cm⁻¹, consistent for the desired product.

NMR(CDCl₃): δ2.48 (s, CH₃ on tetrazole) 3.82 (s, 2XCH₃ O) 5.81 (s, CH-pyrimidin).

EXAMPLE 10 N-[(4-Methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide

To 0.48 g of 1-(2-aminosulfonylphenyl)-5-methyl-1H-tetrazole and 0.52 g of phenyl N-(4-methoxy-6-methyl-1,3,5-triazin-2-yl)carbamate in 25 mL of acetonitrile at ambient temperature and pressure was added 0.3 mL of DBU. The mixture was stirred for three hours and then added to 25 g of ice and acidified with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried in vacuo to yield 0.65 g of the desired product melting at 207°-209° C. Infrared absorption spectra showed absorption at 1700, 1600 and 1550 cm⁻¹, consistent for the desired structure.

EXAMPLE 11 N-[(4-Chloro-6-methoxypyrimidine-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide

To 0.48 g of 5-(2-aminosulfonylphenyl)-1-methyl-1H-tetrazole and 0.56 g of phenyl N-(4-chloro-6-methoxypyrimidine-2-yl)carbamate in 20 mL of dry acetonitrile at ambient temperature was added, with stirring, 0.3 mL of DBU. After stirring 16 hours the mixture was then poured into 25 g of ice followed by the addition of 10 mL of 2N hydrochloric acid. The precipitate thus formed was removed by filtration, washed with water and dried to yield 0.74 g of the desired product, m.p. 225°-227° C.

NMR (CDCl₃): δ3.88 (s, CH₃ on tetrazole); 3.95 (s, CH₃ O); 6.52 (s, CH of pyrimidine); 7.2-7.5 (m, CH of phenyl and NH); 7.84 (m, 2CH of phenyl); 8.6 (m, CH of phenyl); and 11.96 (s, NH).

EXAMPLE 12 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-5-chloro-2-(4-methyl-5-oxo-1H,4H-tetrazol-5-yl)benzenesulfonamide

To a stirred solution of 0.29 g of 1-(2-aminosulfonyl-5-chlorophenyl)-4-methyl-1H-tetrazol-5[4H]-one and 0.27 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate in 10 mL of acetonitrile at ambient temperature was added 0.1 mL of DBU. The mixture was stirred for two hours, poured into 20 g of ice and acidified with 2N hydrochloric acid. The precipitate was removed by filtration, washed with water and dried to yield 0.37 g of product, m.p. 178°-180° C.

NMR (CDCl₃): δ3.63 (s, CH₃ on tetrazole); 3.92 (s, 2XCH₃ O); 5.81 (s, CH of pyrimidine); 7.4-8.6 (m, 3CH of phenyl); and 12.6 (s, w, NH).

EXAMPLE 13 3-(2-Methyl-2H-tetrazole-5-yl)-1-phenyl-1H-pyrazole-5-sulfonamide

To a mixture of 3.1 mL of 12N hydrochloric acid, 12.5 mL of acetic acid, 3.7 mL of formic acid and 4.5 g of 5-amino-1-phenyl-3-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole was added dropwise 1.4 g of sodium nitrite in 2.5 mL of water at -8° to -6° C. The mixture was stirred for 15 minutes and then added to 20 mL of acetic acid containing 3.7 mL (liquid) of sulfur dioxide and 0.75 g of cupric chloride dihydrate. After stirring for thirty minutes and allowing to warm to room temperature, the mixture was poured into an ice and water mixture and the precipitate removed by filtration. After washing with water the solid was dissolved in tetrahydrofuran, cooled to -78° C., and ammonia (liquified, 1.0 mL) was added dropwise. The mixture was allowed to stand overnight at ambient temperature and filtered to yield a brown solid. This solid showed peaks at 3300 and 3200 cm⁻¹, consistent for NH₂, and 1370, 1185 and 1170 cm⁻¹, consistent for SO₂.

By using the procedures described in the foregoing equations and examples or modifications thereof, one skilled in the art can prepare the compounds shown in the following tables. ##STR35##

                                      TABLE I                                      __________________________________________________________________________     General Structure 1                                                            R.sub.1  E  Q   R.sub.3   W      R  X       Y         Z  m.p.                  __________________________________________________________________________                                                              (°C.)          H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 224-226               H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH 222-224               H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 207-210               H        -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 225-227               H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N  196-198               H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  172-187               H        -- Q-1 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               CH.sub.3  CH 200-207               H        -- Q-1 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 CH 203-205               H        -- Q-1 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 CH 214-217               H        -- Q-1 C.sub.2 H.sub. 5                                                                         O      H  Cl      OCH.sub.3 CH 223-225               H        -- Q-1 C.sub.2 H.sub.5                                                                          O      H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                               N  193-200               H        -- Q-1 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 N  192-196               H        -- Q-1 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 N  192-195               H        -- Q-1 CH(CH.sub.3).sub.2                                                                       O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 CH(CH.sub.3).sub.2                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 CH(CH.sub.3).sub.2                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH(CH.sub.3).sub.2                                                                       O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 CH(CH.sub.3).sub.2                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 CH(CH.sub.3).sub.2                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub.4 CH.sub.3                                                                O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 (CH.sub.2).sub.4 CH.sub.3                                                                O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 (CH.sub. 2).sub.4 CH.sub.3                                                               O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.4 CH.sub.3                                                                O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.4 CH.sub.3                                                                O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub.4 CH.sub.3                                                                O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 cyclopentyl                                                                              O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 cyclopentyl                                                                              O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 cyclopentyl                                                                              O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 cyclopentyl                                                                              O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 cyclopentyl                                                                              O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 cyclopentyl                                                                              O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.2 Cl                                                                              O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 CH.sub.2 Cl                                                                              O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 Cl                                                                              O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 Cl                                                                              O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 Cl                                                                              O      H  CH.sub.3                                                                               OCH.sub. 3                                                                               N                        H        -- Q-1 CH.sub.2 Cl                                                                              O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub.2 F                                                                       O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 (CH.sub.2).sub.2 F                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.2 F                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.2 F                                                                       O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.2 F                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub.2 F                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 --CH.sub.2 CH═CH.sub.2                                                               O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 --CH.sub.2 CH═CH.sub.2                                                               O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 --CH.sub.2 CH═CH.sub.2                                                               O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 --CH.sub.2 CH═CH.sub.2                                                               O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 --CH.sub.2 CH═CH.sub.2                                                               O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 -- CH.sub.2 CH═CH.sub.2                                                              O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.2 CH═CHCH.sub.2 Cl                                                            O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 CH.sub.2 CH═CHCH.sub.2 Cl                                                            O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 CH═CHCH.sub.2 Cl                                                            O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 CH═CHCH.sub.2 Cl                                                            O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 CH═CHCH.sub.2 Cl                                                            O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 CH.sub.2 CH═CHCH.sub.2 Cl                                                            O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.2 --C.tbd.C--CH.sub.3                                                             O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 CH.sub.2 --C.tbd.C--CH.sub.3                                                             O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 --C.tbd.C--CH.sub.3                                                             O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 --C.tbd.C--CH.sub.3                                                             O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 --C.tbd.C--CH.sub.3                                                             O      H  CH.sub.3                                                                               OCH.sub. 3                                                                               N                        H        -- Q-1 CH.sub.2 --C.tbd.C--CH.sub.3                                                             O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 C.sub.6 H.sub.5                                                                          O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 C.sub.6 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 C.sub.6 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 C.sub.6 H.sub.5                                                                          O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 C.sub.6 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 C.sub.6 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub.4 OCH.sub.3                                                               O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 (CH.sub.2).sub.4 OCH.sub.3                                                               O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.4 OCH.sub.3                                                               O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.4 OCH.sub.3                                                               O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.4 OCH.sub.3                                                               O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub. 4 OCH.sub.3                                                              O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                      O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                      O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                      O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                      O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                      O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                      O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 235-238               5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH 233-234               5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 213-216               5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 217-219               5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N  200-205               5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  195-198               3-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 192-197               3-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  201-206               3-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  N  159-173               3-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH 219-222               3-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 223-226               3-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 181-186               3-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OC.sub.2                                                                               H.sub.5 NHCH.sub.3                                                                       N  187-190               4-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  N  179-186               4-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 214-218               4-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH 225-229               4-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  191-196               4-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 182-196               4-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 140-150               4-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                               N  152-160               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  197-200               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  N  198-202               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 178-180               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH 180-183               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 213-215               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 196-199               5-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 221-223               5-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH 207-210               5-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 214-216               5-Cl     -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 203-205               5-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N  191-193               5-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  175-180               5-Cl     -- Q-1 CH.sub.3  O      H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                               N  144-158               5-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH(OCH.sub.3).sub.2                                                                      CH 180-183               5-Br     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-Br     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-Br     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-Br     -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-Br     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-Br     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-OCF.sub.2 H                                                                           -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-OCF.sub.2 H                                                                           -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-OCF.sub.2 H                                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-OCF.sub.2 H                                                                           -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-OCF.sub.2 H                                                                           -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-OCF.sub.2 H                                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 198-200               5-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH 218-219               5-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 205-207               5-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 185-188               5-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-CF.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-CF.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-CF.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CF.sub.3                                                                              -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-CF.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-CF.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        6-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 159-164               6-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH 196-199               6-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 153-156               6-Cl     -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 166-170               6-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N  187-189               6-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  202-205               6-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 181-186               6-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH 205-209               6-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 174-181               5-SCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-SCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-SCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-SCH.sub.3                                                                             -- Q-1 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-SCH.sub.3                                                                             -- Q-1 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-1 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-1 C.sub.2 H.sub.5                                                                          O      H  Cl      OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-1 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-SCH.sub.3                                                                             -- Q-1 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      CH.sub.3                                                                          OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      CH.sub.3                                                                          Cl      OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 CH.sub.3  O      CH.sub.3                                                                          OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.3  S      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 CH.sub.3  S      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  S      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  S      H  Cl      OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  S      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-1 CH.sub.3  S      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.3  O      H  H       OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      H  H       OC.sub.2 H.sub.5                                                                         CH                       H        -- Q-1 CH.sub.3  O      H  H       OCF.sub.2 H                                                                              CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CF.sub.3  CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               SCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                       CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.2 OCH.sub.3                                                                      CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               NHCH.sub.3                                                                               CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               N(CH.sub.3).sub.2                                                                        CH                       H        CH.sub.2                                                                          Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        CH.sub.2                                                                          Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        CH.sub.2                                                                          Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        CH.sub.2                                                                          Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       H        CH.sub.2                                                                          Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        CH.sub.2                                                                          Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        O  Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        O  Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        O  Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        O  Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        O  Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        O  Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        O  Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        O  Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       H        O  Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        O  Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.3  O      H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                               CH                       H        -- Q-1 CH.sub.3  O      H  H       OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      H  H       OC.sub.2 H.sub.5                                                                         CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CF.sub.3  CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               SCH.sub.3 CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                       CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               NHCH.sub.3                                                                               CH                       H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               N(CH.sub.3).sub.2                                                                        CH                       H        -- Q-1 CH.sub.3  O      H  H       OCH.sub.3 N                        H        -- Q-1 CH.sub.3  O      H  H       OC.sub.2 H.sub.5                                                                         N                        H        -- Q-1 CH.sub.3  O      H  H       OCF.sub.2 H                                                                              N                        H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                       N                        H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               NHCH.sub.3                                                                               N                        H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               N(CH.sub.3).sub.2                                                                        N                        3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub.2 CH.sub.2 Cl                                                                  -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub.2 CH.sub.2 Cl                                                                  -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-SO.sub.2 N(CH.sub.3).sub.2                                                            -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       6-SO.sub.2 N(CH.sub.3).sub.2                                                            -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       6-SCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       6-SCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-SOCH.sub.3                                                                            -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       6-SOCH.sub.3                                                                            -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-SO.sub.2 CH.sub.3                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-SO.sub.2 CH.sub.3                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CN     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CN     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CO.sub.2 CH.sub.3                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CO.sub.2 CH.sub.3                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-OCH.sub.2 CH.sub.2 Cl                                                                 -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-OCH.sub.2 CH.sub.2 Cl                                                                 -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-OCH.sub.2 CF.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-OCH.sub.2 CF.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-SCH.sub.2 CF.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-SCH.sub.2 CF.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-NH.sub.2                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-NH.sub.2                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-NHC.sub.2 H.sub.5                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-NHC.sub.2 H.sub.5                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-N(CH.sub.3).sub.2                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-N(CH.sub.3).sub.2                                                                     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub.2 OCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-C.sub.2 H.sub.4 OCH.sub.3                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-C.sub.2 H.sub.4 OCH.sub.3                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-C.sub.2 H.sub.4 OC.sub.2 H.sub.5                                                      -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-C.sub.2 H.sub.4 OC.sub.2 H.sub.5                                                      -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CH.sub.2 OC.sub.2 H.sub.4 Cl                                                          -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CH.sub.2 OC.sub.2 H.sub.4 Cl                                                          -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub. 2 OCH.sub.2 CF.sub.3                                                          -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub.2 OCH.sub.2 CF.sub.3                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CH.sub.2 SCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CH.sub.2 SCH.sub.3                                                                    -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub.2 SC.sub.2 H.sub.4 Cl                                                          -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       5-CH.sub.2 SC.sub.2 H.sub.4 Cl                                                          -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CH.sub.2 CN                                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-CH.sub.2 CN                                                                           -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.2 CH.sub.2 CH.sub.2                                                    CH.sub.3  CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.2 CH.sub.2 Cl                                                                    CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.2 CH.sub.2 CH.sub.2                                                    Cl        CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              SCH.sub.2 CH.sub.2 Cl                                                                    CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              SCHF.sub.2                                                                               CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              SCH.sub.2 CH.sub.3                                                                       CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                       CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              C.sub.2 H.sub.4 OC.sub.2                                                       H.sub.5   CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OC.sub.2 H.sub.4 OC.sub.2                                                      H.sub.5   CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.2 CH═CH.sub.2                                                                CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.2 C.tbd.CH                                                                       CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.2 SCH.sub.3                                                                       CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              C.sub.2 H.sub.4 SCH.sub.3                                                                CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              C.sub.2 H.sub.4 SC.sub.2                                                       H.sub.5   CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.2 SO.sub.2 CH.sub.3                                                               CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              C.sub.2 H.sub.4 SO.sub.2                                                       CH.sub.3  CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              C.sub.2 H.sub.4 SOCH.sub.3                                                               CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.2 CH.sub.2 CH.sub.2                                                               CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.2 C.tbd.CH                                                                        CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              N.sub.3   CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CN        CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              COCH.sub.3                                                                               CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              C(CH.sub.3)(OCH.sub.3).sub.2                                                             CH                       H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              2-methyldi-                                                                              CH                                                                   oxolan-2-yl                        H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              N(OCH.sub.3)CH.sub.3                                                                     CH                       H        -- Q-1 CH.sub.3  O      H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                               N  204-208               H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub. 3                                                                               CH 214-222               H        -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-2 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          O      H  Cl      OCH.sub.3 CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-2 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-2 CH(CH.sub.3).sub.2                                                                       O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 CH(CH.sub.3).sub.2                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 CH(CH.sub.3).sub.2                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-2 CH(CH.sub.3).sub.2                                                                       O      H  Cl      OCH.sub.3 CH                       H        -- Q-2 CH(CH.sub.3).sub.2                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-2 CH(CH.sub.3).sub.2                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-2 (CH.sub.2).sub.2 CH.sub.3                                                                O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 (CH.sub.2).sub.2 CH.sub.3                                                                O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 (CH.sub.2).sub.2 CH.sub.3                                                                O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-2 (CH.sub.2).sub.2 CH.sub.3                                                                O      H  Cl      OCH.sub.3 CH                       H        -- Q-2 (CH.sub.2).sub.2 CH.sub.3                                                                O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-2 (CH.sub.2).sub.2 CH.sub.3                                                                O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.2 C.tbd.CH                                                                        O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-1 CH.sub.2 C.tbd.CH                                                                        O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 C.tbd.CH                                                                        O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 C.tbd.CH                                                                        O      H  Cl      OCH.sub.3 CH                       H        -- Q-1 CH.sub.2 C.tbd.CH                                                                        O      H  CH.sub.3                                                                               OCH.sub. 3                                                                               N                        H        -- Q-1 CH.sub.2 C.tbd.CH                                                                        O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCF.sub.2 H                                                                              CH 160-165               H        -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCF.sub.2 H                                                                              CH 195-198               5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCF.sub.2 H                                                                              CH 168-172               5-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCF.sub.2 H                                                                              CH  90-93                H        -- Q-2 CH.sub.2 OCH.sub.3                                                                       O      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 CH.sub.2 OCH.sub.3                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 CH.sub.2 OCH.sub.3                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-2 CH.sub.2 OCH.sub.3                                                                       O      H  Cl      OCH.sub.3 CH                       H        -- Q-2 CH.sub.2 OCH.sub.3                                                                       O      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-2 CH.sub.2 OCH.sub.3                                                                       O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-OCF.sub.2 H                                                                           -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-OCF.sub.2 H                                                                           -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub. 3                                                                               CH                       5-OCF.sub.2 H                                                                           -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-OCF.sub.2 H                                                                           -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-OCF.sub.2 H                                                                           -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-OCF.sub.2 H                                                                           -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        6-Cl     -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       6-Cl     -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-Cl     -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       6-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       6-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  CH                       6-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-SCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-SCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        5-SCH.sub.3                                                                             -- Q-2 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               CH.sub.3  CH                       5-SCH.sub.3                                                                             -- Q-2 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-2 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-2 C.sub.2 H.sub.5                                                                          O      H  Cl      OCH.sub.3 CH                       5-SCH.sub.3                                                                             -- Q-2 C.sub.2 H.sub.5                                                                          O      H  CH.sub.3                                                                               OCH.sub.3 N                        5-SCH.sub.3                                                                             -- Q-2 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-2 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      CH.sub.3                                                                          OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      CH.sub.3                                                                          Cl      OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-2 CH.sub.3  O      CH.sub.3                                                                          OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-2 CH.sub.3  S      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 CH.sub.3  S      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  S      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  S      H  Cl      OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  S      H  CH.sub.3                                                                               OCH.sub.3 N                        H        -- Q-2 CH.sub.3  S      H  OCH.sub.3                                                                              OCH.sub.3 N                        H        -- Q-2 CH.sub.3  O      H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                               N                        H        -- Q-2 CH.sub.3  O      H  H       OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      H  H       OC.sub.2 H.sub.5                                                                         CH                       H        -- Q-2 CH.sub.3  O      H  H       OCF.sub.2 H                                                                              CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               SCF.sub.2 H                                                                              CH                       H        -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                       CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.2 OCH.sub.3                                                                      CH                       H        -- Q-2 CH.sub.3  O      H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                               N                        H        -- Q-2 CH.sub.3  O      H  H       OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      H  H       OC.sub.2 H.sub.5                                                                         CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CF.sub.3  CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               SCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                       CH                       H        -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.2 OCH.sub.3                                                                      CH                       H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OC.sub.2 H.sub.5                                                                         N                        H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH(CH.sub.3).sub.2                                                                      N                        H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.2 CF.sub.3                                                                       N                        H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              CF.sub.3  N                        H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              O(CH.sub.2).sub.2 OCH.sub.3                                                              N                        H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              C.tbd.C-CH.sub.3                                                                         N                        H        -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              N(CH.sub.3)OCH.sub.3                                                                     N                        H        -- Q-2 C.sub.2 H.sub.5                                                                          S      H  CH.sub.3                                                                               CH.sub.3  CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          S      H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          S      H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          S      H  Cl      OCH.sub.3 CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          S      H  CH.sub.3                                                                               OCH.sub.3 N                        6-CH.sub.3                                                                              -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH                       6-CH.sub.3                                                                              -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH                       6-CH.sub. 3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH                       6-CH.sub.3                                                                              -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       6-CH.sub.3                                                                              -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.3  N                        6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  Br      OCH.sub.3 CH 196-198 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3 CH 199-200 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3 N   49-56                6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  H       CH.sub.3  CH 196-199 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  H       OCH.sub.3 CH 163-166 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  C.sub.2 H.sub.5                                                                        OCH.sub.3 CH 160-164               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  C.sub.2 H.sub.5                                                                        OCH.sub.3 N  179-180 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      CH.sub.3                                                                          OCH.sub.3                                                                              OCH.sub.3 N                        6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  cyclopropyl                                                                            OCH.sub.3 N  222-223 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OC.sub.2 H.sub.5                                                                         CH                       6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              CH.sub.2 OC.sub.2 H.sub.5                                                                CH 189-190 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.2 CF.sub.3                                                                       CH 140-145 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OC.sub.2 H.sub.5                                                                         N  159-164 dec.          6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCF.sub.2 H                                                                              CH 168-172               6-CH.sub.3                                                                              -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCF.sub.2 H                                                                              CH  90-93                H        -- Q-1 CH.sub.3  NH     H  OCH.sub.3                                                                              OCH.sub.3 CH                       H        -- Q-1 CH.sub.3  NOCH.sub.3                                                                            H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 CH.sub.3  NOH    H  CH.sub.3                                                                               OCH.sub.3 CH                       H        -- Q-2 C.sub.2 H.sub.5                                                                          NNHCH.sub.3                                                                           H  OCH.sub.3                                                                              OCH.sub.3 CH                       3-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  199-202               3-Cl     -- Q-1 CH.sub.3  O      H  CH.sub. 3                                                                              OCH.sub.3 N  206-209               3-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 143-162               3-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH 226-227               3-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 221-223 dec.          3-Cl     -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 189-192               5-F      -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 CH 209-212               5-F      -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 199-201               5-F      -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  187-190               5-F      -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N  196-201               5-F      -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               CH.sub.3  CH 233-236               5-F      -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 CH 164-168               H        -- Q-1 C.sub.2 H.sub.5                                                                          O      H  OCH.sub.3                                                                              OCF.sub.2 H                                                                              CH  87-94                6-Cl     -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCF.sub.2 H                                                                              CH  93-95                6-Cl     -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCF.sub.2 H                                                                              CH 118-120               6-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N  194-197               6-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N  172-182               6-OCH.sub.3                                                                             -- Q-1 CH.sub.3  O      H  Cl      OCH.sub.3 CH 206-209               6-Cl     -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       6-Cl     -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        6-Cl     -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        6-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  Cl      OCH.sub.3 CH                       6-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  OCH.sub.3                                                                              OCH.sub.3 N                        6-OCH.sub.3                                                                             -- Q-2 CH.sub.3  O      H  CH.sub.3                                                                               OCH.sub.3 N                        __________________________________________________________________________

                                      TABLE Ia                                     __________________________________________________________________________     General structure 1                                                            R.sub.1                                                                               E  Q  R.sub.4 W R  X      Y       Z  m.p.(°C.)                   __________________________________________________________________________     H      -- Q-3                                                                               H       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 214 dec.                           H      -- Q-3                                                                               H       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 204-205                            H      -- Q-3                                                                               H       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 187-188                            H      -- Q-3                                                                               H       O H  Cl     OCH.sub.3                                                                              CH 195-196                            H      -- Q-3                                                                               H       O H  CH.sub.3                                                                              OCH     N  199-202                            H      -- Q-3                                                                               H       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  191-192                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3                                                                             N  167-200 dec.                       H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 221-223                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 213-216                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH 208-210                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  207-209                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  209-216                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 217-220                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 224-228                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 193-196                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  Cl     OCH.sub.3                                                                              CH 200-204                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  174-179                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  194-197                            H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  CH.sub. 3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               cyclopropyl                                                                            O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               cyclopropyl                                                                            O H  OCH.sub.2                                                                             OCH.sub.2                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 195-196                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 175-177                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 188-189                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH 200-201                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  189-190                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  180                                H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 199-200 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 197-198 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 200-201 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH 184-185 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  170-173 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  178-180 dec.                       H      -- Q-3                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 177-186                            5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH 207-208                            5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  200-202                            5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 227-230                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 173-180                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 216-220                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH 227-230                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  188-195                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  192-194                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OC.sub.2 H.sub. 5                                                                     NHCH.sub.3                                                                             N  181-185                            5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              H                                     5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3 OCH.sub.3                                                                     O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     H      -- Q-3                                                                               CH.sub.3 OCH.sub.3                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               O H  cyclopropyl                                                                           OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             N.sub.3 CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CN      CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             C(O)CH.sub.3                                                                           CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH(OCH.sub.3).sub.2                                                                    CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             1,3-dioxo-                                                                             CH                                                                     lan-2-yl                                      H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             1,3-diox-                                                                              CH                                                                     an-2-yl                                       H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      O  Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      O  Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               S H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               S H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               S H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               S H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               S H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               S H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               O H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3                                                                             CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  H      OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  H      OC.sub.2 H.sub.5                                                                       CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  H      OCF.sub.2 H                                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              SCF.sub.2 H                                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                     CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OC.sub.2 H.sub.5                                                                       CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CF.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             O(CH.sub.2).sub.2 OCH.sub.3                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             SCF.sub.2 H                                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             C.tbd.CH                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             C.tbd.C--CH.sub.3                                                                      CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             N(OCH.sub.3)CH.sub.3                                                                   CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               SCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  OCH.sub.3                                                                             CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     H      -- Q-4                                                                               CF.sub.3                                                                               O H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3                                                                             N                                     H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               CH                                    6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 170-171                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 171-173                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  CH.sub. 3                                                                             CH.sub.3                                                                               CH 176-178                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  Cl     OCH.sub.3                                                                              CH 163-167                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  148-152                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  158-160                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 181-184                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 188-190                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 166-168                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH 182-184                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  184-186                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  175-178                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 180-181                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 188-191                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 198-199                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH 184-186                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  204-206                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  175-179                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 192-193                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 182-184                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 181-183                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH 172-175                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  167-170                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  174-176                            H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               OCF.sub. 2 H                                                                           O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub. 3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     __________________________________________________________________________

                                      TABLE 1b                                     __________________________________________________________________________     General structure 1                                                            R.sub.1                                                                              E Q  R.sub.5 W R X   Y    Z  m.p.(°C.)                            __________________________________________________________________________     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N  199-201                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 213-218                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           CH.sub.3                                                                            CH 185-189                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           OCH.sub.3                                                                           CH 201-206                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 191-209                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H Cl  OCH.sub.3                                                                           CH 196-199                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           OCH.sub.3                                                                           N  194-198                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H OCH.sub.3                                                                          OCH.sub.3                                                                           N  166-169                                     H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub. 5                                                                       O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N  202                                         H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 178-180                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH 134-140                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N  202                                         5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCF.sub.2 H                                                                         CH 196-198                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCF.sub.2 H                                                                         CH 162-166                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH 125-128                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N   70-112                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N  190-194                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 153-157                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH 170-173                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH 141-143                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              __________________________________________________________________________

                                      TABLE II                                     __________________________________________________________________________     General Structure 2                                                            R.sub.1                                                                             E Q  R.sub.3    W R X.sub.1                                                                             Y.sub.1                                                                           m.p.(°C.)                              __________________________________________________________________________     H    --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub. 5                                                                          O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCF.sub.2 H                                                                         CH.sub.2                                         H    --                                                                               Q-1                                                                               (CH.sub.2).sub.5 CH.sub.3                                                                 O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               CH.sub.2 CH═CH--CH.sub.2 Cl                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-CN --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CN --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-2                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-2                                                                               C.sub. 2 H.sub.5                                                                          O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-C.sub.2 H.sub.5                                                                   --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         __________________________________________________________________________

                  TABLE IIa                                                        ______________________________________                                         General Structure 2                                                            R.sub.1                                                                               E     Q      R.sub.4                                                                              W   R   X.sub.1                                                                               Y.sub.1                                                                             m.p.(°C.)                 ______________________________________                                         H      --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      O                                     H      --    Q-3    CH.sub.3                                                                             O   H   OCF.sub.2 H                                                                           O                                     H      --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub.5                                                                      O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCF.sub.2 H                                                                           CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     5-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              5-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-Cl   --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-OCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-OCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-OC.sub.2 H.sub.5                                                                    --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-OC.sub.2 H.sub.5                                                                    --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-SCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-SCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-SC.sub.2 H.sub.5                                                                    --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-SC.sub.2 H.sub. 5                                                                   --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-OCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-OCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-SCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-SCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     H      --    Q-4    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      O                                     H      --    Q-4    CH.sub.3                                                                             O   H   OCF.sub.2 H                                                                           O                                     H      --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-4    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-4    CH.sub.3                                                                             O   H   OCF.sub.2 H                                                                           CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub. 5                                                                     O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCF.sub.2 H                                                                           O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCF.sub.2 H                                                                           CH.sub.2                              6-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     6-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     6-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     6-Cl   --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     6-CH.sub.3                                                                            --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-CH.sub.3                                                                            --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     6-CH.sub.3                                                                            --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     6-Cl   --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-Cl   --    Q-4    CH.sub. 3                                                                            O   H   OCH.sub.3                                                                             O                                     6-Cl   --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-3    H     O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    H     O   H   CH.sub.3                                                                              O                                     H      --    Q-3    H     O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    H     O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    OCH.sub.3                                                                            O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    OCH.sub.3                                                                            O   H   CH.sub.3                                                                              O                                     H      --    Q-3    OCH.sub.3                                                                            O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    OCH.sub.3                                                                            O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   CH.sub.3                                                                              O                                     H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    SCH.sub.3                                                                            O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    SCH.sub.3                                                                            O   H   CH.sub.3                                                                              O                                     H      --    Q-3    SCH.sub.3                                                                            O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    SCH.sub.3                                                                            O   H   CH.sub.3                                                                              CH.sub.2                              ______________________________________                                    

                  TABLE IIb                                                        ______________________________________                                         General Structure 2                                                            R.sub.1 E     Q      R.sub.5                                                                             W   R   X.sub.1                                                                              Y.sub.1                                                                             m.p.(°C.)                  ______________________________________                                         H       --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      H       --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               H       --    Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      H       --    Q-5    C.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                            O                                      H       --    Q-5    C.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                            CH.sub.2                               H       --    Q-5    C.sub.2 H.sub.5                                                                     O   H   CH.sub.3                                                                             O                                      5-CH.sub.3                                                                             --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-CH.sub.3                                                                             --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-CH.sub.3                                                                             --    Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      5-Cl    --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-Cl    --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-Cl    --    Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      6-CH.sub.3                                                                             --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      6-CH.sub.3                                                                             --    Q-5    CH.sub.3                                                                            O   H   OCH.sub. 3                                                                           CH.sub.2                               6-CH.sub.3                                                                             --    Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      6-Cl    --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      6-Cl    --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               6-Cl    --    Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      5-F     --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-F     --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-F     --    Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      5-OCH.sub.3                                                                            --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-OCH.sub.3                                                                            --    Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-OCH.sub.3                                                                            --    Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      ______________________________________                                    

                  TABLE III                                                        ______________________________________                                         General Structure 3                                                            R.sub.1                                                                              E     Q      R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                             W   R   X.sub.1                                                                             m.p.(°C.)               ______________________________________                                         H     --    Q-1    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            H     --    Q-1    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           H     --    Q-1    CH.sub.3                                                                            --    --   O   H   OC.sub.2 H.sub.5                    H     --    Q-1    CH.sub.3                                                                            --    --   O   H   OCF.sub.2 H                         H     --    Q-1    C.sub.2 H.sub.5                                                                     --    --   O   H   CH.sub.3                            H     --    Q-1    C.sub.2 H.sub.5                                                                     --    --   O   H   OCH.sub.3                           H     --    Q-1    C.sub.2 H.sub.5                                                                     --    --   O   H   OC.sub.2 H.sub.5                    H     --    Q-2    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            H     --    Q-2    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           H     --    Q-2    CH.sub.3                                                                            --    --   O   H   OC.sub.2 H.sub.5                    H     --    Q-2    C.sub.2 H.sub.5                                                                     --    --   O   H   OCH.sub.3                           H     --    Q-2    C.sub.2 H.sub.5                                                                     --    --   O   H   CH.sub.3                            H     --    Q-3    --   CH.sub.3                                                                             --   O   H   OC.sub.2 H.sub.5                    H     --    Q-3    --   CH.sub.3                                                                             --   O   H   OCH.sub.3                           H     --    Q-3    --   CH.sub.3                                                                             --   O   H   CH.sub.3                            H     --    Q-3    --   C.sub.2 H.sub.5                                                                      --   O   H   CH.sub.3                            H     --    Q-3    --   C.sub.2 H.sub.5                                                                      --   O   H   OCH.sub.3                           6-CH.sub.3                                                                           --    Q-1    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           6-CH.sub.3                                                                           --    Q-1    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            6-Cl  --    Q-1    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            6-Cl  --    Q-1    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           H     --    Q-4    --   CH.sub.3                                                                             --   O   H   OCH.sub.3                           H     --    Q-5    --   --    CH.sub.3                                                                            O   H   OCH.sub.3                           H     --    Q-5    --   --    CH.sub. 3                                                                           O   H   CH.sub.3                            H     --    Q-6    --   --    CH.sub.3                                                                            O   H   OCH.sub.3                           H     --    Q-7    --   --    CH.sub.3                                                                            O   H   OCH.sub.3                           H     --    Q-3    --   H     --   O   H   OCH.sub.3                           H     --    Q-3    --   H     --   O   H   CH.sub.3                            H     --    Q-3    --   OCH.sub.3                                                                            --   O   H   OCH.sub.3                           H     --    Q-3    --   OCH.sub.3                                                                            --   O   H   CH.sub.3                            H     --    Q-3    --   OC.sub.2 H.sub.5                                                                     --   O   H   OCH.sub.3                           H     --    Q-3    --   OC.sub.2 H.sub.5                                                                     --   O   H   CH.sub.3                            H     --    Q-3    --   SCH.sub.3                                                                            --   O   H   OCH.sub.3                           H     --    Q-3    --   SCH.sub.3                                                                            --   O   H   CH.sub.3                            ______________________________________                                    

                                      TABLE IV                                     __________________________________________________________________________     General Structure 4                                                            R.sub.1                                                                             E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X.sub.1                                                                            Y.sub.3                                                                           m.p.(°C.)                                __________________________________________________________________________     H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           H                                                  H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                   H                                                  H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCF.sub.2 H                                                                        CH.sub.3                                           H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           H                                                  H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                           H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                           H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           H                                                  H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                           H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          CH.sub.3                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          CH.sub.3                                           H    --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                           H    --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                           H    --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           H                                                  5-Cl --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           H                                                  6-CH.sub.3                                                                          --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-3                                                                               -- H   -- O H CH.sub.3                                                                           H                                                  H    --                                                                               Q-3                                                                               -- H   -- O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                           H    --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          CH.sub.3                                           H    --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                           H                                                  H    --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                                                          H                                                  H    --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                           H    --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H OCH.sub.3                                                                          CH.sub.3                                           __________________________________________________________________________

                                      TABLE V                                      __________________________________________________________________________     General Structure 5                                                            R.sub.1                                                                            E Q  R.sub.3                                                                              R.sub.4                                                                            R.sub.5                                                                           W R X.sub.2                                                                             Y.sub.2                                                                            m.p.(°C.)                            __________________________________________________________________________     H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.2 CF.sub.3                                                                   OCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SC.sub.2 H.sub.5                                H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                      --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                      --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-2                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-2                                                                               CH(CH.sub.3).sub.2                                                                   --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SC.sub.2 H.sub.5                                H   --                                                                               Q-3                                                                               --    C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CF.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       6-CH.sub.3                                                                         --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       6-Cl                                                                               --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-5                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-6                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-7                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       6-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       5-Cl                                                                               --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    H   -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    H   -- O H C.sub.2 H.sub.5                                                                     OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    OCH.sub.3                                                                          -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    OCH.sub.3                                                                          -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                H   --                                                                               Q-3                                                                               --    SCH.sub.3                                                                          -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    SCH.sub.3                                                                          -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                __________________________________________________________________________

                  TABLE VI                                                         ______________________________________                                         General Structure 6                                                                                                            m.p.                           R.sub.1                                                                              E     Q      R.sub.3                                                                             R.sub.4 R.sub.5                                                                             W   RX.sub.3                                                                              (°C.)                   ______________________________________                                         H     --    Q-1    CH.sub.3                                                                            --      --   O   H CH.sub.3                            H     --    Q-1    CH.sub.3                                                                            --      --   O   H OCH.sub.3                           H     --    Q-1    C.sub.2 H.sub.5                                                                     --      --   O   H CH.sub.3                            H     --    Q-1    C.sub.2 H.sub.5                                                                     --      --   O   H OCH.sub.3                           H     --    Q-2    CH.sub.3                                                                            --      --   O   H CH.sub.3                            H     --    Q-2    C.sub.2 H.sub.5                                                                     --      --   O   H CH.sub.3                            H     --    Q-3    --   CH.sub.3                                                                               --   O   H CH.sub.3                            H     --    Q-3    --   CH.sub.3                                                                               --   O   H OCH.sub.3                           H     --    Q-3    --   C.sub.2 H.sub.5                                                                        --   O   H CH.sub.3                            H     --    Q-3    --   C.sub.2 H.sub.5                                                                        --   O   H  OCH.sub.3                          H     --    Q-3    --   CH(CH.sub.3).sub.2                                                                     --   O   H OCH.sub.3                           H     --    Q-3    --   CH.sub.2 Cl                                                                            --   O   H OCH.sub.3                           H     --    Q-3    --   CF.sub.3                                                                               --   O   H OCH.sub.3                           H     --    Q-4    --   CH.sub.3                                                                               --   O   H OCH.sub.3                           6-CH.sub.3                                                                           --    Q-1    CH.sub.3                                                                            --      --   O   H OCH.sub.3                           6-Cl  --    Q-1    CH.sub.3                                                                            --      --   O   H OCH.sub.3                           5-Cl  --    Q-1    CH.sub.3                                                                            --      --   O   H OCH.sub.3                           H     --    Q-5    --   --      CH.sub.3                                                                            O   H OCH.sub.3                           H     --    Q-5    --   --      CH.sub.3                                                                            O   H CH.sub.3                            H     --    Q-6    --   --      CH.sub.3                                                                            O   H OCH.sub.3                           H     --    Q-6    --   --      CH.sub.3                                                                            O   H CH.sub.3                            H     --    Q-7    --   --      CH.sub.3                                                                            O   H OCH.sub.3                           H     --    Q-3    --   H       --   O   H CH.sub.3                            H     --    Q-3    --   H       --   O   H OCH.sub.3                           H     --    Q-3    --   OCH.sub.3                                                                              --   O   H CH.sub.3                            H     --    Q-3    --   OCH.sub.3                                                                              --   O   H OCH.sub.3                           H     --    Q-3    --   OC.sub.2 H.sub.5                                                                       --   O   H CH.sub.3                            H     --    Q-3    --   OC.sub.2 H.sub.5                                                                       --   O   H OCH.sub.3                           H     --    Q-3    --   SCH.sub.3                                                                              --   O   H CH.sub.3                            H     --    Q-3    --   SCH.sub.3                                                                              --   O   H OCH.sub.3                           ______________________________________                                    

                                      TABLE VII                                    __________________________________________________________________________     General Structure 7                                                            R.sub.1                                                                             E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X.sub.4                                                                              Y.sub.4                                                                            Z.sup.1                                                                           m.p. (°C.)                         __________________________________________________________________________     H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub. 3                                                                         --  -- O H CH.sub.2 OCH.sub.3                                                                   OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OC.sub.2 H.sub.5                                                                   CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            Cl  CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OC.sub.2 H.sub.5                                                                   CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             Cl  CH                                           6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub. 3                                                                          CH                                           5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           6-CH.sub.3                                                                          --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           6-CH.sub.3                                                                          --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            5-Cl --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           5-Cl --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           5-OCH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           5-OCH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           5-OCH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           H    --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-6                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-7                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          N                                            H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub. 3                                                                           CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- H   -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- H   -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                            H    --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            H    --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                            H    --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            __________________________________________________________________________

                                      TABLE VIII                                   __________________________________________________________________________     General Structure 8                                                            R.sub.1                                                                            n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W    R  X   Y    Z  m.p. (°C.)                   __________________________________________________________________________     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  Cl  OCH.sub. 3                                                                          CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub. 3                                                                         CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub. 3                                                                          CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N                                      H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N                                      H   0 --                                                                               Q-3                                                                               -- H     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            N                                      H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3 ).sub.2                                                                   -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub. 3                                                                          N                                      H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub. 3                                                                          N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub. 3                                                                          CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    CH.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- NCH.sub.3                                                                           H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- NOCH.sub.3                                                                          H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    CH.sub.3                                                                          CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     __________________________________________________________________________

                                      TABLE IX                                     __________________________________________________________________________     General structure 9                                                            R.sub.1 n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W  R  X   Y   Z  m.p. (°C.)                  __________________________________________________________________________     H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           N                                     H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub. 3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- H  OCH.sub.3                                                                         OCH.sub.3                                                                          CH                                        4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- S  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- S  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  CH.sub.3                                                                          Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          NH H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       1 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    __________________________________________________________________________

                                      TABLE X                                      __________________________________________________________________________     General Structure 10                                                           R.sub.1                                                                           n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W     R  X   Y   Z  m.p. (°C.)                    __________________________________________________________________________     H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub. 3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub. 3                                                                           -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- S     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     CH.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- NNHCH.sub.3                                                                          H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  1 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      __________________________________________________________________________

                                      TABLE XI                                     __________________________________________________________________________     General Structure 11                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p.(°C.)                __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub. 3                                                                         CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub. 5                                                                    --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub. 3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub. 3                                                                         CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  __________________________________________________________________________

                                      TABLE XII                                    __________________________________________________________________________     General Structure 12                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y    Z  m.p. (°C.)              __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub. 5                                                                    C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 232-233                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH 193-195                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 195-198                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub. 3                                                                           CH 165-170                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N  140-145                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  195-196                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 165-167                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH 125-127                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 189-191                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N  166-170                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  160-172                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  180-183                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 171-173                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH 181-183                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 178-180                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 200-202                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N  179-180                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 195                            H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 172-173                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH 152-156                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH 170-171                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N  173-174                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  168-170                        H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub. 3                                                                           --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                          N                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub. 3                                                                         CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 213-216                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH 186-189                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 207-208                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 170-173                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N  186-191                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N  141-144                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  191-193                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N  179-183                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 165-167                        __________________________________________________________________________

                                      TABLE XIII                                   __________________________________________________________________________     General Structure 13                                                                                                          m.p.                            R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  (°C.)                    __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub. 6 H.sub.5                                                                    --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub. 3                                                                         N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH  OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub. 2 CH.sub.3                                                                  --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub. 3                                                                           CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub. 3                                                                           CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub. 3                                                                           CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub. 3                                                                         CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub. 3                                                                           CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub. 3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  __________________________________________________________________________

                  TABLE XIV                                                        ______________________________________                                         General Structure 14                                                                                                               m.p.                       R.sub.1                                                                            n     E     Q    R.sub.3                                                                             R.sub.4                                                                            W R  X     Y     Z    (°C.)               ______________________________________                                         H   0     --    Q-1  CH.sub.3                                                                            --  O H  CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0     --    Q-1  CH.sub.3                                                                            --  O H  OCH.sub.3                                                                            CH.sub.3                                                                             CH                              H   0     --    Q-1  CH.sub.3                                                                            --  O H  Cl    OCH.sub.3                                                                            CH                              H   0     --    Q-1  CH.sub.3                                                                            --  O H  CH.sub.3                                                                             OCH.sub.3                                                                            N                               H   0     --    Q-1  CH.sub.3                                                                            --  O H  OCH.sub.3                                                                            OCH.sub.3                                                                            N                               H   0     --    Q-1  C.sub.2 H.sub.5                                                                     --  O H  OCH.sub.3                                                                            CH.sub.3                                                                             CH                              H   0     --    Q-1  C.sub.2 H.sub.5                                                                     --  O H  OCH.sub.3                                                                            OCH.sub.3                                                                            CH                              H   0     --    Q-1  C.sub.2 H.sub.5                                                                     --  O H  Cl    OCH.sub.3                                                                            CH                              H   0     --    Q-1  C.sub.2 H.sub.5                                                                     --  O H  CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0     --    Q-1  C.sub.2 H.sub.5                                                                     --  O H  CH.sub.3                                                                             OCH.sub.3                                                                            N                               H   0     --    Q-2  CH.sub.3                                                                            --  O H  OCH.sub.3                                                                            OCH.sub.3                                                                            N                               H   0     --    Q-2  CH.sub.3                                                                            --  O H  OCH.sub.3                                                                            OCH.sub.3                                                                            CH                              H   0     --    Q-2  CH.sub.3                                                                            --  O H  OCH.sub.3                                                                            CH.sub.3                                                                             CH                              H   0     --    Q-2  CH.sub.3                                                                            --  O H  Cl    OCH.sub.3                                                                            CH                              H   0     --    Q-2  CH.sub.3                                                                            --  O H  CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0     --    Q-2  CH.sub.3                                                                            --  O H  OCH.sub.3                                                                            CH.sub.3                                                                             N                               H   0     --    Q-2  C.sub.2 H.sub.5                                                                     --  O H  OCH.sub.3                                                                            OCH.sub.3                                                                            N                               H   0     --    Q-2  C.sub.2 H.sub.5                                                                     --  O H  CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0     --    Q-2  C.sub.2 H.sub.5                                                                     --  O H  CH.sub.3                                                                             OCH.sub.3                                                                            CH                              H   0     --    Q-2  C.sub.2 H.sub.5                                                                     --  O H  Cl    OCH.sub.3                                                                            CH                              H   0     --    Q-2  C.sub.2 H.sub.5                                                                     --  O H  CH.sub.3                                                                             OCH.sub.3                                                                            N                               H   0     --    Q-2  C.sub.2 H.sub.5                                                                     --  O H  OCH.sub.3                                                                            OCH.sub.3                                                                            N                               ______________________________________                                    

                                      TABLE XV                                     __________________________________________________________________________     General Structure 15                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                          __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH 138-143                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH 155-159                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H Cl  OCH.sub.3                                                                          CH 157-158                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH 135-140                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                             H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N   75-78                                     H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                             H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                             H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- H     -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- H     -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- H     -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- H     -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- H     -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- H     -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                            H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H Cl  OCH.sub.3                                                                          CH                                            H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                             __________________________________________________________________________

                                      TABLE XVI                                    __________________________________________________________________________     General Structure 16                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                            __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub. 3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               __________________________________________________________________________

                                      TABLE XVII                                   __________________________________________________________________________     General Structure 17                                                           R.sub.1                                                                            E Q  G  n R.sub.3                                                                           W R X   Y   Z  m.p. (°C.)                              __________________________________________________________________________     H   --                                                                               Q-1                                                                               O  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               S  0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO 0 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO 1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               SO 2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               O  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               S  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               SO 2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 6-CH.sub.3                                                                         --                                                                               Q-1                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 5-Cl                                                                               --                                                                               Q-1                                                                               O  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                5-Cl                                                                               --                                                                               Q-1                                                                               S  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                5-Cl                                                                               --                                                                               Q-1                                                                               SO 1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 5-Cl                                                                               --                                                                               Q-1                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               S  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub. 3                                                                         N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                H   --                                                                               Q-2                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           N                                                 H   --                                                                               Q-2                                                                               SO 2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 __________________________________________________________________________

                                      TABLE XVIIa                                  __________________________________________________________________________     General Structure 17                                                           R.sub.2                                                                           E  Q  G  n R.sub.4                                                                           W R X   Y   Z  m.p. (°C.)                              __________________________________________________________________________     H  -- Q-3                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H  -- Q-3                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H  -- Q-3                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H  -- Q-3                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H  -- Q-3                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H  -- Q-3                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H  -- Q-3                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H  -- Q-3                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H  -- Q-4                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H  -- Q-4                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H  -- Q-4                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H  -- Q-4                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H  -- Q-4                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H  -- Q-4                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H  -- Q-4                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H  -- Q-4                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 __________________________________________________________________________

                                      TABLE XVIIb                                  __________________________________________________________________________     General Structure 17                                                           R.sub.1                                                                           E  Q  G  n  R.sub.5                                                                           W  R  X   Y   Z  m.p. (°C.)                           __________________________________________________________________________     H  -- Q-5                                                                               O  1  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H  -- Q-5                                                                               S  1  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              H  -- Q-5                                                                               SO 1  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              H  -- Q-5                                                                               SO.sub.2                                                                          1  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             H  -- Q-5                                                                               O  2  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              H  -- Q-5                                                                               S  2  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             H  -- Q-5                                                                               SO 2  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H  -- Q-5                                                                               SO.sub.2                                                                          2  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              H  -- Q-6                                                                               O  1  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              H  -- Q-6                                                                               S  1  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             H  -- Q-6                                                                               SO 1  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H  -- Q-6                                                                               SO.sub.2                                                                          1  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              H  -- Q-6                                                                               O  2  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H  -- Q-6                                                                               S  2  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              H  -- Q-6                                                                               SO 2  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              H  -- Q-6                                                                               SO.sub.2                                                                          2  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             H  -- Q-7                                                                               O  1  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H  -- Q-7                                                                               S  1  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              H  -- Q-7                                                                               SO 1  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              H  -- Q-7                                                                               SO.sub.2                                                                          1  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             H  -- Q-7                                                                               O  2  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H  -- Q-7                                                                               S  2  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              H  -- Q-7                                                                               SO 2  CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              H  -- Q-7                                                                               SO.sub. 2                                                                         2  CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             __________________________________________________________________________

                                      TABLE XVIII                                  __________________________________________________________________________     General Structure 18                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (°C.)               __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C H.sub.5                                                                           C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub. 2 Cl                                                                         -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3 ).sub.2                                                                  -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub. 2 Cl                                                                         -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub. 3                                                                         O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  __________________________________________________________________________

                                      TABLE XIX                                    __________________________________________________________________________     General Structure 19                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                            __________________________________________________________________________     H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               __________________________________________________________________________

                                      TABLE XX                                     __________________________________________________________________________     General Structure 19                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                            __________________________________________________________________________     H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H O --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               __________________________________________________________________________

Formulations

Useful formulations of the compounds of Formula I can be prepared in conventional ways. They include dusts, granules, pellets, solutions, suspensions, emulsions, wettable powders, emulsifiable concentrates and the like. Many of these may be applied directly. Sprayable formulations can be extended in suitable media and used at spray volumes of from a few liters to several hundred liters per hectare. High strength compositions are primarily used as intermediates for further formulation. The formulations, broadly, contain about 0.1% to 99% by weight of active ingredient(s) and at least one of (a) about 0.1% to 20% surfactant(s) and (b) about 1% to 99.9% solid or liquid inert diluent(s). More specifically, they will contain these ingredients in the following approximate proportions:

    ______________________________________                                                     Active  Weight Percent*                                                        Ingredient                                                                             Diluent(s)                                                                               Surfactant(s)                                    ______________________________________                                         Wettable Powders                                                                             20-90      0-74     1-10                                         Oil Suspensions,                                                                              3-50     40-95     0-15                                         Emulsions, Solutions,                                                          (including Emulsifiable                                                        Concentrates)                                                                  Aqueous Suspension                                                                           10-50     40-84     1-20                                         Dusts          1-25     70-99     0-5                                          Granules and Pellets                                                                         0.1-95      5-99.9  0-15                                         High Strength 90-99      0-10     0-2                                          Compositions                                                                   ______________________________________                                          *Active ingredient plus at least one of a Surfactant or a Diluent equals       100 weight percent.                                                      

Lower or higher levels of active ingredient can, of course, be present depending on the intended use and the physical properties of the compound. Higher ratios of surfactant to active ingredient are sometimes desirable, and are achieved by incorporation into the formulation or by tank mixing.

Typical solid diluents are described in Watkins, et al., "Handbook of Insecticide Dust Diluents and Carriers", 2nd Ed., Dorland Books, Caldwell, N.J., but other solids, either mined or manufactured, may be used. The more absorptive diluents are preferred for wettable powders and the denser ones for dusts. Typical liquid diluents and solvents are described in Marsden, "Solvents Guide," 2nd Ed., Interscience, New York, 1950. Solubility under 0.1% is preferred for suspension concentrates; solution concentrates are preferably stable against phase separation at 0° C. "McCutcheon's Detergents and Emulsifiers Annual", MC Publishing Corp., Ridgewood, N.J., as well as Sisely and Wood, "Encyclopedia of Surface Active Agents", Chemical Publishing Co., Inc., New York, 1964, list surfactants and recommended uses. All formulations can contain minor amounts of additives to reduce foaming, caking, corrosion, microbiological growth, etc.

The methods of making such compositions are well known. Solutions are prepared by simply mixing the ingredients. Fine solid compositions are made by blending and, usually, grinding as in a hammer or fluid energy mill. Suspensions are prepared by wet milling (see, for example, Littler, U.S. Pat. No. 3,060,084). Granules and pellets may be made by spraying the active material upon preformed granular carriers or by agglomeration techniques. See J. E. Browning, "Agglomeration", Chemical Engineering, Dec. 4, 1967, pp. 147ff, and "Perry's Chemical Engineer's Handbook", 5th Ed., McGraw-Hill, New York, 1973, p. 8-57ff.

For further information regarding the art of formulation, see for example:

H. M. Loux, U.S. Pat. No. 3,235,361, Feb. 15, 1966, Col. 6, line 16 through Col. 7, line 19 and Examples 10 through 41;

R. W. Luckenbaugh, U.S. Pat. No. 3,309,192, Mar. 14, 1967, Col. 5, line 43 through Col. 7, line 62 and Examples 8, 12, 15, 39, 41, 52, 53, 58, 132, 138-140, 162-164, 166, 167 and 169-182;

H. Gysin and E. Knusli, U.S. Pat. No. 2,891,855, June 23, 1959, Col. 3, line 66 through Col. 5, line 17 and Examples 1-4;

G. C. Klingman, "Weed Control as a Science", John Wiley & Sons, Inc., New York, 1961, pp. 81-96; and

J. D. Fryer and S. A. Evans, "Weed Control Handbook", 5th Ed., Blackwell Scientific Publications, Oxford, 1968, pp. 101-103.

In the following examples, all parts are by weight unless otherwise indicated.

EXAMPLE 14 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl )aminocarbonyl]-2-(1-                                                     80%                                                methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    sodium alkylnaphthalenesulfonate                                                                           2%                                                 sodium ligninsulfonate      2%                                                 synthetic amorphous silica  3%                                                 kaolinite                   13%                                                ______________________________________                                    

The ingredients are blended, hammer-milled until all the solids are essentially under 50 microns, reblended, and packaged.

EXAMPLE 15 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-                                                      50%                                                methyl-1H--tetrazol-1-yl)benzenesulfonamide                                    sodium alkylnaphthalenesulfonate                                                                           2%                                                 low viscosity methyl cellulose                                                                             2%                                                 diatomaceous earth          46%                                                ______________________________________                                    

The ingredients are blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in diameter. The product is reblended before packaging.

EXAMPLE 16 Granule

    ______________________________________                                         Wettable powder of Example 15 (above)                                                                    5%                                                   attapulgite granules     95%                                                   (U.S.S. 20-40 mesh: 0.84-0.42 mm)                                              ______________________________________                                    

A slurry of wettable powder containing 25% solids is sprayed on the surface of attapulgite granules while tumbling in a double-cone blender. The granules are dried and packaged.

EXAMPLE 17 Extruded Pellet

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl ]-2-(5-                                                     25%                                                methyl-1H--tetrazol-1-yl)benzenesulfonamide                                    anhydrous sodium sulfate    10%                                                crude calcium ligninsulfonate                                                                               5%                                                sodium alkylnaphthalenesulfonate                                                                            1%                                                calcium magnesium bentonite 59%                                                ______________________________________                                    

The ingredients are blended, hammer-milled and then moistened with about 12% water. The mixture is extruded as cylinders about 3 mm diameter which are cut to produce pellets about 3 mm long. These may be used directly after drying, or the dried pellets may be crushed to pass a U.S.S. No. 20 sieve (0.84 mm openings). The granules held on a U.S.S. No. 40 sieve (0.42 mm openings) may be packaged for use and the fines recycled.

EXAMPLE 18 Oil Suspension

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                      25%                                                methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    polyoxyethylene sorbitol hexaoleate                                                                         5%                                                highly aliphatic hydrocarbon oil                                                                           70%                                                ______________________________________                                    

The ingredients are ground together in a sand mill unitl the solid particles have been reduced to under about 5 microns. The resulting thick suspension may be applied directly, but preferably after being extended with oils or emulsified in water.

EXAMPLE 19 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl] -2-(5-                                                     20%                                                methyl-1H--tetrazol-1-yl)benzenesulfonamide                                    sodium alkylnaphthalenesulfonate                                                                           4%                                                 sodium ligninsulfonate      4%                                                 low viscosity methyl cel1ulose                                                                             3%                                                 attapulgite                 69%                                                ______________________________________                                    

The ingredients are thoroughly blended. After grinding in a hammer-mill to produce particles essentially all below 100 microns, the material is reblended and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) and packaged.

EXAMPLE 20 Low Strength Granule

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                      1%                                                 methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    N,N--dimethylformamide      9%                                                 attapulgite granules        90%                                                (U.S.S. 20-40 sieve)                                                           ______________________________________                                    

The active ingredient is dissolved in the solvent and the solution is sprayed upon dedusted granules in a double cone blender. After spraying of the solution has been completed, the blender is allowed to run for a short period and then the granules are packaged.

EXAMPLE 21 Aqueous Suspension

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                      40%                                                methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    polyacrylic acid thickener  0.3%                                               dodecylphenol polyethylene glycol ether                                                                    0.5%                                               disodium phosphate          1%                                                 monosodium phosphate        0.5%                                               polyvinyl alcohol           1.0%                                               water                       56.7%                                              ______________________________________                                    

The ingredients are blended and ground together in a sand mill to produce particles essentially all under 5 microns in size.

EXAMPLE 22 Solution

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       5%                                                methyl-1H-- tetrazol-5-yl)benzenesulfonamide, Sodium                           Salt                                                                           water                       95%                                                ______________________________________                                    

The salt is added directly to the water with stirring to produce the solution, which may then be packaged for use.

EXAMPLE 23 Low Strength Granule

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       0.1%                                              methyl-1H--tetrazoI-5-yl)benzenesulfonamide                                    attapulgite granules        99.9%                                              (U.S.S. 20-40 mesh)                                                            ______________________________________                                    

The active ingredient is dissolved in a solvent and the solution is sprayed upon dedusted granules in a double-cone blender. After spraying of the solution has been completed, the material is warmed to evaporate the solvent. The material is allowed to cool and then packaged.

EXAMPLE 24 Granule

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       80%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    wetting agent                 1%                                               crude ligninsulfonate salt (containing                                                                      10%                                               5-20% of the natural sugars)                                                   attapulgite clay              9%                                               ______________________________________                                    

The ingredients are blended and milled to pass through a 100 mesh screen. This material is then added to a fluid bed granulator, the air flow is adjusted to gently fluidize the material, and a fine spray of water is sprayed onto the fluidized material. The fluidization and spraying are continued until granules of the desired size range are made. The spraying is stopped, but fluidization is continued, optionally with heat, until the water content is reduced to the desired level, generally less than 1%. The material is then discharged, screened to the desired size range, generally 14-100 mesh (1410-149 microns), and packaged for use.

EXAMPLE 25 High Strength Concentrate

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        99%                                              methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    silica aerogel               0.5%                                              synthetic amorphous silica   0.5%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce a material essentially all passing a U.S.S. No. 50 screen (0.3 mm opening). The concentrate may be formulated further if necessary.

EXAMPLE 26 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        90%                                              methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    dioctyl sodium sulfosuccinate                                                                               0.1%                                              synthetic fine silica        9.9%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce particles essentially all below 100 microns. The material is sifted through a U.S.S. No. 50 screen and then packaged.

EXAMPLE 27 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       40%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    sodium ligninsulfonate       20%                                               montmorillonite clay         40%                                               ______________________________________                                    

The ingredients are thoroughly blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in size. The material is reblended and then packaged.

EXAMPLE 28 Oil Suspension

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       35%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    blend of polyalcohol carboxylic                                                                              6%                                               esters and oil soluble petroleum                                               sulfonates                                                                     xylene                       59%                                               ______________________________________                                    

The ingredients are combined and ground together in a sand mill to produce particles essentially all below 5 microns. The product can be used directly, extended with oils, or emulsified in water.

EXAMPLE 29 Dust

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       10%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    attapulgite                  10%                                               Pyrophyllite                 80%                                               ______________________________________                                    

The active ingredient is blended with attapulgite and then passed through a hammer-mill to produce particles substantially all below 200 microns. The ground concentrate is then blended with powdered pyrophyllite until homogeneous.

Utility

Test results indicate that the compounds of the present invention are highly active preemergent or postemergent herbicides or plant growth regulants. They have utility for broad-spectrum pre- and/or post-emergence weed control in areas where complete control of all vegetation is desired, such as around fuel storage tanks, ammunition depots, industrial storage areas, parking lots, drive-in theaters, around billboards, highway and railroad structures. Some of the compounds have utility for selective weed control in crops such as corn, rice, wheat, barley and rape. Alternatively, many of the subject compounds are useful to modify plant growth.

The rates of application for the compounds of the invention are determined by a number of factors, including their use as plant growth modifiers or as herbicides, the crop species involved, the types of weeds to be controlled, weather and climate, formulations selected, mode of application, amount of foliage present, etc. In general terms, the subject compounds should be applied at levels of about 0.001 to 10 kg/ha, the lower rates being suggested for use on lighter soils and/or those having a low organic matter content, for plant growth modification or for situations where only short-term persistence is required.

The compounds of the invention may be used in combination with any other commercial herbicide, examples of which are those of the triazine, triazole, uracil, urea, amide, diphenylether, carbamate, phenoxyacetic acid and bipyridylium types, as well as other sulfonylureas. They are particularly useful in combination with the following herbicides.

    ______________________________________                                                  Chemical Name                                                         ______________________________________                                         Common Name                                                                    alachlor   2-chloro-2',6'-diethyl-N--(methoxymethyl)-                                     acetanilide                                                         atrazine   2-chloro-4-(ethylamino)-6-(isopropyl-                                          amino)- .sub.-s-triazine                                            butylate   S--ethyl-diisobutylthiocarbamate                                    cyanazine  2-[[4-chloro-6-(ethylamino)- .sub.-s-triazin-2-                                yl]amino]-2-methylpropionitrile                                     dicamba    3,6-dichloro- .sub.-o-anisic acid                                   EPTC       S--ethyl dipropylthiocarbamate                                      linuron    3-(3,4-dichlorophenyl)-1-methoxy-1-                                            methylurea                                                          metolachlor                                                                               2-chloro-N--(2-ethyl-6-methylphenyl)-N--                                       (2-methoxy-1-methylethyl)acetamide                                  metribuzin 4-amino-6-tert-butyl-3-(methylthio)-as-                                        triazine-5(4H)--one                                                 tridiphane 2-(3,5-dichlorophenyl)-2-(2,2,2-tri-                                           chloroethyl)oxirane                                                 2,4-D      (2,4-dichlorophenoxy)acetic acid                                    thiobencarb                                                                               S--4-chlorobenzyldiethylthiocarbamate                               molinate   S--ethyl N,N--hexamethylenethiocarbamate                            butachlor  N--(butoxymethyl)-2-chloro-2',6'-di-                                           ethylacetanilide                                                    naproanilide                                                                              N--phenyl-2-(1-naphthyloxy)propionamide                             pyrazolate 4-(2,4-dichlorobenzoyl)-1,3-dimethyl-                                          pyrazol-5-yl-4-toluenesulfonate                                     pretilachlor                                                                              2-chloro-2',6'-diethyl-N--( -n-propoxy-                                        ethyl)acetanilide                                                   oxidiazon  3-[2,4-dichloro-5-(1-methylethoxy)-                                            phenyl]-5-(1,1-dimethylethyl)-1,3,4-                                           oxadiazol-2(3H)--one                                                Trade Name or                                                                  Code Number                                                                    Harmony ®                                                                             3-[[(4-methoxy-6-methyl-1,3,5-triazin-                                         2-yl)aminocarbonyl]aminosulfonyl]-2-                                           thiophenecarboxylic acid, methyl ester                              Cinch ®                                                                               exo-1-methyl-4-(1-methylethyl)-2-[(2-                                          methylphenyl)methoxy]-7-oxabicyclo-                                            [2.2.1]heptane                                                      MY-93      S--(1-methyl-1-phenethyl)piperidine-1-                                         carbothioate                                                        CH-83      S--(2-methylpropyl)-hexanhydro-1H--aze-                                        pine-1-carbothioic acid, ester                                      X-52       2,4-dichlorophenyl-3-methoxy-4-nitro-                                          phenyl ether                                                        SC-2957    S--benzyl-N--ethyl-N--propylthiocarbamate                           HW-52      N--(2,3-dichlorophenyl)-4-(ethoxy-                                             methoxy)benzamide                                                   NTN-801    2-(benzothiazol-2-yl)-N--methyl-N--                                            phenylacetamide                                                     SL-49      2-[4-[(2,4-dichlorophenyl)carbonyl]-                                           1,3-dimethyl-1H--pyrazol-5-yloxy]-1-                                           phenylethanone                                                      BAS-514    3,7-dichloro-8-quinoline carboxylic                                            acid                                                                ______________________________________                                    

The herbicidal properties of the subject compounds were discovered in a number of greenhouse tests. The test procedures and results follow.

    __________________________________________________________________________     COMPOUNDS                                                                      General Structures for Compound 1-58                                            ##STR36##                                                                      ##STR37##                                                                     Compound                                                                             Q  R.sub.1                                                                            R.sub.3                                                                              R.sub.4                                                                            R.sub.5                                                                           X    Y     Z                                         __________________________________________________________________________      1    Q-3                                                                               H   --   CH.sub.3                                                                            -- OCH.sub.3                                                                           CH.sub.3                                                                             N                                          2    Q-3                                                                               H   --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         3    Q-1                                                                               H   CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         4    Q-3                                                                               H   --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         5    Q-3                                                                               H   --   CH.sub.3                                                                            -- Cl   OCH.sub.3                                                                            CH                                         6    Q-3                                                                               H   --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          7    Q-3                                                                               H   --   CH.sub.3                                                                            -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                          8    Q-3                                                                               H   --   H    -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          9    Q-3                                                                               H   --   H    -- Cl   OCH.sub.3                                                                            CH                                        10    Q-3                                                                               H   --   H    -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        11    Q-3                                                                               H   --   H    -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        12    Q-3                                                                               H   --   H    -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         13    Q-3                                                                               H   --   H    -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        14    Q-3                                                                               5-CH.sub.3                                                                         --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        15    Q-3                                                                               5-CH.sub.3                                                                         --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         16    Q-3                                                                               5-CH.sub.3                                                                         --   CH.sub.3                                                                            -- Cl   OCH.sub.3                                                                            CH                                        17    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        18    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        19    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        20    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- Cl   OCH.sub.3                                                                            CH                                        21    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         22    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         23    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        24    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        25    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         26    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         27    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        28    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- Cl   OCH.sub.3                                                                            CH                                        29    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         30    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         31    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         32    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        33    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        34    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        35    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- Cl   OCH.sub.3                                                                            CH                                        36    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         37    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         38    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         39    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub. 3                                                                           CH                                        40    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        41    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        42    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- Cl   OCH.sub.3                                                                            CH                                        43    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         44    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         45    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         46    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        47    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        48    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        49    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- Cl   OCH.sub.3                                                                            CH                                        50    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         51    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         52    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         53    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        54    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        55    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        56    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- Cl   OCH.sub.3                                                                            CH                                        57    Q-5                                                                               H   --   --   CH.sub.3                                                                          OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        58    Q-5                                                                               H   --   --   CH.sub.3                                                                          CH.sub.3                                                                            OCH.sub.3                                                                            N                                         __________________________________________________________________________

    ______________________________________                                         General Structures for Compounds 59- 63                                         ##STR38##                                                                     Compound     X          Y          Z                                           ______________________________________                                         59           OCH.sub.3  OCH.sub.3  CH                                          60           CH.sub.3   OCH.sub.3  CH                                          61           CH.sub.3   CH.sub.3   CH                                          62           OCH.sub.3  OCH.sub.3  N                                           63           Cl         OCH.sub.3  CH                                          ______________________________________                                    

    __________________________________________________________________________     General Structures for Compounds 64- 179                                        ##STR39##                                                                      ##STR40##                                                                     Compound                                                                             Q  R  R.sub.1                                                                             R.sub.3                                                                             R.sub.4 R.sub.5                                                                             X      Y       Z                            __________________________________________________________________________      64   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             65   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             66   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            67   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            68   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            69   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                            70   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             71   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             72   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            73   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            74   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            75   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                            76   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            77   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            78   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            79   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   Cl     OCH.sub.3                                                                              CH                            80   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             81   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             82   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            83   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            84   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            85   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                            86   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub. 3                                                                             N                             87   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             88   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            89   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            90   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            91   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   Cl     OCH.sub.3                                                                              CH                            92   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             93   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             94   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                            95   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                            96   Q-1                                                                               H  H    CH.sub.2 CH.sub.3                                                                   --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                            97   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            98   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                            99   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           100   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   Cl     OCH.sub.3                                                                              CH                           101   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              CH.sub.3                                                                               CH                           102   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           103   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           104   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           105   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           106   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           107   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           108   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           109   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub. 3                                                                             CH.sub.3                                                                               CH                           110   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                           111   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            112   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            113   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            114   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            115   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           116   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           117   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            118   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              N                            119   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           120   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            121   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           122   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            123   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           124   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           125   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           126   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            127   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           128   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              N                            129   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   Cl     OCH.sub.3                                                                              CH                           130   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              CH.sub.3                                                                               CH                           131   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           132   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           133   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           134   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                           135   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            136   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            137   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   Br     OCH.sub.3                                                                              CH                           138   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           139   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            140   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              H       CH                           141   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             H       CH                           142   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              CH                           143   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              N                            144   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            145   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   cyclopropyl                                                                           OCH.sub.3                                                                              N                            146   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.2 CH.sub.                                                                      CH                           147   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             CH.sub.2 OCH.sub.2 CH.sub.3                                                            CH                           148   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.2 CF.sub.3                                                                     N                            149   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                     N                            150   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            151   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            152   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           153   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           154   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           155   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           156   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                            157   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             CH(OCH.sub.3).sub.2                                                                    CH                           158   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           159   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            CH.sub.3                                                                              OCH.sub.3                                                                              CH                           160   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            CH.sub.3                                                                              OCH.sub.3                                                                              N                            161   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           162   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           163   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           164   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           165   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           166   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           167   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            168   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            169   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                            170   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           171   Q-5                                                                               H  H    --   --      CH.sub.3                                                                            OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           172   Q-5                                                                               H  H    --   --      CH.sub.3                                                                            OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           173   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           174   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            175   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            176   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           177   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           178   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           179   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           __________________________________________________________________________

    ______________________________________                                         General Structure for Compounds 180- 205                                        ##STR41##                                                                      ##STR42##                                                                     Compound                                                                               Q      R.sub.1                                                                               R.sub.3                                                                               X       Y      Z                                  ______________________________________                                         180     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.3                                                                               CH.sub.3                                                                              CH                                 181     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 182     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              OCH.sub. 3                                                                             OCH.sub.3                                                                             CH                                 183     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              Cl      OCH.sub.3                                                                             CH                                 184     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                     NHCH.sub.3                                                                            N                                  185     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             N                                  186     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  187     Q-2    H      CH.sub.3                                                                              CH.sub.3                                                                               CH.sub.3                                                                              CH                                 188     Q-2    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 189     Q-2    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             CH                                 190     Q-2    H      CH.sub.3                                                                              Cl      OCH.sub.3                                                                             CH                                 191     Q-2    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             N                                  192     Q-2    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  193     Q-2    H      CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                     NHCH.sub.3                                                                            N                                  194     Q-1    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 195     Q-1    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             CH                                 196     Q-1    H      CH.sub.3                                                                              CH.sub.3                                                                               CH.sub.3                                                                              CH                                 197     Q-1    H      CH.sub.3                                                                              Cl      OCH.sub.3                                                                             CH                                 198     Q-1    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             N                                  199     Q-1    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  200     Q-2    H      CH.sub.2 CH.sub.3                                                                     CH.sub.3                                                                               CH.sub.3                                                                              CH                                 201     Q-2    H      CH.sub.2 CH.sub.3                                                                     CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 202     Q-2    H      CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              OCH.sub.3                                                                             CH                                 203     Q-2    H      CH.sub.2 CH.sub.3                                                                     Cl      OCH.sub.3                                                                             CH                                 204     Q-2    H      CH.sub.2 CH.sub.3                                                                     CH.sub.3                                                                               OCH.sub.3                                                                             N                                  205     Q-2    H      CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  ______________________________________                                    

TEST A

Seeds of crabgrass (Digitaria spp.), giant foxtail (Setaria faberii) (in some cases), barnyardgrass (Echinochloa crusgalli), cheatgrass (Bromus secalinus), wild oats (Avena fatua), velvetleaf (Abutilon theophrasti), morningglory (Ipomoea spp.), cocklebur (Xanthium pensylvanicum), sorghum, corn, soybean, sugarbeet, cotton, rice, barley (in some cases), wheat and purple nutsedge (Cyperus rotundus) tubers were planted and treated preemergence with the test chemicals dissolved in a non-phytotoxic solvent. At the same time, these crop and weed species were treated with a soil/foliage application. At the time of treatment, the plants ranged in height from 2 to 18 cm. Treated plants and controls were maintained in a greenhouse for sixteen days, after which all species were compared to controls and visually rated for response to treatment. The ratings, summarized in Table A, are based on a numerical scale extending from 0=no injury, to 10=complete kill. The accompanying descriptive symbols have the following meanings:

C=chlorosis/necrosis;

B=burn;

D=defoliation;

E=emergence inhibition;

G=growth retardation;

H=formative effect;

U=unusual pigmentation;

X=axillary stimulation;

S=albinism; and

6Y=abscised buds or flowers.

    TABLE A       Cmpd. 1 Cmpd. 2 Cmpd. 3 Compound 4 Compound 5 Compound 6 Compound 7      Compound 8 Compound 9 Compound 10 Compound 11 Rate kg/ha 0.05 0.05 0.05      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01        POSTEMERGENCE Morningglory 3C,8G 10C 10C 10C 10C 10C 9C 1C,1H 1C 6C,9G      4C,9H 1H 3H 0 5C,9G 2C,5G 10C 9C 2C,6G 2H Cocklebur 3C,7H 9C 9C 9C 9C      10C 9C 1H 0 8G 2G 0 2H 0 9C 3C,9H 9C 9C 9C 5C,9G Velvetleaf 2C,4G 10C 9C      9C 9C 9C 4C,9H 0 0 4C,8H 3C,5G 2G 0 0 4C,8G 1C 9C 4C,8G 5C,9H 4C,9H      Nutsedge 8G 9C 9C 4C,9G 3C,9G 9C 4C,9G 0 0 6G 0 0 0 0 4C,9G 3C,9G 9C 9C      4C,9G 3C,9G Crabgrass 5G 5C,9G 9C 5C,9G 3C,8G 4C,8G 3C,5G 0 0 4C,8G      2C,5G 0 0 0 2G 0 3C,7G 2H 3C,5G 1H Giant Foxtail    -- -- -- -- -- -- --      -- 0 -- -- -- -- -- -- -- -- Barnyardgrass 5C,9G 9C 5C,9G 9C 9C 9C 9C      4C,9H 0 5C,9H 3C,9H 1H 2H 0 9H 2C,5H 9H 3C,7H 5C,9H 2C,3H Cheatgrass 0      7G 9C 3C,9G 6G 4G 0 0 0 6G 2G 0 0 0 7G 0 9C 3C,9G 9C 8G Wild Oats 3C,8G      9C 9C 5C,9G 5C,9G 4C,9G 3C,9G 2G 0 5C,9G 4C,9G 0 0 0 0 0 5C,9G 2C,7H 9C      9H Wheat 4C,9G 9C 9C 5C,9G 2C,9G 4C,9H 8G 3G 0 4C,9G 2C,9G 0 0 0 0 0 9G      3G 9G 5G Corn 9C 9C 9C 5C,9G 3C,9H 5C,9G 9H 4C,9H 3C,7H 6C,9G 4C,9H 5H      5H 2G 7H 1C,3G 9C 3C,9H 5C,9G 3C,9H Barley    -- -- -- -- -- -- -- -- 0      -- -- -- -- -- -- -- -- Soybean 5C,9G 9C 9C 5C,9G 5C,9G 4C,9G 4C,9H      4C,8H 1C,1H 3C,7G 3G 2G 3H 0 5G 0 5C,9G 3C,8H 3C,7H 2H Rice 6C,9G 9C 9C      9C 9C 6C,9G 9C 5C,9G 5G 9C 9C 2G 2G 0 4C,8G 0 9C 2C,7G 9C 5C,9G Sorghum      6C,9H 9C 9C 5C,9G 6C,9G 9C 9C 4C,8H 3G 5C,9G 4C,9H 5G 0 0 5C,9H 3C,8H 9C      3C,9H 9C 4C,9H Sugar Beets 6C,9H 9C 9C 8G 10C 9C 9C 4C,6G 0 5C,9H 4C,6H      2C,3H 3C,5H 0 10C 4C,9H 10C 10C 9C 9C Cotton 6C,9H 9C 9C 9C 9C 9C 4C,9G      4C,6G 3C,4G 3C,5G 3C,5G 2G 0 0 9C 3C,8H 9C 9C 9C 9H PREEMERGENCE      Morningglory 3G 9H 9G 9G 9G 9G 9G 0 0 9G 7G 0 0 0 9G 4C,8H 9G 8G 8G      3C,5H Cocklebur 0 9H 9H 9H 9H 9H 9H 0 0 8G 7G 0 0 0 8H 2C,5G -- 9H 9H 8H      Velvetleaf 0 10C 10C 9C 9C 9C 4C,8G 0 0 4C,9G 0 0 0 0 7H 4G 9C 6C,9G 9C      3C,7H Nutsedge 0 10E 10E 10E 4C,8G 10E 10E 0 0 0 0 0 0 0 10E 3G 10E 9G      10E 4G Crabgrass 0 3C,8G 8G 5C,9G 5C,9G 4C,9G 7G 0 0 4C,8G 0 0 0 0 2C 0      4C,7G 2C,4G 2C,3G 0 Giant Foxtail    -- --  -- -- -- -- -- -- 0 -- -- --      ---- -- -- -- Barnyardgrass 0 4C,9H 9H 5C,9H 5C,9H 4C,9H 4C,9H 0 0 9H 3G      0 0 0 3C,7G 0 4C,9H 2C,6G 3C,5G 0 Cheatgrass 0 7G 9H 9G 7G 5G 3G 0 0 5G      0 0 0 0 3C,7H 4G 10E 4C,9H 5C,9H 5G Wild Oats 0 5C,9G 5C,9G 6C,9H 4C,8H      5C,9G 3C,7G 0 0 5C,9H 3C,6G 0 1C 0 2C,7G 0 9C 4C,9G 9C 3C,7G Wheat 5G      10E 10E 10E 5C,9H 4C,9H 9G 4G 0 4C,9H 2C,6G 0 0 0 6G 0 4C,9G 7G 9G 5G      Corn 3C,8G 4C,9G 3C,9H 9H 5C,9H 3C,9G 8G 2G 0 9G 3C,7G 0 4G 0 3C,8H 0 9H      4C,9H 2C,9H 3C,7H Barley    -- -- -- -- -- -- -- -- 0 -- -- -- -- -- --      -- -- Soybean 5G 9H 9H 9H 4C,7G 3C,8H 4C,6G 0 0 2G 0 0 2G 0 3G 0 9H      4C,8H 2C,7G 2C,3G Rice 1C 10E 10E 10E 10E 10E 10E 3G 0 10E 4C,8H 0 5G 0      10E 7G 10E 4C,9H 10E 3C,8G Sorghum 3C,6G 5C,9H 10H 10E 5C,9H 10E 9H 0 0      10E 4C,9H 0 0 0 4C,9H 4C,8G 10E 5C,9H 9H 3C,8H Sugar Beets 0 5C,9G 9C      5C,9G 5C,9G 5C,9G 5C,9G 0 0 5C,9G 4C,8G 0 4G 3H 9C 4C,8G 5C,9G 5C,9G 9C      5C,9G Cotton 0 3C,9G 9C 3C,9G 3C,9G 3C,9G 3C,9G 0 0 2C,5G 0 0 0 0 9G 8G      9C 9G 9G 9G        Cmpd. 12 Cmpd. 13 Compound 14 Compound 15 Compound 16 Compound 17      Compound 18 Compound 19 Compound 20 Compound 21 Compound 22 Rate kg/ha      0.01 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE Morningglory 2G 10C 5C,9G 4G 3C,8H 0 10C 5C,9G 10C 10C      10C 9C 10C 4C,9G 10C 9C 4C,9G 3C,7H 4C,8H 3C,7H Cocklebur 0 10C 10C 10C      2C,4G 0 10C 8G 10C 10C 10C 10C 9C 7G 10C 9C 5C,9H 5H 5C,9G 3C,7H      Velvetleaf 0 9C 10C 10C 2C,4H 0 9C 3C,8G 9C 9C 10C 9C 9C 9C 9C 2C,7G      3C,6G 1H 3C,7H 3C,5H Nutsedge 0 9C 9C 5C,9G 0 0 5C,9G 2C,8G 5C,9G 3C,9G      10C 10C 5C,9G 3C,8G 5C,9G 4C,9G 4G 3C,8G 5G 0 Crabgrass 0 4G 2C,7G 1C 0      0 5G 0 3C,8G 3C,5G 9C 3C,7G 4C,8G 3C,4G 3C,7G 3C,3G 3C,5G 2G 3C,7H 3C,6G      Giant Foxtail -- -- -- -- -- -- -- -- 9C 9C 9C 5C,9H 9C 5C,9G 5C,9H      4C,8G 9C 4C,9G 9C 4C,9H Barnyardgrass 0 5C,9H 9C 9C 3C,8H 3G 9C 3C,8H 9C      9C 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C Cheatgrass 0 4C,9G 3G 0 0 0 0 0 5C,9G      3C,8G 9C 2C,8G 3C,7G 5G 5G 2G 0 0 2C 0 Wild Oats 0 3C,5G 5C,9G 3C,9G      2C,9G 2C,2G 3C,9G 2C,5G 9C 5C,9G 5C,9G 4C,9G 9C 9C 3C,9G 3C,7G 2C 0      2C,6G 0 Wheat 0 0 5C,9G 2C,9G 0 0 8G 5G 4C,9G 9G 9C 3C,9G 9C 5C,9G 3C,9G      9G 5G 0 8G 0 Corn 0 9H 9C 5C,9H 1C,5G 2G 4G 2G 9C 5C,9G 10C 3C,9H 9C      4C,9H 4C,9H 3C,9H 10C 9C 10C 9C Barley -- -- -- -- -- -- -- -- 5C,9G      3C,8H 6C,9G 3C,8G 9C 4C,9G 2C,8G 3C,7G 0 0 2G 0 Soybean 1H 9C 9C 9C      4C,9G 3H 3C,9G 2H,7G 9C 9C 9C 9C 9C 4C,9G 9C 4C,9G 5C,9G 4C,9G 9C 5C,9G      Rice 0 2C,8G 9C 9C 5G 0 5C,9G 7G 9C 9C 9C 9C 9C 9C 9C 5C,9G 5C,9G 7G 9C      6G Sorghum 0 9H 9C 5C,9H 3C,9H 0 9C 3C,9H 9C 9C 9C 9C 10C 9C 9C 9C 9C      4C,9G 9C 9C Sugar Beets 1C,1H 5C,9G 5C,9G 9C 3C,6G 2C,3G 9C 4C,8G 10C      5C,9G 10C 9C 10C 4C,8G 9C 4C,9G 3C,6H 3C,5G 9C 3C,8G Cotton 1C 9C 9C      5C,9G 3C,9H 1H 2C,9G 8G 9C 5C,9G 9C 10C 9C 4C,9G 5C,9G 9C 4C,9H 4C,9H      4C,9H 3C,8H PREEMERGENCE Morningglory 0 9G 9G 8G 5H 3H 9C 9H 9C 7H 9G 8G      8H 3C,7G 9G 7H 5H 0 3C,8H 2H Cocklebur 0 9H 9H 9H 7H 0 9H 9H 9H 9H 9H 9H      8H -- 9H 9H 9H -- 9H 2C Velvetleaf 0 5C,9G 10C 9C 6G 0 9C 2C,4G 9C 3C,8G      9C 9C 9C 3C,7H 5C,9G 7G 7G 0 8H 5G Nutsedge 0 10E 10E 4C,9G 0 0 10E      3C,9G 10E 10E 10E 10E 9G 7G 10E 9G 0 0 0 0 Crabgrass 0 3G 2C,7G 3G 0 0      4G 2G 4C,8G 3C,7G 8G 4G 5G 0 9C 2G 2C,5G 0 2C,5G 4G Giant Foxtail -- --      -- -- -- -- -- -- 4C,9H 3C,8H 9H 3C,6G 9H 5G 4C,8G 4G 2C,5G 2G 3C,7G 3G      Barnyardgrass 0 3C,8H 5C,9H 3C,8H 1C 0 3C,9H 3C,3G 5C,9H 4C,9H 5C,9H      3C,9H 3C,8H 3C,6G 9H 3C,8H 3C,6G 0 3C,8G 0 Cheatgrass 0 8G 6G 2G 0 0 0 0      4C,8H 3G 7H 6G 2G 0 3G 0 0 0 0 0 Wild Oats 0 5G 9C 5C,9G 2C,5G 0 5C,9G      3C,6G 5C,9G 4C,9G 5C,9G 2C,9G 5C,9G 3C,8H 3C,9H 2C,5G 2G 0 2C 0 Wheat 0      0 4C,9G 3C,8G 0 0 8G 3G 10H 3C,8G 10H 9G 5C,9H 3C,8H 3C,9H 7G 0 0 3G 0      Corn 2G 8G 3C,9G 7G 6G 0 6G 2G 10H 4C,9H 4C,9H 8G 4C,9H 3C,7H 3C,9H 9H      4C,9H 2C,6G 9H 3C,8H Barley -- -- --  -- -- -- -- -- 9G 3C,9G 3C,9G 9G      4C,9G 9G 3C,9G 8G 0 0 7G 0 Soybean 2C 3C,8H 3C,9H 2C,7G 2C,2H 1C 3C,7G      3C,3H 9H 4C,8H 9H 4C,8H 9H 3C,6H 3C,8H 3C,5G 3C,7H 0 3C,7H 2C,3G Rice 0      2C,9H 10E 3C,8G 5G 1C 10E 2C,8G 10E 9H 10E 10E 10E 4C,8H 10E 9H 8G 2G 9H      0 Sorghum 1C 3C,9H 10E 3C,9H 3C,6G 0 10H 3C,9H 10H 6C,9H 10H 10H 5C,9H      6C,9H 10H 10H 5C,9H 3C,6G 4C,9H 3C,8H Sugar Beets 3H 10C 5C,9G 5C,9G      3C,7H 0 10E 5C,9G 10E 9C 5C,9G 5C,9G 9C 5G 9C 5C,9G 5G 3G 4C,7H 5G      Cotton 0 9G 9G 9G 2C 0 9G 2C,5G 9C 2C,9G 4C,9G 4C,9G 9G 2C,8G 9G 8G 5G 0      2C,5G 1C        Compound 23  Compound 24 Compound 25 Compound 26 Compound 27 Compound      28 Compound 29 Compound 30 Compound 31 Compound 32 Rate kg/ha 0.05 0.01      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01        POSTEMERGENCE Morningglory 10C 8G 5G 0 0 3C,5G 0 2C,6G 2G 10C 3C,8G      3C,9G 3C,7H 10C 4C,8H 10C 3C,8H 10C 10C Cocklebur 10C 10C 10C 3H 2H      4C,8H 2H 10C 5C,9G 10C 9C 3H 0 9C 4C,9G 10C 9C 10C 10C Velvetleaf 10C      5C,9G 5C,9G 0 0 2C,5G 0 9C 3C,7G 4C,9G 3C,9G 3C,7H 0 9C 7G 9C 4C,8H 10C      10C Nutsedge 10C 10C 5C,9G 0 0 3C,6G 0 10C 3C,8G 10C 4C,9G 0 0 4C,8G 4G      7G 0 10C 9C Crabgrass 5G 3G 0 0 0 3C,4H 0 2G 2G 3G 0 3C,5G 0 6C,9H 4C,6G      9C 3C,8G 5C,8G 7G Giant Foxtail 5C,9G 3C,8G 3C,7G 3C,8H 2H 4C,9H 3C,5G      4C,9G 4G 7G 2G 5C,9G 3C,7G 9C 10C 10C 9C 9C 9C Barnyardgrass 9C 3C,9H      3C,7G 5C,9H 0 5C,9H 2C,5G 4C,9H 4C,8H 3C,7H 1C,4G 3C,8H 2H 10C 9C 10C 9C      9C 9C Cheatgrass 5G 2G 2G 0 0 3G 0 4G 0 0 0 0 0 3G 0 3G 0 7G 5G Wild      Oats 5G 2G 0 4C,8G 0 4C,9G 3C,4G 9G 3C,6G 2G 0 4C,9G 7G 4G 3G 7G 4G      4C,9G 9G Wheat 8G 6G 5G 5C,9G 0 3C,9G 7G 5C,9G 2C,6G 4G 0 9G 7G 4G 0      2C,6G 3G 10C 6C,9G Corn 9H 6H 0 3C,9H 2H 9H 0 2G 0 0 0 4C,8H 5H 10C 10C      10C 9C 10C 2C,7H Barley 3C,9H 6G 3G 9G 2G 8G 0 9G 3G 2G 0 9C 9G 0 0      1C,4G 0 9C 8G Soybean 9C 9C 9C 2H,4G 0 3C,8G 2H 5C,9G 4C,9H 3H,8G 3H,8G      3C,7H 4H 9C 5C,9G 9C 4C,9G 9C 9C Rice 9C 4C,9G 3C,7G 9C 2G 9C 8G 9C      5C,9G 2C,8G 6G 9C 3C,8G 5C,9G 4C,9G 9C 4C,9G 9C 9C Sorghum 9C 9C 4C,9H      4C,9H 3G 5C,9G 3C,7H 9C 4C,9G 4C,9H 4C,9G 5C,9G 4C,9G 9C 9C 10C 9C 10C      9C Sugar Beets 10C 10C 10C 5G 0 9C 2H 10C 9C 9C 9C 3C,7H 4H 10C 5C,9G      10C 9C 10C 10C Cotton 9C 9C 4C,9G 0 0 3C,7G 0 9C 9H 9H 9G 5H 0 9C 9H 9C      9C 9C 10C PREEMERGENCE Morningglory 9H 7H 7H 0 0 2H 1H 6G 0 3C,9G 5H 5H      1C 9C 4C,4H 4C,8H 3C,5H 9C 8H Cocklebur 9H 9H 9H 0 0 2C 0 8H 6H 9H 3C,4H      0 0 9H 3C 9H 2C,5G 9H 8H Velvetleaf 10C 9G 9C 3G 0 0 0 3C,8H 7G 5C,9H 2G      0 0 9C 9C 9C 0 10C 10C Nutsedge 10E 9G 3C,7G 0 0 0 0 5G 0 10E 0 0 0 4G 0      4G 0 10E 10E Crabgrass 0 0 2G 0 0 0 0 0 0 0 0 0 0 3C,7G 3C,4G 3C,5G 0 7G      4G Giant Foxtail 4C,9H 1C 3C,5G 3G 0 0 0 3C,6G 3C 3C,3H 3G 5G 0 9H 3G      3C,6G 1C 5C,9G 4C,7G Barnyardgrass 5C,9H 3C,8H 3C,6G 0 0 2C 0 4C,9H      3C,3G 5C,9H 3C,3G 3C,5G 0 5C,9H 3C,7G 9C 3C,4H 9C 9H Cheatgrass 4G 0 0 0      0 0 0 0 0 3G 3G 0 0 3G 0 2G 0 7G 0 Wild Oats 6G 0 2C 0 0 0 0 3C,7G 2C 2C      0 3C,6G 0 2C 0 2C,4G 0 5C,9G 3C,8G Wheat 4C,9G 4G 5G 0 0 0 0 7G 2G 6G 0      9H 2G 2G 0 2G 0 10E 4C,9G Corn 3C,8G 2C,5G 0 3G 0 0 0 2C 0 2G 0 2C,5G 0      5C,9H 9H 9H 0 3C,9H 3C,7G Barley 3C,9G 2C,8G 2C,8G 5G 0 5G 3G 9G 6G 8G      5G 2C,8G 2G 5G 0 5G 0 5C,9G 4C,9G Soybean 3C,8H 3C,8H 3C,7H 0 0 0 0      2C,7G 2C,2H 3C,5G 3C,4G 2C,2H 0 3C,8H 3C,7H 3C,8H 2H 9H 3C,7H Rice 9H      4C,9G 3C,6H 5G 0 3C,5G 2C 9H 3C,7H 5C,9H 4C,8H 3C,8H 2C 9H 3C,6H 4C,9H      2C,4G 10E 10E Sorghum 10E 3C,9H 4C,8H 2C 0 3C,5G 2G 9H 2C,6G 5C,9H 5C,9H      3C,8H 1C 6C,9H 4C,8H 10H 4C,7G 6C,9H 9C Sugar Beets 5C,9G 5C,9G 5C,9G 0      0 2H 3G 4C,8G 3C,7H 10C 3C,7G 3G 4H 10E 5H 5C,9G 5H 4C,8G 9C Cotton 10C      9C 2C,7H -- 0 1C 0 4C,8G 2C,3G 3C,7G 2C,4G 0 2H 4C,9G 2C,2H 4C,8H 2C 9C      9G        Compound 33 Compound 34 Compound 35 Compound 36 Compound 37 Compound      38 Compound 39 Compound 40 Compound 41 Compound 42 Rate kg/ha 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01        POSTEMERGENCE Morningglory 10C 10C 10C 5C,9G 10C 10C 9C 10C 3C,8H      3C,5H 3C,8H 1C 10C 10C 10C 9C 4C,8H 2C,4G 2C,8G 2C,7G Cocklebur 10C 9C      10C 5C,9G 10C 10C 9C 3C,8H 2C,2G 0 3C,7H 0 9C 9C 9C 9C 5C,9H 2C,4G 5C,9H      3C,8G Velvetleaf 10C 9C 10C 5C,9G 10C 4C,9G 9C 9C 2C,4G 0 2C,5G 1C 9C      10C 10C 5C,9H 4C,8H 3C,5H 4C,8H 5G Nutsedge 9C 5C,9G 5C,9G 5C,9G 10C      4C,9G 3C,7G 3G 0 0 0 0 9C 5C,9G 2C,8G 5G 0 0 3G 4G Crabgrass 3C,7G 2G      2C,9G 2C,4G 3C,7H 3G 9C 3C,7G 2C,3G 0 2G 0 5C,9G 3C,7G 3C,7G 4G 2G 0 0 0      Giant Foxtail 9C 4C,9H 10C 9C 9C 4C,9G 9C 9C 4C,8G 4G 3C,8H 2G 5C,9G      3C,7G 3C,7G 2G 5G 0 4G 0 Barnyardgrass 10C 9C 10C 4C,9H 10C 10C 9C 10C      9C 3C,7H 5C,9G 4H 9C 9C 9C 3C,7H 2C,7H 3H 4C,9H 4G Cheatgrass 7G 5G 6G      2G 6G 2G 7G 3G 2C,6G 2G 2G 0 10C 9C 9C 4C,9G 3C,8G 4G 7G 0 Wild Oats      5C,9G 3C,7G 9C 4C,9G 3C,9G 3C,6G 9C 9C 2C,6G 0 2C,5G 0 5C,9G 9G 4C,9G      3C,6G 7G 3G 2C,7G 0 Wheat 9C 4C,9G 9C 3C,9G 5C,9G 2C,8G 9C 5C,9G 0 0 4G      0 3C,9G 9G 9G 9G 4G 2G 2G 0 Corn 3C,9H 3C,7H 4C,9H 1H 4G 0 9C 9C 4C,9G      3C,8H 3C,9H 3C,7H 3C,9G 2U,9G 3C,8H 1C,3G 0 0 2G 0 Barley 3C,9G 4C,9G 9C      2C,8G 9C 6G 9C 4C,9G 0 0 0 0 4C,9G 9G 5G 2G 0 0 0 0 Soybean 10C 5C,9G 9C      4C,9G 4C,9G 4C,9G 5C,9G 4C,9G 4C,9G 3C,3G 3C,8G 2C,4H 6C,9G 5C,9G 9C      4C,9G 4C,8H 3C,5H 2C,7G 1H Rice 9C 9C 9C 9C 9C 5C,9G 9C 9C 5C,9G 4C,9G      5C,9G 5G 9C 5C,9G 9C 4C,9G 5C,9G 3C,5G 2C,9G 5G Sorghum 10C 10C 9C 4C,9H      9C 9C 9C 9C 4C,9G 4C,9G 4C,9G 2C,6G 3U,9G 9G 4C,9H 3C,8G 2C,6G 2C,4G 9G      7G Sugar Beets 9C 5C,9G 10C 9C 10C 10C 9C 10C 3C,7H 2H 3C,7H 3C,4H 10C      9C 10C 3C,8H 3C,6H 2C,3G 3C,8G 2C,6G Cotton 9C 9C 10C 9C 10C 10C 9C 9C      3C,8H 2C,3G 3C,7H 2C,2G 9C 4C,9G 4C,9G 4C,9H 4C,9H 2C,3G 2C,8G 5G      PREEMERGENCE Morningglory 9C 9G 9H 8H 9C 8H 2C,9H 3C,7H 0 0 1C 0 9C 8G      3C,8H 2C,3H 1C 2G 2C,4H 1H Cocklebur 9H -- 8H 9H 9H 7H 9H 3H -- 0 0 0 9H      8H 3C,7H 2C,3H 3C,3G --  3C,7H 7H Velvetleaf 4C,9G 9G 9H 3C,9G 9G 8G 9G      3C,5H 5G 0 0 0 3C,9G 4C,9G 3C,8H 3C,5H 1H 0 0 2G Nutsedge 10E 3C,5G      4C,8G 2C,3G 10E 9G 5G 0 2G 0 3G 0 10E 8G 4G 0 0 0 0 0 Crabgrass 3C,7G      2C,4G 3C,5G 1C 2C,5G 3C,4G 4C,9G 3C,6G 0 0 -- 0 3C,3G 2G 2C,5G 0 0 0 6G      0 Giant Foxtail 4C,8H 3C,4G 4C,8G 2G 3C,6G 4G 4C,9H 3C,5G 0 0 0 0 4C,9H      3C,6G 3C,7G 2G 0 0 2C,7G 0 Barnyardgrass 4C,9H 2C,2H 3C,7H 0 4C,9H 3C,7G      3C,9H 3C,7H 1C 0 3G 0 5C,9H 4C,9H 3C,8H 2C,3G 0 0 9H 6G Cheatgrass 8G 2G      6G 0 0 0 8G 0 0 0 2G 0 5C,9H 9H 9H 3C,6G 0 0 8G 4G Wild Oats 4C,9H 6C,9G      4C,9H 4C,8G 3C,8G 3C,5G 6C,9H 3C,8G 0 0 0 0 4C,9H 3C,8H 3C,8G 3C,5G 0 0      2G 0 Wheat 9C 4C,9G 4C,8G 8G 5C,9H 7G 6C,9H 5G 0 0 0 0 5C,9H 3C,9G 3C,8G      5G 0 0 2G 0 Corn 3C,8H 1C,5G 4C,8H 2G 2C,8G 4G 10H 4C,9H 3C,7H 2C 2C,5G      0 3C,9H 2C,8G 3C,5G 2C,2G 2G 0 2G 0 Barley 5C,9G 9G 5C,9G 9G 9G 9G 9C      5C,9G 0 0 0 0 9G 9G 3C,9G 8G 2G 0 5G 0 Soybean 9H 9H 9H 3C,7H 3C,8H      3C,7H 9H 3C,7H 3C,3H 1C 3C,3H 0 9H 3C,6H 4C,6H 3C,4H 3C,3H 1C 7G 0 Rice      10E 10E 10E 3C,8H 10E 10E 10E 3C,9H 3C,6H 3C,3G 2C,7G 2G 10E 5C,9H 4C,9H      2C,6G 0 0 8H 7G Sorghum 10H 7C,9H 6C,9H 4C,8H 10H 10H 10H 6C,9H 3C,8G      3C,4G 3C,8G 2C 4C,9G 4C,8H 4C,9G 3C,6G 3C,3G 0 8G 2C,7G Sugar Beets 9C      9C 9C 4C,8H 4C,9G 3C,8G 10C 4C,9G 3C,5G 7G 5H 3G 9G 8G 5C,9G 4C,8G 6G 3H      8G 0 Cotton 9G 8G 4C,8G 2G 9G 4C,9G 8G 1C 2C,4G 1C 2G 0 9G 9G 8G 2C,6G      2C,3G 0 5G 2G        Compound 43 Compound 44 Compound 45 Compound 46 Compound 47 Compound      48 Compound 49 Compound 50 Compound 51 Compound 52 Rate kg/ha 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01       0.05 0.01  0.05 0.01        POSTEMERGENCE Morningglory 3C,8H 3C,7H 3C,7H 3C,3H 4C,9H 2C,5G 10C 10C      9C 4C,9H 4C,9H 2C,2H 4C,8G 2C,5G 2C,5H 0 4C,8H 1C 5C,9G 4C,9H Cocklebur      3G 0 2C,5G 2C 4C,9H 1C 10C 8H 7H 2G 1H 1H 4C,9H 5G 0 0 3C,6G 0 4C,9H      3C,4G Velvetleaf 7G 2C,5G 3C,6H 0 3C,7H 3C,3G 10C 9C 5C,9G 3C,8G 3C,7H      3G 3C,8H 3H 2C,5G 0 2G 0 3C,8H 3C,4G Nutsedge 0 0 0 0 3G 0 2C,9G 4C,8G      7G 3G 4G 0 5G 0 0 0 8G 0 9G 2C,7G Crabgrass 3G 0 0 0 2G 0 7G 5G 4G 0 0 0      0 0 0 0 2C,2G 0 3C,7G 2C Giant Foxtail 2G 0 1C 0 2G 0 5C,9G 3C,8G 5G 2G      0 0 3C,6G 0 2C,4G 0 6C,9H 3C,7H 9C 4C,8G Barnyardgrass 4G 3G 3C,7H 2C,4G      3C,9H 2C,5H 10C 5C,9G 3C,9H 3C,8H 3C,7H 1H 3C,8H 3H 3C,7H 0 9C 3C,8H 9C      9H Cheatgrass 8G 7G 0 0 3G 0 9G 8G 2C,6G 4G 2G 0 0 0 0 0 8G 0 3C,8G 5G      Wild Oats 4C,9G 5C,9G 0 0 2G 0 2C,9G 9G 3C,8G 3G 2G 0 0 0 0 0 4C,9G 0      4C,9G 3C,7G Wheat 9G 9G 0 0 2G 0 5C,9G 9G 8G 2G 2G 0 2G 0 0 0 8G 2G 8G      4G Corn 0 0 3C,7G 0 2C,6G 0 2C,9G 9H 3C,8H 2G 1H 0 1H 0 2G 0 4C,9H 2C,5G      3C,8H 0 Barley 9G 9G 2C 0 0 0 3C,9G 9G 3C,8G 4G 2G 0 1C 0 0 0 3G 0 3C,7G      2G Soybean 3H,8G 2H,5G 2C,7H 3H 3C,8G 2C,6H 9C 5C,9G 4C,9G 3C,8G 2C,7G      2H 2H 1H 0 0 3C,7H 2C,5G 4C,9G 2C,8H Rice 4C,9G 4C,9G 4C,9G 4G 5C,9G 5G      9C 9C 4C,9G 4C,9G 4C,9G 2G 4C,9G 4C,9G 6G 0 9C 5C,9G 9C 4C,9G Sorghum      4C,8G 2C,5G 5C,9H 5G 4C,9H 2C,8G 9C 5C,9G 4C,9G 4C,9G 4C,8G 6G 4C,9G      4C,9H 8G 4G 9C 4C,9H 9C 5C,9G Sugar Beets 3C,7G 2C,5G 3C,7H 3C,6G 5C,9G      3C,7H 10C 9C 9C 9C 4C,8H 2C,6G 3C,8H 2C,5G 3C,7G 0 9C 3C,7H 9C 4C,8H      Cotton 5G 0 3C,6G 1C 3C,8H 2C,4G 10C 2C,8G 8H 3C,8G 6H 0 7G 3G 2G 0 8H      7H 4C,9G 3C,8H PREEMERGENCE Morningglory 3H 0 2C 5G 4H 4H 9G 9G 9G 7G 2G      3G 8G 7G 0 0 5G 7G 8G 0 Cocklebur 8G 0 1H 0 6H 4H 9H 8G 8H -- 0 -- 9H 7H      8G -- 4H -- 7H 0 Velvetleaf 0 0 7G 0 2G 3G 9C 9G 4C,9G 7H 0 -- 3H 0 7G      -- 0 5G 5G 0 Nutsedge 0 0 0 0 0 0 4C,9G 0 4G 0 0 0 4G 0 0 0 0 0 5G 0      Crabgrass 0 0 0 0 0 0 3G 0 2G 0 0 0 0 0 0 0 0 0 0 0 Giant Foxtail 5G 0      3G 0 0 0 9H 7G 8G 2C 0 0 3C,4G 2G 0 0 4G 2G 6G 2G Barnyardgrass 0 0 3G 0      4G 0 9H 3C,9H 8H 2C 0 0 3C,8H 2G 0 0 2G 2G 5G 0 Cheatgrass 7G 3G 0 0 0 0      7G 3G 6G 0 0 0 0 0 0 0 2G 0 5G 0 Wild Oats 2C,6G 0 0 0 0 0 4C,9H 8H      2C,8G 2G 0 0 2G 0 0 0 0 0 2G 0 Wheat 6G 0 0 0 0 0 10H 3C,9H 8G 3G 0 0 3G      0 0 0 2G 0 7G 0 Corn 2C,6G 0 3C,7H 0 3C,8H 0 10H 3C,9H 2C,9G 2C,6G 0 0      4G 0 0 0 2C,8G 0 3C,8H 2G Barley 9G 7G 0 0 0 0 9G 9H 9G 2C,7G 2G 0 8G 0      0 0 6G 0 8G 3G Soybean 1C 0 0 0 2C,2H 0 9H 8H 3C,7H 7H 2C 0 4G 0 0 0      2C,5G 1H 8H 5H Rice 9H 4G 3C,8H 2C,4G 3C,7H 0 10E 10E 5C,9H 6G 0 3G      3C,8H 4G 2C 0 9H 2G 9H 5H Sorghum 3C,6H 0 3C,8H 2C 3C,8G 2C,4G 10H 5C,9H      5C,9H 2C,8G 2C -- 10H 3C,BH 2C,5G 0 2C,9H 2C,5G 3C,9H 3C,8G Sugar Beets      9G 2G 7G 5G 4G 4G 5C,9G 5C,9G 4C,9G 7G -- 2G 3C,8G 8G 4G 0 5G 5G 9G 8G      Cotton 0 0 2C 0 5G 2C 9G 9G 9G 2C,5G 2G -- 2C,7G 1C 0 0 7G 0 2C,7G      2G      Compound 53 Compound 54 Compound 55 Compound 56 Compound 57      Compound 58 Compound 59 Compound 60 Compound 61 Compound 62 Compound 63      Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE Morningglory 9C 10C 10C 10C 10C 8C 10C 10C 10C 2C,8G      1C,7G 0 10C 10C 3C,8G 1C, 1C,1H 0 0 0 10C 4C,8G                 1H      Cocklebur 9C 9C 10C 10C 10C 9C 10C 4C,9G 10C 10C 0 0 10C 10C 2C,8G 2H 3H      0 0 0 4C,9H 3C,7H Velvetleaf 9C 9C 10C 9C 10C 9C 10C 3C,8G 10C 2C,9H 2G      0 10C 9C 3C,9G 4G 4H 0 0 0 4C,8H 3C,7H Nutsedge 9C 9C 9C 5C,9G 9C 9G      5C,9G 4C,9G 5C,9G 2C,9G 0 0 10C 10C 2C,5G 0 0 0 0 0 9G 2C,8G Crabgrass      8G 3G 6G 3G 3C,6G 2C,5G 6G 2G 7G 0 0 0 3C,9G 7G 0 0 0 0 0 0 3C,6G 5G      Giant Foxtail 9C 3C,8G 5C,9G 3C,9G 9C 3C,8G 4C,9G 7G 3C,9G 2C,7G 0 0 9C      9C 3C,8G 4G 5G 2G 2G 0 9C 2C,8G Barnyardgrass 9C 9C 10C 9C 9C 10C 9C 9H      2C,9G 2C,5H 0 0 9C 9C 3C,7H 2H 2C,5G 3G 2C,5G 0 9C 3C,9G Cheatgrass 9C      9G 9C 4C,9G 9C 5C,9G 4C,9G 9G 8C 2C,9G 2G 0 9C 10C 9G 3G 6G 0 6G 0 5C,9G      9G Wild Oats 2G 0 3C,5G 0 5C,9G 3C,3G 3G 0 2C,9G 2C,6G 0 0 9C 5C,9G      2C,7G 0 2C,5G 2G 2C,5G 0 3C,8G 2C,5G Wheat 9G 7G 3C,9G 9G 9G 9G 8G 3G      1C,6G 0 0 0 9C 4C,9G 9G 0 9G 8G 6G 0 9G 7G Corn 3H 0 2H 0 2H 0 0 0 1C,8H      3C,8H 0 0 9C 10C 3C,8H 0 2C,7G 3G 3G 0 5C,9G 3C,9G Barley 3C,9G 2C,6G 8G      5G 9G 3C,7G 2G 0 5C,9G 3C,9G 0 0 9C 5C,9G 2C,4G 0 2C,5G 3G 4G 0 9G 8G      Soybean 9C 5C,9G 9C 4C,9G 5C,9G 4C,8G 3C,8G 3C,5H 5C,8H 2C,6H 0 0 9C 9C      3G 2H 2C,6H 3H 0 0 3C,8H 3C,4H Rice 9C 5C,9G 9C 9C 5C,9G 5C,9G 9C 5C,9G      5C,9G 2C,8G 3C 0 9C 9C 5C,9G 0 3C,9G 3G 7G 0 6C,9G 4C,9G Sorghum 9C 10C      9C 9C 5C,9G 5C,9G 9C 5C,9G 3C,9G 3C,9G 1C,5G 0 9C 9C 2C,9G 5G 4G 2G 7G 0      3C,9G 4C,9G Sugar Beets 9C 10C 10C 9C 9C 9C 10C 9C 9C 10C 2C,4H 0 9C 9C      9C 3G 2C,4G 0 2C 0 9C 5C,9G Cotton 9C 9C 9C 5C,9G 9G 9G 10C 3C,8G 10C      2C,8H 2G 0 10C 9C 3C,8G 0 0 0 0 0 4C,9G 3C,8H PREEMERGENCE Morningglory      9C 9G 9G 9G 9G 8G 9G 9G 8H 3C,7H 0 0 9G 9G 0 0 0 0 0 0 3H 0 Cocklebur 9H      -- 9H 9H 9H 9H 9H 5H 2C,8H 2C,7H 0 0 9H 9H 2H 0 0 0 0 0 4G 1H Velvetleaf      9C 9C 5C,9G 5C,9G 4C,9G 8G 8H 6H 2C,7H 2C,5H 0 0 9C 3C,9G 0 0 0 0 0 0 0      0 Nutsedge 10E 10E 10E 10E 10E 9G 10E 4G 10E 9G 0 0 10E 10E 0 0 0 0 0 0      7G 0 Crabgrass 2G 0 3G 0 2G 0 2G 0 1C,5G 2C,4G 0 0 3C,7G 3G 0 0 0 0 0 0      3G 0 Giant Foxtail 9H 8H 9H 3C,8H 9H 3C,8G 3C,7G 6G 2C,7H 2C,6G 0 0      5C,9H 3C,7G 0 0 0 0 0 0 3G 2G Barnyardgrass 9H 9H 9H 9H 9H 3C,8H 9H 8H      2C,6H 2C,4H 0 05C,9H 4C,9H 0 0 0 0 0 0 4G 2G Cheatgrass 10H 9H 9H 10E 9H      8G 8H 6G 3C,9H 2C,9H 0 0 10E 9H 0 0 0 0 0 0 5G 0 Wild Oats 0 0 8G 2C,5G      8G 0 0 0 2C,6G 2C,6G 0 0 4C,9H 3C,6G 0 0 0 0 0 0 2C 0 Wheat 9H 7H 10H      4C,9H 9G 2G 8G 5G 4G 0 0 0 10H 4C,9H 0 0 0 0 0 0 3G 0 Corn 2C,7G 4G 7G      6G 3G 1C,2G 1C 0 2C,7G 3C,4G 0 0 5C,9H 4C,9H 0 0 0 0 0 0 3C,3G 0 Barley      9G 9G 9G 9G 9G 8G 4C,8G 5G 6G 6G 0 0 4C,9G 3C,9G 0 0 0 0 0 0 3C,9G 4G      Soybean 9H 9H 9H 3C,8H 3C,8H 2C,6G 7H 2H 2C,5G 1C,2G 0 0 9H 9H 0 0 0 0 0      0 1C 0 Rice 10E 10E 10E 10E 10E 9H 10E 8H 3C,9H 2C,8H 0 0 10E 10E 0 0 0      0 0 0 4C,8H 3G Sorghum 5C,9H 9H 10H 5C,9H 10H 9H 9H 5C,9H 2C,9H 2C,8H 0      0 10H 4C,9H 0 0 0 0 0 0 4C,9H 3C,5G Sugar Beets 9C 9C 9C 5C,9G 9G 9G      4C,9G 8G 9C 4C,8G 1C 0 5C,9G 4C,9G 0 0 0 0 0 0 7G 3C,5G Cotton 9G 9G      4C,9G 9G 9G 9G 9G 7G 2C,8G 2C,8G 0 0 9G 9G 0 0 0 0 0 0 3C,6G 5G

      CMPD 64* CMPD 65* CMPD 66 CMPD 67 CMPD 68 CMPD 69 CMPD 70 CMPD 71 CMPD      72 CMPD 73 PD 73 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.01 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE COTTON 0 0 0 0 10C 4C,9G 9C 4C,9H 4C,9G 4C,9H 4C,8G      4C,9H 3C,8H 0 4C,9H 3C,8H 9C 4C,9G 4C,9H 4C,9H MORNING GLORY 0 0 0 0 10C      10C 10C 10C 9C 5C,9G 10C 4C,9H 3C,8G 3C,7G 4C,9H 3C,8H 10C 4C,9G 10C 9C      COCKLEBUR 0 0 0 0 10C 10C 10C 9C 10C 5C,9G 9C 4C,9H 2G 0 4C,9H 2C,2H 10C      5C,9G 10C 4C,9G NUTSEDGE 0 0 0 0 6G,9G 5C,9G 5C,9G 4C,8G 5C,9G 7G 2C,8G      5G 0 0 4G 0 5C,9G 5C,9G 5C,9G 3C,9G CRABGRASS 0 0 0 0 2C,6G 4G 4G 3H 6G      3G 3H 2H 0 0 0 0 2H 0 0 2H BARNYARD GRASS 0 0 0 0 9C 9C 9C 9C 9C 5C,9H      9C 4C,9H 5C,9H 5G 5C,9H 9C 10C 9C 4C,9H 3C,7H WILD OATS 0 0 0 0 2G 0      2C,6G 2G 4C,9G 2C,3G 3G 0 4C,8G 2G 3C,8G 3G 5C,9G 3C,7G 6G,9G 2C,2G      WHEAT 0 0 0 0 9G 8G 9G 7G 9G 9G 6G 0 3C,8G 3G 3G 0 5C,9G 8G 4C,9G 2C,5G      CORN 0 0 0 0 4G 2G 0 0 2H 0 0 0 5C,9G 6G 6G 3G 4C,9G 4G 3C,5G 3G SOYBEAN      0 0 0 0 9C 9C 9C 5C,9G 4C,9G 5C,9G 5C,9G 3C,7H 4C,9G 3C,7H 4C,9G 3C,8G      9C 5C,9G 5C,9G 4C,9G RICE 0 0 0 0 9C 9C 9C 9C 9C 9C 9C 4C,9G 4C,9G 5G 8G      2C,5G 9C 5C,9G 5C,9G 3G SORGHUM 0 0 0 0 9C 9C 9C 5C,9G 9C 4C,9G 9C 4C,9G      3C,9H 4C,8H 5C,9H 3C,9H 10C 9C 9C 4C,9H CHEATGRASS 0 0 0 0 9C 4C,9G 9C      4C,9G 10C 4C,9G 4C,9G 4C,9G 3C,8G 2C,5G 3C,6G 4G 9C 9C 9C 4C,9G SUGAR      BEETS 0 0 0 0 9C 10C 10C 9C 10C 9C 9C 5C,9G 3C,7H 2C,2H 4C,8H 3C,6H 10C      10C 10C 3C,8H VELVETLEAF 0 0 0 0 10C 9C 10C 4C,9H 9C 5C,9G 3C,7H 2C 0 0      4C,6H 0 10C 10C 10C 4C,9H GIANT FOXTAIL 0 0 0 0 9C 4C,9G 9C 5C,9G 9C      5C,9G 5C,9G 7G 4C,9H 3G 4C,9H 3C,7G 3C,8G 3G 3C,7H 2G BARLEY 0 0 0 0 7G      3G 3G 0 2G 0 0 0 2G 0 5G 0 9G 4G 3G 0 PREEMERGENCE COTTON 0 0 0 0 4C,9G      2C,8G 3C,7H 6G 3C,8H 2C 2C,6G 2C 0 0 0 0 8G 3G 2G 0 MORNING GLORY 0 0 0      0 9H 2C,9H 8H 2C,6H 9G 3H 8G 2C,2H 2G 0 3H 0 7H 4H 2G 0 COCKLEBUR 0 0 0      0 9H 7H 3C,7H 2C,5G 3C,7H 1C 3C,7H 2C 0 0 0  8H 2C 0 0 NUTSEDGE 0 0 0 0      10E 9G 5G 5G 10E 0 2C,5G 3G 0 0 0 0 10E 3C,7G 5G 0 CRABGRASS 0 0 0 0 4G      0 0 0 2G 0 2G 0 0 0 0 0 0 0 0 0 BARNYARD GRASS 0 0 0 0 9H 3C,9H 3C,9H 2G      3C,9H 1C 3C,7H 0 2C,5G 0 0 0 9H 2C,5G 3C,7G 0 WILD OATS 0 0 0 0 2G 0 2C      0 2C,4G 0 0 0 0 0 0 0 3C,7G 2G 3C,5G 0 WHEAT 0 0 0 0 4C,9H 2C,8H 3C,8H      5G 8G 6G 5G 0 0 0 0 0 8G 2G 7G 0 CORN 0 0 0 0 4C,8H 6G 4G 0 2G 2G 0 0 3G      0 2C,4G 0 3C,8H 3G 2G 0 SOYBEAN 0 0 0 0 9H 9H 9H 3C,7H 3C,9H 3C,6H 3C,7H      2C,4G 0 0 0 0 7H 3C,5H 3C,4H 1C,1H RICE 0 0 0 0 9H 9H 3C,9H 3C,7G 5C,9H      3C,7G 9H 7G 6G 0 0 0 10E 9H 9H 3G SORGHUM 0 0 0 0 10H 5C,9H 3C,9H 3C,9H      5C,9H 3C,7H 3C,9H 2C,8H 2G 0 3C,5G 0 10H 9H 9H 3C,3G CHEATGRASS 0 0 0 0      9H 8G 9G 8G 3C,9G 8G 9H 8G 5G 0 0 0 9H 3C,9H 9H 0 SUGAR BEETS 0 0 0 0      5C,9G 4C,9G 9G 7G 4C,8H 3C,8G 3C,7H 2C,5G 2G 0 3G 0 9G 9G 7G 1H VELVETLEA      F 0 0 0 0 5C,9G 2C,7G 3C,7H 0 3C,5H 1C 2H 2C,2G 1C 0 0 0 5H 0 2G 0 GIANT      FOXTAIL 0 0 0 0 9H 2C,8H 3C,8G 3G 3C,9H 2C,5G 9H 3C,5G 2C,2G 0 2G 0      3C,8H 2C,2G 3C,3G 0 BARLEY 0 0 0 0 9G 2C,6G 2G 2G 3C,7G 0 2G 0 0 0 0 0      8G 5G 2G 0      *It is noted that Compounds 64 and 65 were inactive at the levels tested.      However, it is believed that at higher levels, herbicidal activity would      be present.     CMPD 74 CMPD 75 CMPD 76 CMPD 77 CMPD 78 CMPD 79 CMPD 80 CMPD 81 CMPD 82      CMPD 83 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE COTTON 9G 9G 9G 9G 9C 9C 9C 5C,9G 3C,9G 9G 10C 9C 9C      2C,8H 9C 2C,8H 9C 5C,9G 9C 9C MORNING GLORY 4C,9G 3C,8H 9C 2C,9G 10C 7G      10C 10C 10C 3C,8H 10C 9C 3C,8H 4C,8H 10C 4C,8H 10C 10C 10C 10C COCKLEBUR      4C,9G 3C,8H 5C,9G 3C,8H 10C 10C 10C 10C 9C 3C,8H 10C 9C 5C,9H 4C,8H 10C      10C 10C 10C 10C 10C NUTSEDGE 4C,9G 2C,5G 3C,9G 5C,9G 10C 10C 10C 5C,9G      4C,9G 2C,9G 10C 4C,9G 8G 6G 3C,8G 0 9C 9C 9C 4C,8G CRABGRASS 0 0 0 0      2C,7G 7G 2C,6G 3G 6G 0 6G 2G 5G 0 2C,5G 0 6C,9G 4C,6G 4C,8G 4G BARNYARD      GRASS 3C,8H 4G 3C,8H 3C,5H 10C 9C 9C 9C 9C 4C,9H 3C,9G 2C,8G 9C 2C,9H      10C 3C,9G 9C 9C 9C 9C WILD OATS 9C 3C,7G 2C,3G 0 2C,9G 2C,6G 3C,9G 2C,7G      3C,9G 3C,9G 6G 2C,6G 3C,7G 2C,5G 5C,9G 3C,8G 9C 3C,9G 5C,9G 4C,9G WHEAT      4C,8G 3G 2C,3G 0 4C,9G 10C 2C,9G 9C 3C,9G 9G 2C,9G 9G 4G 0 2G 0 9C 3C,9G      6C,9G 4C,9G CORN 1C 0 0 0 6U,9C 3U,8G 4U,9G 2C,9G 3C,8H 1C,4G 3C,9G      2C,7H 6U,9C 3U,9G 6U,9C 3U,9C 10C 3C,9G 9C 9C SOYBEAN 4C,9G 4C,9G 3C,8G      4H 10C 9C 6C,9G 5C,9G 5C,9G 3C,9G 3C,8H 2H,7G 5C,9H 4C,8H 4C,9G 3C,9G      5C,9G 5C,9G 9C 4C,9G RICE 5C,9G 2C,8G 3C,8G 2G 6C,9G 9C 9C 5C,9G 9C      3C,9G 5C,9G 2C,9G 9C 8G 4C,9G 8G 6C,9G 9C 9C 9C SORGHUM 9H 2C,5G 10C 9G      9G 3U,9G 9C 9C 10C 2C,9G 5C,9G 5C,9G 9C 2C,9G 9C 9C 9C 9C 9C 9C CHEATGRAS      S 4C,9G 2C,7G 3C,8G 2C,5G 10C 10C 10C 9C 10C 5C,9G 9C 9G 9G 5G 3C,9G 6G      9C 9C 9C 9C SUGAR BEETS 3C,8H 3C,8G 4C,9G 1C,2G 10C 10C 10C 10C 10C 10C      10C 10C 10C 5C,9H 10C 3C,9H 9C 10C 10C 10C VELVETLEAF 9C 3C,7H 5C,9G      3C,5G 10C 10C 10C 9C 10C 5C,9H 10C 5C,9H 5C,9H 3C,6H 9C 3C,8H 10C 9C 10C      9C GIANT FOXTAIL 3G 2G 1C 0 4C,9G 2C,9G 9C 4C,9G 10C 3C,9G 9G 6G 9C      2C,8G 10C 9C 10C 9C 10C 10C BARLEY 3C,7G 0 0 0 3C,9G 9G 9C 9G 4C,9G 9G      9G 9G 2C,6G 5G 6G 2G 4C,9G 4C,9G 5C,9G 3C,9G PREEMERGENCE COTTON 1C 0 2G      0 9G 9G 3C,9G 8G 9G 5G 9G 8G 9G 0 3C,9G 0 9G 9G 9G 9G MORNING GLORY 0 0      3C,8H 6G 9G 8G 9G 9G 9G 2C,7H 9G 9G 2C,8H 2C,6H 9G 2C,4H 9G 9G 9G 9G      COCKLEBUR 0 0 2C,2H 1C 9H 9H 9H 8H 9H 2C,3H 9  8H 2C,4G 9H 1C,2G 9G 9H      9H 9H NUTSEDGE 10E 0 3C,8G 0 10E 10E 10E 9G 9G 6G 10E 9G 4C,9G 4G 9G 2G      10E 10E 10E 10E CRABGRASS 0 0 0 0 7G 6G 3C,8G 2C,7G 10E 0 5G 0 3C,7H 0      3C,7H 0 8G 7G 4C,8G 4C,8H BARNYARD GRASS 2G 0 3C,8H 0 9H 9H 9H 3C,9H      3C,9H 3G 3C,8H 2C,7H 5C,9H 5G 9H 0 9H 9H 9H 9H WILD OATS 0 0 0 0 7G 7G      3C,8G 2C,7G 2C,8H 2C,7G 2C,8G 0 7G 4G 8G 2C,4G 3C,9G 4C,8G 6C,9H 4C,8G      WHEAT 0 0 0 0 3C,9G 2C,9G 10C 4C,9H 10H 8H 3C,9H 7G 5G 0 6G 0 4C,9H      3C,9G 5C,9H 8G CORN 0 0 0 0 9G 9G 10C 9G 9G 2C,7G 9G 2C,7G 9G 8G 9G 9G      2U,9G 2U,9H 9H 9G SOYBEAN 1H 0 2C 0 9H 9H 9H 8H 9H 2C,6C 3C,8H 2C,7G      4C,8H 3C,7H 9H 2C,6G 9H 9H 9H 9H RICE 7H 0 7H 6H 10E 10E 10E 10H 10E 9H      10E 10E 9H 3C,8H 10E 2C,8H 10E 10E 10E 10E SORGHUM 3C,7G 0 9H 3C,7G 10C      10C 10E 10E 9H 9H 10H 10H 10H 9H 10E 3C,8H 9H 4C,9H 10E 10H CHEATGRASS      5G 0 8H 0 10E 10H 10H 9H 9H 8H 9H 9H 9H 1C,4G 9H 4G 9H 9H 9H 9H SUGAR      BEETS 5H 0 5H 2G 9G 9G 5C,9G 5C,9G 4C,9G 3C,9G 3C,9G 2C,6G 4C,9G 5G 9G      2C,6G 9G 9G 9G 9G VELVETLEAF 2G 0 2G 4G 9G 9G 3C,9G 3C,9G 2C,8G 2C,7H 9G      9G 2C,7H 3C 3C,8H 2C 4C,9G 8G 5C,9G 8G GIANT FOXTAIL 0 0 2C 0 9H 8G      3C,9H 3C,9H 2C,9H 2C,5H 8G 5G 7G 2G 9H 5G 9H 9H 9H 9H BARLEY 0 0 0 0 9G      9G 10C 9G 9C 8G 9G 9G 7G 6G 9G 6G 3C,9G 2C,9G 4C,9H 4C,9H        CMPD 84 CMPD 85 CMPD 86 CMPD 87 CMPD 88 CMPD 89 CMPD 90 CMPD 91 CMPD      92 CMPD 93 RATE RATE = KG/HA 0.05 0.01 0.5 0.01 0.05 0.01 0.5 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05  0.01 0.05 0.01        POSTEMERGENCE COTTON 9C 4C,9G 9C 4C,9G 4C,9H 3C,4G 4C,9H 4C,8H -- --      -- -- -- -- -- -- -- -- -- -- MORNING GLORY 10C 10C 10C 10C 3C,8H 3C,6H      5C,9G 3C,9G 2C 0 3C,8H 2C,7G 2C,4H 0 2C,4G 2G 2C,7G 2H 3C,8H 2C,6H      COCKLEBUR 10C 10C 10C 10C 4G 0 9C 3C,8H 4C,9H 3C,8H 5C,9H 4C,8H 4C,9H 0      3C,8H 1C,5G 4C,8H 2C,7H 3C,8H 2C NUTSEDGE 9C 9C 9C 5C,9G 3C,5G 0 4C,9G      3C,5G 2C,6G 6G 2C,8G 3G 0 0 0 0 0 0 0 0 CRABGRASS 4C,9G 7G 3C,6G 2G      3C,5G 0 5C,9G 4G 0 0 0 0 0 0 0 0 0 0 0 0 BARNYARD GRASS 9C 9C 10C 9C 9C      5C,9H 9C 9C 3C,6G 4G 3C,8H 0 2G 0 0 0 3C,6H 0 2C,7G 3G WILD OATS 9C      4C,9G 5C,9G 4C,9G 5C,9G 5C,9G 6C,9G 4C,9G 2C,2G 2G 2C,5G 2C,3G 3C,5G 2G      0 0 0 0 4G 0 WHEAT 9C 4C,9G 4C,9G 8G 5C,9G 4C,9G 3C,9G 3C,7G 6G 3G 3C,9G      2C,7G 2C,4G 2G 0 0 0 0 2G 0 CORN 6G,9G 3C,9G 5C,9G 9G 9C 9G 9C 9C 2C,6H      2G 3C,8H 3G 0 0 0 0 3C,7H 0 2C,7H 0 SOYBEAN 6C,9G 4C,9G 5C,9G 3C,9G      4C,9G 4C,9G 5C,9G 4C,9G 4C,9G 4C,8G 5C,9G 3C,9H 3C,7H 0 0 0 3C,9G 2C,6H      3C,8H 2C,7H RICE 9C 9C 9C 5C,9G 5C,9G 3C,8G 4C,9G 4C,9G 3C,8G 7G 2C,8G      2C,5G 4G 0 2G 0 4G 0 4G 3G SORGHUM 9C 5C,9G 9C 9C 5C,9G 3C,8H 9C 9C      3C,8H 6G 3C,9H 2C,8H 2C,7H 0 3G 0 2C,8H 1C,5G 2C,8H 2C,7G CHEATGRASS 9C      9C 9C 3C,9G 4C,8G 4C,8G 6C,9G 2C,9G 2C,9G 2C,8G 9G 2C,9G 9G 4G 0 0 7G 0      5G 0 SUGAR BEETS 10C 10C 10C 9C 10C 3C,7H 10C 5C,9G 10C 1C,3G 3C,9G 0      2C,5G 0 0 0 4C,8G 2C,7G 5C,8G 3C,7G VELVETLEAF 10C 10C 10C 9C 3C,5H 1C      9C 3C,4H 3C,9H 2C,7G 4C,9G 2C,7G 2C,7G 5G 0 0 2C,4H 2G 3C,7H 2C,2H GIANT      FOXTAIL 9C 9C 9C 9C 9C 3C,7H 10C 9C 4G 0 5G 2G 2G 0 0 0 4G 0 6G 2G      BARLEY 9C 4C,9G 4C,9G 3C,7G 2C 0 3C,6G 0 5G 0 5G 5G 5G 0 0 0 2G 0 0 0      PREEMERGENCE COTTON 9G 9G 9G 9G 4C,8G 7G 5G 4G 0 0 0 0 0 0 0 0 0 0 2G 0      MORNING GLORY 9G 9G 9G 9G 8H 2H 9G 8H 0 0 2C,3G 0 0 0 0 0 0 0 0 0      COCKLEBUR 9H -- 9H 9H 4G -- 8H 8G -- 2G 3C,8H 0 0 0 0 -- 2C 0 0 --      NUTSEDGE 10E 10E 10E 10E 3G 5G 7G 4G 4G 0 2G 0 0 0 0 0 0 0 0 0 CRABGRASS      10E 2G 8H 0 9G 0 5G -- 2G 0 2G 0 0 0 0 0 9G 8G 0 0 BARNYARD GRASS 9H 9H      9H 9H 3C,9H 3G 9H 7H 0 0 2G 0 0 0 0 0 0 0 0 0 WILD OATS 6C,9H 4C,9G      3C,9H 3C,5G 2C,3G 0 2C,4G 0 0 0 2G 0 0 0 0 0 0 0 0 0 WHEAT 10H 4C,8G      2C,9H 3C,8H 3G 0 5G 0 7G 0 4G 0 0 0 0 0 0 0 0 0 CORN 9H 9H 9H 9H 3C,9H      4C,8G 9H 3C,9G 2C,3H 0 3C,6G 2G 0 0 0 0 0 0 1C 0 SOYBEAN 9H 9H 9H 9H 9H      2H 9H 3C,6H 2C,3G 0 3C,5G 1C,3G 0 0 0 0 1C,2G 0 2C,4G 0 RICE 10E 10E 10E      10E 9H 7H 9H 5G 3C,8H 0 2C,3H 0 0 0 0 0 0 0 0 0 SORGHUM 10E 10E 10E 10H      3C,9H 4C,9G 10H 4C,9H 2C,9H 0 3C,7H 2C,3H 0 0 0 0 2C,5G 1C 3C,7H 0      CHEATGRASS 9H 9H 9H 8H 7G 6G 9H 5G 8G 2G 8H 3G 0 0 0 0 0 0 0 0 SUGAR      BEETS 9C 9G 3C,9G 9G 4C,8G 4H 4C,9G 3G 6G 0 2C,4G 4G 0 0 0 0 4G 2G 2H 0      VELVETLEAF 4C,9G 4C,9G 9C 7H 2C 2G 7H 3G 0 0 2C,3H 0 0 0 0 0 0 0 2G 0      GIANT FOXTAIL 9H 9H 9H 10H 3C,8H 3G 4C,9H 4C,8G 0 0 3G 0 0 0 0 0 0 0 0 0      BARLEY 9H 9H 3C,9H 4C,9H 4C,8G 0 9G 0 8G 0 2C,7H 2G 0 0 0 0 0 0 0      0        CMPD 94 CMPD 95 CMPD 96 CMPD 97 CMPD 98 CMPD 99 CMPD 100 CMPD      101 CMPD 102 CMPD 103 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 4C,9G 1C,5G 0 0 4C,9G 4C,9G 9C 4C,9H      4C,9G 3C,9H 9C 3C,9G 4C,9H 2C,7G 3C,9G 2C,4G 4C,9H 3C,8H 9C 4C,9H      MORNING GLORY 5C,9G 5C,9G 0 0 10C 10C 10C 10C 9C 9C 10C 10C 3C,5G 2H      4C,9G 3C,8H 10C 5C,9G 10C 4C,9G COCKLEBUR 4C,9H 3C,8H 4G 3G 10C 10C 10C      4G 10C 5C,9G 10C 10C 3C,9H 6G 5C,9G 3C,8H 9C 4C,9G 10C 10C NUTSEDGE 6G 0      0 0 5C,9G 3C,8G 10C 9C 4C,9G 4C,8G 10C 9C 3C,8G 3G 3C,8G 0 5C,9G 4C,9G      9C 5C,9G CRABGRASS 0 0 0 0 7G 2G 4C,8G 5G 1C 0 2G 0 0 0 2G 0 0 0 0 0      BARNYARD GRASS 4C,9H 2C,7H 0 0 10C 10C 10C 10C 9C 3C,8H 3C,9H 1C,4H 2H 0      2C,5H 0 3C,8H 1H 3C,9H 7H WILD OATS 2G 0 0 0 9G 2C,5G 4C,9G 3C,6G 5G 0      3C,7G 0 0 0 2C,5G 0 3C,6G 3G 2C,5G 2G WHEAT 4G 3G 0 0 9G 2C,6G 3C,9G 8G      2C,7G 3G 2C,8G 7G 0 0 2C,7G 3G 5C,9G 7G 7G 2G CORN 0 0 0 0 2G 0 2C,7G 2G      0 0 10C 10C 3G 0 3C,9H 4G 4C,9H 2C,7G 1H 0 SOYBEAN 4C,9G 3C,7H 0 0 4C,9G      4C,9G 9C 9C 4C,9G 4C,9G 9C 4C,9G 3H 0 3C,7H 2C,5H 5C,9G 4C,9G 3C,9G 8H      RICE 2C,5G 0 0 0 9C 4C,8G 9C 5C,9G 4C,9G 5G 4C,9G 8G 2G 0 7G 0 8G 0      5C,9G 7G SORGHUM 4C,9G 3C,9G 0 0 9C 9C 10C 10C 10C 9C 5C,9G 10C 4C,9G 7H      2C,9G 3C,8H 9C 4C,9H 9C 9C CHEATGRASS 10C 4G 0 0 2C,5G 0 4C,9G 6G 3C,7G      0 9C 3C,8G 2C,5G 0 8G 2G 4C,9G 3C,7G 8G 3G SUGAR BEETS 9C 2C,3H 0 0      4C,9G 2C,3G 10C 10C 10C 4C,8G 10C 9C 3C,5G 1C 10C 3C,7G 9C 3C,7G 10C 10C      VELVETLEAF 4C,9H 2C,4H 3G 2G 10C 5C,9G 10C 10C 4C,9H 4C,8H 10C 10C 3C,8H      3C,7G 4C,8H 3C,7H 9C 4C,9G 10C 5C,9G GIANT FOXTAIL 2C,7G 2G 0 0 4C,9G      3C,9G 5C,9G 6G 3C,8G 2C,6G 2C,7G 3G 2G 0 2C,G 2G 4C,9G 4G 6G 3G BARLEY      2G 0 0 0 9G 6G 9G 5G 2C,2G 0 9C 8G 2G 0 2C,6G 0 2C,9G 2C,6G 7G 2G      PREEMERGENCE COTTON 5G 0 0 0 2C,8G 6G 9G 9G 3C,8G 2C,4G 7H 6G 1C 0 0 0      8G 2C,3G 9G 2G MORNING GLORY 3C,8G 5G 0 0 9G 8G 9G 9G 9H 4H 9G 6H 2G 0      3C,4H 0 8H 3C,4H 9G 6H COCKLEBUR 2C,4H 0 0 -- 9H 3C,8H 3G 5G 2C,7G 0 8H      8H 5G 0 2C,2G 0 8H 3C,3H 9G 9H NUTSEDGE 0 0 10E 4G 10E 3C,9G 10E 10E 10E      10E 10E 9G 9G 0 3G 0 10E 0 10E 10E CRABGRASS 2C,5G 2G 0 0 2C,7G 5G 10E      2C,5G 2C,3G 2G 10E 6G 5G 0 0 0 0 0 2G 0 BARNYARD GRASS 4C,9H 5G 0 0 9H      2C,7H 9H 9H 9H 3C,7H 7H 0 0 0 0 0 6H 2G 8H 4G WILD OATS 0 0 0 0 7G 0      3C,8G 2C,6G 2C 0 7G 5G 0 0 0 0 3C,8G 0 5G 0 WHEAT 7G 0 0 0 9G 9G 10H 9H      7G 0 9G 8G 0 0 5G 0 9H 3C,8G 7G 2G CORN 2C,3G 0 0 0 4C,7G 1C,3G 3C,8G 3G      0 0 3C,9G 7G 0 0 0 0 3C,9H 3C,6G 0 0 SOYBEAN 2C,3G 0 0 0 9G 3C,7H 9H 9H      3C,8H 3C,4G 3C,8H 6H 2C 0 2C 0 3C,6H 3C,5H 8H 3C,7H RICE 5G 0 6G 0 10E      8G 10E 9H 10H 3C,7G 9H 9H 6G 0 4G 0 8H 0 10H 3C,7G SORGHUM 4C,9H 3C,8H      4G 0 10E 6C,9G 10E 5C,9H 10H 10H 10H 10H 3C,8G 2G 2C,6G 0 10H 4C,8H 10E      9H CHEATGRASS 8G 0 0 0 7G 7G 9G 7G 9G 2G 9G 8H 0 0 5G 0 8G 7G 8G 5G      SUGAR BEETS 4C,8G 5G 6G 0 4C,9G 8G 9G 9G 4C,9G 8H 4C,9G 6H 2H 2G 7G 0      4C,9G 4C,8H 9G 9G VELVETLEAF 3G 0 0 0 4C,9G 2C,8G 5C,9G 7H 2C,7H 2C,3H      4C,9G 8G 3H 0 3C,5G 0 4C,8H 1H 7H 1H GIANT FOXTAIL 3C,8H 4G 0 0 2C,9G 8G      2C,7G 2C,5G 2C,9H 3G 4G 0 0 0 3G 0 8G 2G 7G 1C BARLEY 3G 0 0 0 9G 7G 9G      9G 2C,8G 7G 9G 8G 0 0 5G 0 9G 3C,7G 9G 6G        CMPD 104 CMPD 105 CMPD 106 CMPD 107 CMPD 108 CMPD 109 CMPD 110 CMPD      111 CMPD 112 CMPD 113 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 9C 4C,9G 5C,9G 4C,9H 4C,9G 4C,9H 10C      5C,9G 5C,9G 10C 9C 5C,9G 6C,9G 3C,9G 4C,8H 3C,7H 4C,9H 4C,8G 1H 0      MORNING GLORY 10C 10C 10C 3C,8G 10C 0 10C 2H 10C 9C 2C,7G 5G 10C 10C      4C,8H 3C,7G 10C 4C,9G 0 0 COCKLEBUR 10C 10C 9C 10C 10C 10C 10C 10C 10C      10C 10C 10C 10C 10C 4C,9H 2C,4G 10C 4C,8H 1H 0 NUTSEDGE 9C 9C 5C,9G 8G      9C 4C,8G 5C,9G 3C,8G 3C,8G 2C,7G 4C,9G 6C,9G 5C,9G 3C,8G 2C,4G 0 3C,9G 0      0 0 CRABGRASS 3G 0 3G 0 5G 0 3C,7G 2G 3C,7G 5G 3C,6G 5G 3C,5G 3G 0 0 2G      0 2G 0 BARNYARD GRASS 10C 9C 9C 3C,8H 10C 5C,9H 10C 9C 9C 9C 10C 9C 9C      4C,9H 3C,7H 2C,5H 9C 3C,7G 5C,9H 3C,6G WILD OATS 3C,9G 3C,7G 3C,7G 3C,5G      3C,9G 3C,8G 3C,9G 3C,8G 4C,9G 3C,7G 4C,9G 4C,9G 3C,9G 2C,3G 0 0 3C,5G 0      3C,5G 2G WHEAT 2C,9G 3C,9G 6C,9G 2C,8G 3C,9G 5C,9G 5C,9G 3C,9G 9C 5C,9G      9C 2C,9G 3C,9G 3G 0 0 4G 0 9C 8G CORN 0 0 0 0 0 0 9C 3C,9G 4C,9G 4C,9H      3C,8H 3C,7H 3C,8H 2G 3C,7G 0 9G 3C,6G 2C,9G 2C,5H SOYBEAN 9C 9C 9C 5C,9G      5C,9G 5C,9G 9C 5C,9G 5C,9G 9C 9C 4C,9G 4C,9G 3C,6G 4C,9G 3C,8G 4C,9G      4C,8G 2G 0 RICE 9C 3C,9G 5C,9G 4C,9G 5C,9G 5C,9G 9C 5C,9G 9C 9C 9C 9C 9C      4C,9G 3G 0 4G 0 9C 8G SORGHUM 9C 9C 9C 5C,9G 10C 3C,9H 9C 9C 10C 9C 9C      9C 9C 4C,9H 3C,7H 0 3C,9G 3C,8H 4C,9G 3C,7H CHEATGRASS 7G 3G 7G 5G 5C,9G      5C,9H 10C 2C,8G 5C,9G 3C,8G 5C,9G 8G 4C,8G 6G 0 0 0 0 3C,9G 0 SUGAR      BEETS 10C 10C 10C 4C,9H 10C 10C 10C 9C 10C 10C 10C 9C 9C 9C 3C,5H 3C,8H      10C 4C,8H 3C,8G 3G VELVETLEAF 10C 10C 10C 4C,8G 9C 4C,9H 10C 9C 9C 10C      9C 4C,8H 9C 9C 3C,7H 0 4C,9G 3C,6H 4G 0 GIANT FOXTAIL 3C,7H 3C,6G 4C,8G      7G 4C,8G 3C,8G 5C,9G 3C,8G 5C,9G 4C,8G 4C,8G 2C,6G 3C,8G 3G 2G 0 3C,7G      2C,2G 3C,8H 2G BARLEY 3C,9G 3C,8G 8G 6G 2C,9G 3C,8G 4C,9G 9G 3C,9G 8G      4C,9G 2C,8G 9G 5G 0 0 3G 0 2C,9G 9G PREEMERGENCE COTTON 9H 5G 2C,8H 0      2C,4G 2G 9G 9G 3C,8G 7G 8H 3G 8G 7G 0 0 2G 0 0 0 MORNING GLORY 9G 2C,5G      3H 0 2C,5G 0 5G 2G 9H 3G 5G 1H 9G 7H 2C,3H 0 8G 0 0 0 COCKLEBUR -- 1H 8H      2H 2C,5G 3C,7H 9H 9H 9H 9H -- 3C,8H 9H 8H 0 -- 7H 2C,5G 0 -- NUTSEDGE 9G      10E 9G 0 8G 0 10E 10E 10E 4C,9G 10E 10E 10E 10E 10E 0 10E 0 0 0 CRABGRASS       4G 0 0 0 10H 0 8G 2C,5G 4C,8G 3C,7G 4C,8G 2C,2G 3C,5G 3G 2G 0 2G 0 2G 0      BARNYARD GRASS 9H 2G 4C,9H 0 0 0 5C,9H 9H 9H 3C,9H 5C,9H 2C,7H 9H 3C,9H      7H 0 9H 6H 4G 0 WILD OATS 7G 0 2C,6G 0 0 2G 8G 5G 5C,9G 3C,8G 4C,8H      3C,7G 3C,8G 3G 0 0 0 0 0 0 WHEAT 9H 5G 8H 0 5G 5G 9H 7G 9H 3C,9G 3C,9H      6G 3C,7G 3G 0 0 0 0 2G 0 CORN 3G 0 0 3G 0 0 9G 7G 3C,9H 3C,8G 3C,7G      2C,3G 3C,7G 2C,2G 3C,3G 0 2G 3G 2G 0 SOYBEAN 9H 6H 3C,7H 3C,3H 9H 3C,4H      9H 3C,6H 3C,8H 3C,7H 9H 3C,6G 4C,8H 3C,6H 2C,4H 0 3C,7G 3C,4G 0 0 RICE      9H 7G 10H 0 8H 3C,6G 10E 9H 10E 4C,9H 10E 10H 10E 9H 2C,5G 0 3C,7H 3G      2C,5G 0 SORGHUM 6C,9H 9H 9H 2C 4C,9H 3C,8H 10H 9H 10E 4C,9H 10H 9H 5C,9H      5C,9H 3C,6G 0 8H 3C,5G 3C,5G 0 CHEATGRASS 8G 0 8G 0 8G 5G 10E 4C,9G 10E      3C,8G 5C,9G 8H 9G 3C,7G 0 0 4G 0 0 0 SUGAR BEETS 5C,9G 8G 5C,9G 7G 3C,8G      7H 9C 10C 10C 4C,9G 9C 9G 9C 9C 5G 2G 3C,9H 7H 1H 0 VELVETLEAF 4C,8G 3G      6H 2G 2C,2H 2H 5C,9G 8H 5C,9G 3C,5H 5C,9G 3C,7G 4C,8H 5H 2G 0 2C,2H 0 2G      0 GIANT FOXTAIL 3G 0 3G 0 0 0 9H 3C,7G 9H 3C,7G 3C,8G 3C,5G 3C,8G 3C,6G      1H 0 7G 0 2G 0 BARLEY 8G 4G 8G 3G 9G 3C,7H -- -- -- 2C,8G 8G 7G -- 2C,5G      0 0 0 3G 9G 0        CMPD 114 CMPD 115 CMPD 116 CMPD 117 CMPD 118 CMPD 119 CMPD 120 CMPD      121 CMPD 122 CMPD 123 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 2C,3H 2G 4C,9G 9H 5C,9G 10C 5C,9G 4C,8G      9H 8H 9C 9C 1C 0 10C 4C,9G 0 -- 4C,9H 4C,9H MORNING GLORY 1H 0 10C 5C,9G      10C 10C 5C,9G 4C,9H 9C 3C,8H 10C 10C 3H 0 10C 10C 0 -- 10C 9C COCKLEBUR      2H 2H 8G 2G 10C 2C,3H 4C,9H 3C,5H 4C,9G 3C,7H 10C 10C 1H 0 10C 9C 2H --      9C 4C,9H NUTSEDGE 4C,9G 0 10C 4C,8G 9C 3C,8G 9G 8G 9C 4C,8G 5C,9G 4C,9G      0 0 9G 8G 0 -- 3C,8G 2C,5G CRABGRASS 3C,6G 3G 6G 2G 3C,6G 2C 0 0 0 0      3C,5G 2G 0 0 3C,5G 2G 0 -- 2C,5G 2G BARNYARD GRASS 9C 3C,8H 9C 5C,9G 9C      9C 2H 0 4H 0 9C 9C 4H 0 9C 9C 1H -- 9C 4C,9H WILD OATS 9C 3C,6H 5C,9G 3G      3C,7G 3G 0 0 0 0 4C,8G 3C,5G 3C,7G 0 4C,9G 3C,5G 2C,5G -- 4C,9G 5G WHEAT      9C 3C,7H 9G 2C,9G 5C,9G 9G 2G 0 0 0 9C 4C,9G 8G 0 5C,9G 8G 6G -- 9G 8G      CORN 4H 0 2G 0 6H 0 0 0 0 0 2C,7H 3H 0 0 0 0 0 -- 0 0 SOYBEAN 3C,8G 0      5C,9G 4C,9G 9C 5C,9G 4C,9G 3C,7H 3C,7H 3C,7H 5C,9G 5C,9G 3C,4G 0 5C,9G      4C,9G 2G -- 4C,9G 3C,8G RICE 5C,9G 9G 9C 9C 9C 3C,8G 2G 0 2G 0 9C 9C 8G      0 9C 9C 3G -- 9C 5C,9G SORGHUM 9C 4C,9G 9C 9C 9C 9C 3C,3H 0 6H 0 9C 9C      4C,9H 0 9C 4C,9G 2C,5G -- 9C 4C,9G CHEATGRASS 9C 3C,7G 8G 6G 3C,8G 3C,6G      0 0 0 0 5C,9G 4C,8G 3C,8G 0 4C,9G 4C,9G 3C,8G -- 9C 9G SUGAR BEETS 3C,7H      3C,6G 9C 9C 10C 9C 9C 3C,7G 9C 3C,7H 10C 9C 1H 0 10C 10C 0 -- 10C 4C,8H      VELVETLEAF 2H 0 9C 9C 10C 9C 3C,8H 3C,4H 4C,8H 3C,6H 10C 9C 1C 0 10C 9C      1C -- 9C 3C,7H GIANT FOXTAIL 9C 3C,8H 9C 4C,9G 4C,9H 3C,7G 0 0 1C 2G 9C      9C 2C,5G 0 9C 4C,9G 0 -- 5C,9G 3C,7H BARLEY 10C 2C,8G 3C,8G 3C,6G 3C,8G      3G 0 0 0 0 5C,9G 4C,9G 7G 0 4C,9G 3C,8G 8G -- 3C,8G 3C,6G PREEMERGENCE      COTTON 2H 0 3C,5G 6G 3C,5G 0 2G 0 2G 0 4C,8G 6G 0 0 3C,7H 0 0 -- 5G 0      MORNING GLORY 0 0 7H 0 2C,6G 0 7H 0 8H 0 9G 3C,7H 0 0 3C,7H 3C,3H 0 --      3C,8H 2C,6H COCKLEBUR 0 0 3G 0 -- 3G 3C,5G 1C 3C,3H 0 9H 2C,2H 0 0 3C,8H      3C,3G 0 -- 3C,6H -- NUTSEDGE 0 0 9G 0 8G 0 4G 0 9G 0 10E 3C,9G 0 0 4C,8G      0 0 -- 9G 10E CRABGRASS 7G 3G 4G 0 9G 0 0 0 0 0 3C,4G 3C,5G 0 0 3C,6G 3G      0 -- 7G 0 BARNYARD GRASS 6G 0 8H 2G 3C,9H 2G 0 0 3G 0 4C,9H 3C,7H 0 0      4C,9H 4G 0 -- 3C,9H 3C,8H WILD OATS 0 0 2C 0 1C 0 0 0 0 0 3C,6G 0 0 0 2G      0 0 -- 3G 0 WHEAT 7G 0 2G 0 3C,7H 0 0 0 0 0 3C,9H 3G 0 0 8G 6G 0 -- 8G 0      CORN 0 0 0 0 3G 0 0 0 7G 0 3C,6H 0 0 0 2H 0 0 -- 1H 0 SOYBEAN 0 0 3C,6H      2C 8H 3C,6H 3C,5G 2C 2C,6H 0 4C,8H 3C,6H 0 0 3C,7H 0 0 -- 3C,5H 2C,3H      RICE 2C,5G 0 9H 3C,5G 10H 5G 0 0 4G 0 10E 3C,8H 0 0 3C,8H 4G 0 -- 9H      3C,8G SORGHUM 3C,7G 0 9H 3C,7G 10E 8G 0 0 3G 0 5C,9H 3C,8H 0 0 4C,9H      2C,6G 0 -- 5C,9H 3C,9H CHEATGRASS 0 0 7G 0 9H 2G 0 0 0 0 5C,9G 3C,9G 0 0      9H 7G 0 -- 5C,9G 8G SUGAR BEETS 4H 0 4C,9G 7H 4C,9G 6H 3C,7G 2H 7G 0 9C      9C 3G 0 9C 4C,8H 2G -- 9C 5G VELVETLEAF 0 0 3C,5H 0 3C,8H 1C 2C 0 3C,4G      0 4C,8H 3C,6H 0 0 3C,7H 1C 0 -- 5G 0 GIANT FOXTAIL 3G 0 7G 0 3C,8G 0 0 0      0 0 4C,9H 3C,8G 0 0 3C,8H 0 0 -- 9H 2G BARLEY 9G 2G 2C,9G 3G 9G 0 0 0 4G      0 3C,9G 3C,8G 0 0 8G 0 0 -- 7G 3C,7G        CMPD 124 CMPD 125 CMPD 126 CMPD 127 CMPD 128 CMPD 129 CMPD 130 CMPD      131 CMPD 132 CMPD 133 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01  0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01     POSTEMERGENCE COTTON 4C,9H 3C,8H 5C,9G 9C 9H -- 10C 3C,9G 2C,9H      2C,5H 3C,9H 2C,8H 2C,8H 3C,6H 10C 5C,9G 9C 10C 9C 7G MORNING GLORY 4C,9G      4C,9H 10C 10C 4C,9G -- 10C 9C 6C,9G 4C,8H 3C,8H 2C,8G 6C,9G 4C,8H 10C      4C,9G 10C 9C 9C 7G COCKLEBUR 5C,9G 4C,9H 10C 10C 4C,9G -- 10C 5C,9H      3C,9H 3C,4H 9C 4C,9H 10C 2C,3H 10C 10C 10C 10C 10C 5C,9G NUTSEDGE 9G      3C,9G 10C 5C,9G 8G -- 2C,8G 8G 2C,6G 0 6G 2C,7G 3C,8G 2C,4G 9C 3C,8G      4C,9G 2C,9G 9C 3C,9G CRABGRASS 3C,4G 2G 3C,8G 5G 0 -- 0 0 0 0 0 0 0 0      4C,8G 2G 4C,8G 3G 5C,9G 6G BARNYARD GRASS 5C,9H 4C,8H 5C,9H 3C,6H 0 --      3C,9H 2C,7H 2C,5H 0 2G 3G 2C,6H 2C,6G 9C 9C 10C 9C 10C 10C WILD OATS      4C,9G 7G 8G 4G 0 -- 2C,6G 2C 2C 0 2G 0 2C,5G 3G 3C,9G 5G 4C,9G 3C,6G      4C,9G 4C,9G WHEAT 3C,9G 9G 8G 4G 0 -- 9G 9G 2C 0 2G 0 2C,9G 2G 3C,9G 9G      3C,9G 9G 4C,9G 9C CORN 0 0 3C,9G 9G 2H -- 3C,9G 3C,7H 2C,8H 2C,3G 2C 0      3C,8H 2C,2H 10C 3C,9G 5C,9G 4G 3C,9H 2H SOYBEAN 5C,9G 4C,9G 4C,9G 4C,9G      3C,5G -- 3C,8H 3C,8G 3C,8H 2C,3H 2H 0 4C,8H 3C,4H 9C 9C 5C,9G 9C 9C      4C,9G RICE 9C 5C,9G 5C,9G 3C,9G 0 -- 2C,9G 6G 4G 0 2C,5G 0 3C,9G 2C,4G      9C 9C 9C 9C 9C 5C,9G SORGHUM 5C,9G 3C,9G 5C,9G 3C,9G 3C,6G -- 5C,9G      2C,9G 9H 2C,7H 9G 3C,8H 2C,9G 2C,7H 10C 9C 9C 9C 10C 5C,9G CHEATGRASS      6C,9G 3C,9G 9C 9C 5G -- 10C 3C,9G 5G 3G 2C,8G 5G 8G 8G 9C 9C 10C 9C 10C      9C SUGAR BEETS 9C 4C,9H 10C 10C 3C,8G -- 10C 6C,9G 3C,9H 2C,3G 3C,6G      2C,7G 3C,9G 3C,5H 9C 10C 10C 10C 10C 9C VELVETLEAF 9C 4C,8H 10C 10C      3C,6G -- 9C 9C 3C,7H 2C,4G 2C,8G 2C,7G 5C,9H 3C,7G 10C 10C 10C 5C,9G 10C      10C GIANT FOXTAIL 6C,9G 4C,8G 3C,7G 5G 0 -- 2C,9G 6G 3G 2G 2G 3G 2C,7G      3G 9C 4C,9G 9C 3C,8G 9C 4C,8G BARLEY 5C,9G 2C,9G 8G 5G 0 -- 9G 6G 4G 0 0      0 7G 0 4C,9G 5G 9C 7G 4C,9G 8G PREEMERGENCE COTTON 2G 0 9G 8G 0 -- 2C,8G      4G 0 0 2G 0 4G 0 9G 6G 8G 3H 9G 2G MORNING GLORY 7H 1H 9G 9G 1H -- 9G      3C,9H 2C,3H 0 2C,6H 0 0 0 9G 3G 2C,3G 2G 7G 0 COCKLEBUR 2H 1H 9H 9H 7G      -- 3C,8H 3C,7H 2H 0 3C,8H 0 0 0 8H 9H 9H 2C,2H 8H 2C,8H NUTSEDGE 3G 0      10E 10E 0 -- 10E 2C,9G 8G 0 9G 0 0 0 10E 10E 9G 3C,9G 10E 10E CRABGRASS      0 0 5G 0 0 -- 2C 0 2G 0 2G 0 0 0 5G 0 3C,9G 5G 8G 0 BARNYARD GRASS 5G 0      9H 3C,7G 0 -- 4C,8H 2C,3G 5G 0 6G 0 3G 0 9H 5G 3C,9H 3C,7G 9H 8G WILD      OATS 2G 0 6G 3G 0 -- 4C,7G 3G 0 0 2G 0 0 0 3C,6G 0 3C,5G 0 3C,7G 2C,3G      WHEAT 3G 0 7G 2G 0 -- 8G 3G 0 0 0 0 0 0 9H 0 3C,9H 0 3C,9H 5G CORN 0 0      9H 2C,9G 0 -- 4C,8H 2C,3G 0 0 3G 0 0 0 3C,9H 2G 3C,8H 3G 3C,9H 3C,5G      SOYBEAN 3C,6G 0 2C,7H 3C,2H 2G -- 3C,5G 2C 2C 0 2C 0 0 0 9H 3C,4G 3C,7G      3C,5H 9H 3C,6H RICE 3C,6G 0 9H 9H 4G -- 9H 3C 0 0 2C,8H 0 5G 0 10E 8G      10E 9H 10E 9H SORGHUM 3C,7G 2C 9H 5C,9H 2C -- 5C,9H 3C,8H 2C,3G 0 3C,9H      0 2C,5G 2G 5C,9H 3C,8G 5C,9H 3C,9H 10H 3C,9H CHEATGRASS 8G 0 9H 8G 0 --      4C,9H 3C,8H 0 0 4G 0 3C,7G 2G 9H 8G 8G 8H 9H 8H SUGAR BEETS 9G 4G 10C 9C      8G -- 3C,9G 3C,9G 0 0 3C,8G 0 9C 0 5C,9G 9C 5C,9G 7H 4C,9G 4C,9G      VELVETLEAF 2C,3G 2H 5C,9G 4C,8H 0 -- 4C,8H 3C,6G 0 0 3G 0 0 0 8H 7G      2C,6H 2C,2H 7H 3G GIANT FOXTAIL 0 0 8G 2C,5G 0 -- 3C,8H 6G 0 0 3G 0 2G 0      9H 6G 3C,9H 4G 9H 6G BARLEY 7G -- 8G 8G 0 -- 8G 2G 0 0 2G 0 7G 0 9G      2C,4G 3C,8G 2C,8G 9G 9G        CMPD 134 CMPD 135 CMPD 136 CMPD 137  CMPD 138 CMPD 139 CMPD 140 CMPD      141 CMPD 142 CMPD 143 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 9C 3C,8H 2C,3G 1C 8H 2C,2G 10C 4C,9G      3C,7G 0 4C,9G 3C,8G 9C 3C,9G 5C,9H 4C,8H 10C 5G 5C,9G 4C,8H MORNING      GLORY 10C 9C 4C,8H 3C,4H 4C,8H 3C,8H 10C 4C,8G 10C 3C,7H 4C,9G 4C,8G 9C      5C,9G 9C 4C,8H 10C 5C,9G 10C 5C,9G COCKLEBUR 10C 10C 3C,5H 3G 4C,8H      3C,5G 10C 10C 2H 0 4C,9G 4C,9G 10C 8H 10C 4C,9H 9C 3C,7H 10C 9C NUTSEDGE      9C 9G 0 2C,4G 3C,7G 3C,5G 3C,9G 3C,8G 0 0 3C,5G 2C,4G 4C,9G 9G 2C,5G 3G      4C,9G 4C,9G 4C,8G 2C,5G CRABGRASS 3G 0 2G 0 3G 0 4G 0 0 0 5G 0 5G 0 0 0      3G 0 3G 3G BARNYARD GRASS 9C 5C,9H 3C,8H 3C,7H 9C 4C,9H 9C 3C,9H 9H      4C,9H 9C 3C,8H 9C 5C,9H 4C,9H 3C,7H 4C,9H 3C,7H 9C 3C,8H WILD OATS 4C,9G      2G 0 0 2C,3G 2G 0 0 0 0 2C 0 1C 0 1C 0 0 0 2C,5G 0 WHEAT 9G 4G 2G 0 0 0      2G 0 7G 0 9G 3G 5G 0 2G 0 4G 0 7G 3G CORN 0 3G 3C,9G 3C,7H 9C 3C,8H 0 0      0 0 0 0 3G 0 0 0 1C 0 3C,7G 2G SOYBEAN 4C,9G 3C,8H 3C,8G 4H 4C,9G 4C,8H      3C,9G 1H 3C,5H 2H 4C,9G 4C,8G 5C,9G 3C,5H 4C,9G 1H 4C,9G 5C,9G 5C,9G      4C,9G RICE 9C 7G 3G 0 2C,3G 0 5C,9G 3C,6G 3C,7G 3G 5C,9G 2C,5G 6C,9G 6G      5G 0 5C,9G 8G 9C 6C,9G SORGHUM 9C 3C,8H 3C,9H 3C,7H 9C 3C,9G 9C 9G 5C,9G      4C,9H 4C,9G 2C,5G 6C,9G 4C,9H 5C,9H 3C,6G 5C,9H 3C,9H 9C 6C,9G CHEATGRASS       9C 9G 8G 6G 5C,9G 7G 8G 5G 3C,8G 6G 5G 0 9C 3C,9G 9G 8G 3C,9G 8G 3C,9G      2G SUGAR BEETS 9C 9C 8H 5H 9C 3C,7G 9C 3C,8G 3C,4H 2H 5C,9H 4C,9H 10C 9C      9C 9C 9C 9G 10C 9C VELVETLEAF 9C 5C,9G 2G 2G 3C,7G 1C 10C 3C,8G 3C,7H 2G      10C 3C,8H 10C 9C 9C 4C,7G 10C 9C 10C 4C,8H GIANT FOXTAIL 5C,9G 3C,7G      2C,8G 7G 9C 3C,7G 3C,9G 3C,7G 3C,7G 5G 5C,9G 3C,5G 3C,8G 3C,5G 3C,7G 3G      3C,7G 3C,5G 9C 5C,9G BARLEY 7G 0 0 0 2G 0 0 0 0 0 2G 0 0 0 0 0 2C,3G 0      8G 0 PREEMERGENCE COTTON 7H 1H 0 0 0 0 6G 0 0 0 0 0 2C 0 1C 0 2C 0 3C,5G      0 MORNING GLORY 9G 7G 1H 0 3C,7H 0 9G 4G 0 0 0 0 8H 0 3C,3H 0 2C,2H 0 8G      0 COCKLEBUR 8H -- 4H -- 3C,5G 2C 3C,5H 2C,5G -- 0 0 0 8G 0 2C 0 2C 0      3C,3H 0 NUTSEDGE 10E 9G 10E 0 7G 0 9G 0 0 0 0 0 9G 0 0 0 10E 0 0 0      CRABGRASS 3G 0 0 -- 3C,7G 0 3G 0 0 0 0 0 4G 0 0 0 2G 0 0 0 BARNYARD      GRASS 9H 7H 5G 0 4C,8H 0 9H 0 0 0 0 0 3C,7G 0 1C 0 3C,7H 0 7G 0 WILD      OATS 6G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 1C 0 0 0 WHEAT 7G 0 0 0 0 0 3G 0 0      0 0 0 0 0 0 0 6G 0 6G 0 CORN 3C,7G 5G 6H 0 3C,8H 2C 2G 0 0 0 0 0 0 0 0 0      2C,3G 0 3C,7G 0 SOYBEAN 3C,7H 3C,4H 0 0 3C,3G 0 3C,3H 2G 0 0 0 0 3C,3H 0      2G 0 3C,5H 0 3C,7G 3C,4H RICE 10E 9H 2G 0 4G 0 9G 9G 0 0 0 0 9H 0 0 0      3C,9H 0 10E 2C,5G SORGHUM 10H 5C,9H 3C,7G 0 5C,9H 3C,6G 10H 9H 0 0 0 0      4C,8G 3C 4C,7G 0 3C,9H 0 9H 3C,9H CHEATGRASS 9H 8G 6G 0 8H 0 9G 0 0 0 0      0 8G 0 2G 0 9H 0 4G 0 SUGAR BEETS 9G 8G 7G 2H 4C,8H 1H 9H 8H 4G 0 0 0 9G      4G 4C,7H 0 9G 0 4C,9G 7H VELVETLEAF 7H 5G 0 2G 0 0 5H 0 0 0 0 0 7H 0 2C      0 2H 0 3C,6H 0 GIANT FOXTAIL 9H 6G 2G 2G 3C,8G 0 9H 0 0 0 0 0 3C,4G 0 3G      0 2C,5G 0 8G 0 BARLEY 9G 7G 0 0 4G 0 2C,3G 0 0 0 0 0 0 0 0 0 2C,3G 0      2C,4G 2G        CMPD 144  CMPD 145 CMPD 146 CMPD 147 CMPD 148 CMPD 149 CMPD 150 CMPD      151 CMPD 152 CMPD 153 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 3C,7G 2C,2G 4C,9H 4C,9H 10C 4C,8G 3C,8H 0      8H 0 9G 4C,8H 0 0 3C,7G 0 10C 9C 10C 10C MORNING GLORY 3C,8G 3C,6G 9C      5C,9H 10C 4C,8G 3C,5G 0 3C,4H 0 4C,9G 3C,8H 2C,3G 0 4C,8H 0 10C 10C 10C      9C COCKLEBUR 4C,8H 2H 10C 3C,9G 10C 4C,9H 5C,9G 2H 3C,3H 0 4C,9G 3C,3H      2C 0 4C,8H 0 10C 10C 10C 10C NUTSEDGE 0 -- -- -- 4C,9G 4C,9G -- -- -- 0      -- 2G 0 0 0 0 4C,9G 4C,9G 4C,9G 9G CRABGRASS 0 0 5G 0 5G 4G 2G 0 3G 0 5G      3G 0 0 3C,5G 3G 3C,7G 3C,6G 3C,7G 3G BARNYARD GRASS 3C,6H 0 5C,9H 3C,7H      9C 4C,8H 4C,8H 2H 5C,9H 3C,7H 9C 3C,8H 3C,9H 5G 9C 3C,9H 9C 9C 9C 4C,8H      WILD OATS 0 0 2G 0 0 0 1C 0 3C,7G 0 3C,8G 2G 2C,9G 3C,4G 5C,9G 3C,8G      4C,9G 2C,6G 3C,7G 2C,3G WHEAT 0 0 -- -- 7G -- 3G 0 -- 0 -- -- 9G 9G 9G      9G 2C,9G 9G 4C,9G 8G CORN 0 0 3C,9H 2C,5G 3C,7H 1H 2H 0 5C,9G 3C,3G 9C      3C,8H 3G 0 0 0 0 0 0 0 SOYBEAN 3C,6H 2C,2H 5C,9G 3C,9H 5C,9G 4C,8G 3C,8G      0 3C,7G 2G 5C,9G 3C,7G 3C,7H 1H 3C,8G 3C,6G 5C,9G 9C 9C 9C RICE 2C 0 9C      3C,8G 5C,9G 3C,5G 4C,9G 0 8G 2G 9C 5C,9G 3C,9G 5G 4C,9G 6G 5C,9G 5C,9G      5C,9G 6C,9H SORGHUM 3C,7G 2G 9C 5C,9G 9C 4C,9H 4C,9G 3G 4C,9H 3C,6G 9C      4C,9G 3C,8H 3G 5C,9G 3C,9G 9C 9C 9C 6C,9H CHEATGRASS 0 0 3C,7G 2G 9C 9G      3C,5G 0 4C,9G 6G 8G 6G 5G 0 8G 2C,5G 9G 8G 4C,9G 7G SUGAR BEETS 3C,8G 0      9C 9C 10C 5C,9H 3C,7G 3G 3C,7H 2H 9C 4C,8H 3C,7H 5H 4C,8G 4C,5G 10C 9C      9C 6C,9G VELVETLEAF 3C,7G 0 6C,9G 3C,6G 10C 5C,9H 3C,6G 0 0 -- 4C,8G 2C      3G 0 1C 0 10C 5C,9G 10C 9C GIANT FOXTAIL 3G 0 5C,9G 5C,9G 5C,9G 3C,8G      3C,7G 0 4C,8G 3G 5C,9G 3C,8G 2G 0 5C,9G 2C,5G 4C,8G 3C,7G 3C,8G 5G      BARLEY 0 0 7G 0 5G 0 3C,7G 0 0 0 6G 0 8G 7G 8G 6G 8G 8G 8G 5G PREEMERGENC      E COTTON 0 0 1C 0 2G 0 0 0 0 0 2C,2G 0 0 0 1C 0 9G 8G 8G 3G MORNING      GLORY 0 0 3C,3H 0 0 0 0 0 0 0 3C,5H 0 0 0 0 0 9G 6G 8H 7H COCKLEBUR 0 0      1C 0 0 0 0 -- 0 -- 2C 0 0 0 6G 2H 9H -- -- -- NUTSEDGE 0 0 0 0 8G 0 0 0      0 0 2G 0 0 0 0 0 10E 9G 10E 9G CRABGRASS 0 0 0 0 1C 0 0 0 0 0 0 0 0 0 0      0 8G 6G 7G 2G BARNYARD GRASS 0 0 5G 0 3C,8H 0 2C 0 0 0 3C,7G 0 0 0 2H 0      9H 8H 3C,8H 0 WILD OATS 0 0 0 0 1C 0 0 0 0 0 0 0 0 0 2C,5G 0 7G 3G 4C,8G      2C,3G WHEAT 0 0 0 0 5G 0 0 0 0 0 2G 0 8G 0 3C,9H 0 9H 9G 4C,9H 8G CORN 0      0 3C,5G 0 3C,4G 1C 0 0 0 0 3C,6G 1C 1C,1H 0 0 0 3G 0 0 0 SOYBEAN 0 0      3C,5G 0 2C,2H 0 0 0 0 0 3C,2H 2C 0 0 0 0 9H 8H 9H 3C,6H RICE 0 0 4C,9H 0      9H 0 2C 0 0 0 3C,9H 2C,3G 7H 0 10H 0 10E 9H 9H 9H SORGHUM 0 0 4C,9H      3C,7G 3C,9H 3C,5G 3C,3G 0 3C,6G 0 3C,9H 3C,8H 3C,4G 0 9H 0 10H 9H 10H 9H      CHEATGRASS 0 0 0 0 2C,8G 0 0 0 0 0 0 0 0 0 0 0 8G 6G 9H 3C,7G SUGAR      BEETS 0 0 4C 6H 9G 2H 4H 0 3G 4G 5H 3H 5G 0 5G 1H 9C 3C,7G 9G 3C,8H      VELVETLEAF 0 0 2C 0 0 0 0 0 0 0 2C 0 0 0 0 0 5C,9G 4C,6H 4C,8H 3C,4H      GIANT FOXTAIL 0 0 3G 0 4C,9H 0 0 0 0 0 4C,8G 0 0 0 5G 0 6G 2G 6G 0      BARLEY 0 0 2C 0 2C 0 2C 0 0 0 2G 0 7H 0 4C,9G 0 9G 8G 9G 6G        CMPD 154 CMPD 155 CMPD 156 CMPD 157 CMPD 158 CMPD 159 CMPD 160 CMPD      161 CMPD 162 CMPD 163 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 10C 3C,8H 10C 9C 2G 2H 2G 0 10C 10C 10C      4C,9G 3C,7H 1C 9C 3C,8G 6G 0 9C 5C,9G MORNING GLORY 4C,9H 2C,6G 10C 10C      4C,9G 3C,7H 2C,5G 0 9C 10C 9C 9C 4C,8H 1H 10C 9C 1C 0 10C 10C COCKLEBUR      9C 4C,9H 10C 10C 7H 2H 3C,8H 2C,3H 10C 10C 10C 10C 1H 1H 10C 10C 7H 0 9C      2G NUTSEDGE 9G 2C,9G 9G 9G 0 0 0 0 9C 2C,9G 3C,8G 2C,9G 4G 0 2C,9G 9G 0      0 5C,9G 5C,9G CRABGRASS 5G 3G 3C,6G 5G 3C,6G 2C,4G 5G 0 1H 0 4G 0 4G 0      5G 0 0 0 4C,9G 3C,6G BARNYARD GRASS 4C,8H 3C,7H 3C,8H 6C,9H 3C,8H 3C,4G      2C,3H 9C 4C,9H 3C,7H 0 9C 9C WILD OATS 3C,8G 2C,5G 3C,5G 0 9C 4C,9G      2C,5G 0 3C,6G 2C,2H 3C,8G 2C,5G 2C,9G 4C,9G 4G 0 0 0 6C,9G 5C,9G WHEAT      8G 4G 7G 3G 3C,9G 9G 7G 4G 9G 5G 9G 2C,9G 7G 3G 5G 0 0 0 9C 9G CORN 2G      2G 0 0 0 0 0 0 5G 2G 3C,8H 3G 2C,5H 0 2G 0 0 0 1H 0 SOYBEAN 4C,9G 4C,9G      4C,9G 3C,9G 8G 3C,7G 3C,8G 2C,3H 9C 5C,9G 9C 4C,9G 3C,6H 2H 9C 9C 3H 0      4C,9G 6C,9G RICE 5C,9G 5C,9G 4C,9G 2C,8G 6C,9G 4C,9G 6G 4G 9G 3C,8G      2C,8G 4G 4C,9G 4G 2C,9G 7G 2G 0 5C,9G 9C SORGHUM 4C,9G 5C,9H 5C,9G 5C,9H      5C,9G 3C,8H 3C,6G 2C,4G 2C,9G 5C,9G 4C,9G 4C,9G 3C,9H 2C,5G 9C 5C,9G 7G      0 10C 9C CHEATGRASS 8G 3C,5G 2C,5G 2G 3C,8G 2C,7G 3C,4G 2G 5C,9G 3C,6G      9C 5C,9G 4C,9G 3C,8G 3C,9G 2C,8G 5G 0 5C,9G 2C,9G SUGAR BEETS 9C 4C,9G      5C,9G 3C,7H 3C,7H 3C,7H 3C,3G 0 10C 9C 9C 5C,9G 3C,7H 4H 4C,9G 3C,7H      2C,5G 0 9C 9C VELVETLEAF 4C,9H 3C,7H 4C,8H 3C,6H 2C,5G 3C,3G 2G 3G 10C      10C 10C 10C 2C,2G 0 10C 6C,9G 2C,5G 0 10C 10C GIANT FOXTAIL 3C,7G 3G      3C,7G 2C,5G 4C,9G 3C,8G 2C,7G 3G 2C,8G 4G 4C,9G 7G 4C,9G 3C,6G 3C,9G      3C,8G 3C,6G 0 9C 9C BARLEY 7G 5G 8G 5G 7G 4C,9G 4C,9G 5G 9G 3C,4G 2C,9G      3G 4C,9G 2C,5G 3C,9G 2C,5G 2C,5G 0 3C,9G 9G PREEMERGENCE COTTON 2G 4G      3C,7G 1C 0 0 0 0 5C,9G 4C,8G 8G 2C,4G 0 0 8G 2C,3G 2G 0 3C,8H 2G MORNING      GLORY 7H 0 4C,8H 5H 2C 1H 0 0 7H 6H 9H 5H 2C,3G 0 9G 3C,8H 5G 0 8H 5H      COCKLEBUR 8H 8H 3C,8H 3C,5H 3H 3H 0 0 -- -- 9H 3C,3H 2H 0 3C,8H 3C,3H      2C,4G 0 0 0 NUTSEDGE 3C,8G 0 10E 9G 0 0 0 0 9G 9G 10E 5G 0 0 7G 3C,8G 0      0 10E 8G CRABGRASS 3G 0 7G 3G 3G 0 3G 0 0 0 4G 0 0 0 5G 0 0 0 4C,8G      2C,8G BARNYARD GRASS 3C,7H 0 6H 3G 4G 0 2G 0 8G 6G 3C,8H 0 2C 0 4C,9H      4C,9H 3G 0 3C,8H 2C,4G WILD OATS 2C,3G 0 0 0 3C,6G 3G 0 0 2C,3G 2G 4C,8H      2C,4G 6G 0 0 2G 0 0 3C,9H 2C,3G WHEAT 2C,6G 0 8G 0 2C,8H 5G 0 0 2C,8G 6G      4C,9H 8H 4G 0 8G 2G 0 0 3C,9H 8G CORN 0 0 0 0 0 0 0 0 3C,3G 0 3C,7H 2G 0      0 3C,7G 2C,5G 0 0 0 0 SOYBEAN 3C,6H 2C,2H 3C,8H 3C,4H 1C,1H 0 0 0 3C,6H      5G 3C,7H 3C,3H 0 0 4C,8H 3C,6H 0 0 8H 7H RICE 9H 8G 10E 9H 9H 0 2G 0      5C,9H 8H 10E 7G 3C,6G 0 5C,9H 4C,9H 6G 0 10E 9H SORGHUM 9H 3C,5G 9H      4C,9H 3C,9G 2C,5G 2G 0 5C,9H 9H 4C,9H 3C,7H 3C,6G 0 9H 4C,9H 3G 0 5C,9H      9H CHEATGRASS 7G 0 5G 0 4G 0 0 0 9G 6G 9H 8G 6G 0 3C,9G 8G 0 0 9H 8G      SUGAR BEETS 4G 5G 7H 3H 5H 6G 0 0 9C 4C,9G 5C,9G 3C,8G 6H 0 9G 3C,7G 3G      0 5C,9G 8G VELVETLEAF 3C,5H 1C 3C,5H 3G 2H 1H 0 0 9G 8H 8H 3G 2H 0 3C,7G      2H 2G 0 8H 3C,5H GIANT FOXTAIL 5G 0 6G 2G 2C,5H 0 2H 0 7G 0 4C,8H 5G      2C,5G 0 4C,9G 3C,9H 2G 0 4C,9H 2C,5G BARLEY 8G 2G 8G 4G 9G 2G 2G 0 9H 6G      3C,9G 2G 2C,8G 0 3C,9G 4G 0 0 9G 2C,7G        CMPD 164 CMPD 165 CMPD 166 CMPD 167 CMPD 168 CMPD 169 CMPD 170 CMPD      171 CMPD 172 CMPD 173 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 10C 10C 10C 10C 10C 9C 4C,9H 3C,8G 3C,6G      0 10C 3C,7H 9C 4C,9G 5C,9H 4C,9H 0 -- 3C,9G 10C MORNING GLORY 10C 10C      10C 10C 10C 10C 4C,8H 4C,8H 4C,8H 3C,7H 9C 4C,8H 10C 9C 5C,9H 3C,6G 0 --      0 0 COCKLEBUR 10C 9H 9C 6H 10C 10C 5C,9H 1H 1H 0 1H 0 10C 10C 10C 4C,9H      2G -- 8G 2C,6G NUTSEDGE 5C,9G 4C,9G 9C 5C,9G 9C 2C,9G 5G 0 0 0 3G 0 10C      4C,9G 8G 3C,7G 3G -- 0 0 CRABGRASS 3C,7H 2C,5G 6C,9G 2C,8G 3C,7G 3G      3C,7G 2C,5G 4G 0 4C,9H 2C,8G 4C,8G 2C,6G 2G 0 0 -- 0 0 BARNYARD GRASS 9C      9C 10C 9C 9C 9C 9C 4C,8G 10C 0 9C 9C 9C 9C 4G 2H 0 -- 2C,5H 0 WILD OATS      9C 3C,8G 5C,9G 4C,9G 4C,9G 2C,6G 3C,6G 2C 3G 0 5C,9G 5C,9G 5C,9G 3C,8G      2C,5G 0 0 -- 0 0 WHEAT 9C 3C,9G 9C 4C,9G 2C,9G 6G 4C,9G 2G 3G 0 9G 9G 9G      6G 4G 0 0 -- 5G 0 CORN 3C,7H 1H 3H,7G 3G 0 0 2C,4H 2H 10C 5H 2C,8H 3H      3C,7H 0 0 0 0 -- 0 0 SOYBEAN 9C 9C 9C 9C 5C,9G 4C,9G 5C,9G 4C,9G 5C,9G      2C,7G 3C,8H 5H 9C 9C 3C,9G 4C,8G 0 -- 0 0 RICE 9C 9C 9C 9C 9C 9C 9C      3C,6G 4C,9G 3G 9C 9C 9C 4C,9G 4C,9G 2C,6G 0 -- 0 0 SORGHUM 10C 9C 10C 9C      9C 9C 9C 4C,9H 4C,9G 2C,3G 9C 4C,9G 9C 9C 4C,9H 3C,8G 0 -- 3G 0 CHEATGRAS      S 9C 4C,9G 9C 4C,9G 3C,9G 6G 2C,8G 2C,5G 4G 0 4C,9G 9G 9C 3C,9G 2C,8G 8G      0 -- 3G 0 SUGAR BEETS 9C 9C 10C 10C 9C 10C 10C 9C 9C 2C,5G 9C 3C,7H 10C      5C,9G 9C 5C,9H 3G -- 3H 2G VELVETLEAF 10C 10C 10C 10C 10C 10C 5C,8H      3C,5H 2C,4G 0 9C 4C,8H 10C 10C 5C,9H 4C,8H 0 -- 3G 2C,3G GIANT FOXTAIL      9C 9C 9C 6C,9G 9C 9C 9C 4C,8H 9C 0 9C 9C 9C 4C,9G 5G 2H 0 -- 2C,6G 0      BARLEY 4C,9G 3C,8G 4C,9G 9G 9G 7G 2G 0 0 0 9C 4C,9G 3C,8G 7G 2C,4G 0 0      -- 0 0 PREEMERGENCE COTTON 4C,9G 2C,5G 5C,9G 9G 2C,8H 5G 3G 0 0 0 3G 0      4C,8H 3C,8G 2C,6G 0 0 -- 2G 0 MORNING GLORY 9C 3C,9H 9C 9C 9G 3C,8H 2H      1H 0 0 8H 0 9H 8H 8H 3C,3H 0 -- 0 0 COCKLEBUR 5G 0 6G 3G 7H 3H 2G 1H 0 0      0 0 9H 8H -- 2C,2H 0 -- 3G 0 NUTSEDGE 9G 10E 10E 10E 10E 10E 0 0 0 0 0 0      10E 8G 0 0 0 -- 0 0 CRABGRASS 4C,7G 3C,6G 4C,9G 3C,6G 2C,6G 3C,6G 0 0 0      0 4C,8G 0 3C,7G 0 0 0 0 -- 0 0 BARNYARD GRASS 9H 4C,8H 9H 9H 9H 3C,9H      2C,6G 3G 0 0 4C,9H 3G 9H 6H 3G 0 0 -- 0 0 WILD OATS 4C,9H 2C 4C,8G 2C,6G      2C,8G 1C 0 0 0 0 2C,8H 2G 3C,9G 3G 1C 0 0 -- 0 0 WHEAT 4C,9H 2C,8H 4C,9H      2C,8H 9H 7H 7G 0 0 0 9H 4G 3C,9G 5G 0 0 0 -- 0 0 CORN 3C,9H 0 4C,9H 4G      2G 0 6H 0 2C,3G 0 4C,9H 0 3C,8H 2G 1C,2G 0 0 -- 0 0 SOYBEAN 9H 7H 9H 9H      9H 3C,8H 2C,6H 2C,2H 2G 0 3G 0 9H 8H 2C,6G 0 0 -- 0 0 RICE 10E 9H 10E      10E 10E 10E 8H 2C,5G 0 0 10E 9H 5C,9H 2C,8G 4G 2G 0 -- 2G 0 SORGHUM 10E      5C,9H 10H 4C,9H 10E 10E 4C,9H 2C,4G 2C,5G 0 10H 9H 5C,9H 9H 3C,9G 3G 0      -- 4G 0 CHEATGRASS 9H 9H 9H 9H 9G 7G 3G 0 0 0 9H 0 5C,9G 8G 5G 0 0 -- 0      0 SUGAR BEETS 5C,9G 8H 5C,9G 9G 4C,9G 9G 6G 0 0 0 0 0 5C,9G 4C,9G 5C,9G      5G 0 -- 7G 5G VELVETLEAF 5C,9H 2C,5H 5C,9G 2C,8H 5C,9G 3G 0 0 0 0 2G 0      5C,9G 5G 3C,7H 2C,2G 0 -- 0 0 GIANT FOXTAIL 4C,9H 3C,8H 9H 4C,9H 9H      2C,6G 2C,5G 0 0 0 9H 3C,8G 5C,9H 4C,8H 3G 0 0 -- 2G 0 BARLEY 3C,9G 4G 9G      9G 9G 2C,8G 7G 0 0 0 2C,9H 2C 3C,9G 8G 5G 0 0 -- 5G 0        CMPD 174 CMPD 175 CMPD 176 CMPD 177 CMPD 178 CMPD 179 CMPD 180 CMPD      181 CMPD 182 CMPD 183 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 5C,9G 3G 9C 4C,9G 9C 10C 9C 10C 9C 4C,9H      10C 4C,9H 10C 4C,8H 10C 9C 10C 10C 10C 4C,8H MORNING GLORY 3C,8H 2C,4H      5C,9G 4C,8H 10C 9C 10C 5C,9G 10C 2C,7G 10C 5C,9G 3C,8H 6C,9G 10C 10C 10C      10C 10C 2C,8H COCKLEBUR 4C,9G 2G 10C 4C,8H 10C 10C 10C 10C 10C 9C 10C      10C 9C 5C,9H 10C 10C 10C 10C 10C 3C,7H NUTSEDGE 0 0 2C,8G 0 9G 9G 9G      3C,9G 8G 2C,4G 9C 3C,9G 5C,9G 2C,9G 9C 6C,8G 10C 9C 9C 9G CRABGRASS 0 0      3G 0 3C,8G 5G 3C,7G 2G 3G 0 5G 0 6G 4G 2C,7G 4G 2C,9G 5G 2C,4G 2G      BARNYARD GRASS 7H 3G 9H 5G 9C 4C,9H 5C,9H 3C,9H 9H 3C,7H 4C,9H 3C,7H 10C      3C,7H 9C 4C,9G 10C 10C 9C 5C,8G WILD OATS 0 0 3C,8G 5G 4C,9G 9G 5C,9G      3C,7G 4C,9G 4C,9G 3C,5G 2C,3G 3C,8G 2C,7G 2C,6G 7G 2C,6G 2G 2C,8G 0      WHEAT 0 0 3G 0 9G 9G 9G 9G 9G 9G 9G 5G 2C,9G 9G 9G 8G 3C,9G 7G 2C,9G 3G      CORN 2G 0 0 0 2H 0 1H 0 0 0 1H 0 4U,8G 2C,7G 6U,9G 3U,8G 10C 6U,9G 6U,9G      3C,7G SOYBEAN 4C,9G 7H 5C,9G 4C,9G 9C 9C 9C 5C,9G 5C,9G 4C,9G 3C,8H      2C,5H 5C,9G 5C,8H 6C,9G 6C,9G 6C,9G 9C 4C,8H 2C,6H RICE 7G 0 9G 4G 9C 9C      9C 5C,9G 4C,9G 4C,9G 4C,9G 4C,9G 5C,9G 6C,8G 3C,7G 3G 5C,8G 2C,8G 3C,8G      3G SORGHUM 2G 0 3C,9G 3C,7G 5C,9G 4C,9G 5C,9G 3C,9G 3C,9G 3C,8G 3C,9G      4C,9H 10C 3U,8G 6C,9G 3C,8G 6C,9G 5C,9G 6C,9G 2C,8G CHEATGRASS 0 0 3G 0      6G 4G 8G 0 0 0 3G 0 5C,9G 4C,9G 10C 9C 10C 9C 9C 3C,8G SUGAR BEETS 9C      4C,8H 9C 10C 10C 10C 10C 9C 10C 10C 10C 9C 9C 9C 10C 10C 10C 9C 6C,9G      5C,9G VELVETLEAF 3C,7H 0 4C,9H 3C,6H 10C 10C 10C 6C,9G 10C 4C,9H 10C      4C,9G 9C 6C,9H 10C 10C 10C 10C 10C 6C,9H GIANT FOXTAIL 2G 0 3C,6G 3G      4C,9G 3C,7G 4C,9G 3C,6G 2C,4G 3G 3C,7H 3C,6G 10C 3C,9G 9C 4C,9G 10C      6C,9G 3C,9G 2C,7G BARLEY 0 0 6G 0 3C,9G 9G 3C,9G 3C,9G 9G 7G 9G 5G 6C,9G      3C,8G 2C,8G 7G 8G 5G 8G 2C,4G PREEMERGENCE COTTON 3G 0 2G 0 2C,9G 8G      3C,6G 1C 2G 0 9G 2C,6G 2C,6G 0 3C,7G 3G 3C,9G 3C,8G 2C,8G 4G MORNING      GLORY 5H 0 6H 1H 9H 4G 7G 0 2H 0 3C,8G 3C,7H 7H 3G 9G 6G 9H 9C 9H 3C,8H      COCKLEBUR 2C,6H 0 2C,5G 0 9H 7H -- 3C,4G 2C,3H 0 9H 8H -- 3C 8H 2G 2C,9H      -- 8H 4C,8G NUTSEDGE 0 0 0 0 9G 5G 8G 3G 2C,5G 0 10E 10E 7G 0 9G 0 10E      9G 10E 3C,8G CRABGRASS 0 0 0 0 9G 0 2C 0 0 0 2G 0 0 2G 0 3G 2C,4G 6G 2C      0 BARNYARD GRASS 2H 0 0 0 9G 1H 3H 0 1C 0 8H 7H 0 0 3C,7G 0 9H 2C,7H 9H      7G WILD OATS 0 0 0 0 3C,7G 2C,5G 3C,5G 0 3C,4G 0 2C,5G 0 2C,4G 0 2C,6G 0      2C,7G 3G 2C,4G 0 WHEAT 0 0 0 0 9H 9H 9H 0 6G 0 8H 3G 2C,8H 4G 2C,8G 7G      2C,8H 7G 2C,8H 4G CORN 6G 0 0 0 5G 0 0 0 0 0 0 0 9H 0 2C,9H 3C,7H 9H      2C,9H 9H 9H SOYBEAN 2C,5G 0 3C,6H 1C,1H 9H 3C,6H 3C,7H 2C,4G 2C,5G 0      3C,7H 5G 2C,8H 5G 3C,8H 2C,4G 2C,8H 3C,8H 2C,7H 3H RICE 8H 0 8G 2G 10E      10H 9H 1C 2C,3G 0 10E 9H 3C,9H 2C 2C,7G 0 3C,8H 2C,6G 2C,9H 3C,8H      SORGHUM 2G 0 2C,8H 2G 4C,9H 9H 9H 3C,5G 3C,7G 0 9H 9H 3C,9H 3C,6G 3C,7H      3C,7G 10H 2C,9H 10H 10H CHEATGRASS 0 0 0 0 5G 0 4G 0 0 0 0 0 2C,8H 2G      3C,9H 3G 9H 2C,9H 2C,9H 9H SUGAR BEETS 4G 0 7H 2G 9G 9G 9G 7G 4C,9G      3C,6H 9G 9G 4C,8G 3G 4C,9G 2C,8G 3C,9G 4C,9G 4C,8G 4C,8H VELVETLEAF 2G 0      0 0 4C,9G 3H 6G 3C,3H 3C,3H 0 3C,7H 3C,3H 4C,7H 2H 4C,8H 7G 4C,9H 2C,8H      4C,8H 2C,4G GIANT FOXTAIL 0 0 0 0 2C,5G 0 4G 1C 0 0 5G 3G 0 2G 3G 3G      2C,9H 3C,9H 2C,7G 2C BARLEY 0 0 8G 0 9G 2C,6H 3C,9G 0 2C,8G 0 9G 4G      2C,9H 4G 2C,8G 2C,5G 8G 8G 8G 5G        CMPD 184 CMPD 185 CMPD 186 CMPD 187 CMPD 188 CMPD 189 CMPD 190 CMPD      191 CMPD 192 CMPD 193 RATE RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01      POSTEMERGENCE COTTON 4C,8H 3C,7H 3C,8H 2C,8H 2C,8H 3C,8H 2C,7H      2C,6H 9C 5C,9H 10C 5C,9G 3C,9H 8H 8H 0 1H 0 7H 3G MORNING GLORY 10C      5C,9H 5C,9G 4C,8H 4C,9G 3C,8H 4C,9H 4C,8H 10C 10C 10C 10C 4C,9G 3C,5G      3C,6H 0 8H 5G 4C,9H 3C,7H COCKLEBUR 2C,9H 7G 5C,9G 5C,9H 4C,9H 4C,8H      3C,8H 2C,7H 10C 10C 10C 10C 3C,8G 6H 3C,7H 0 7H 0 5G 2G NUTSEDGE 3G 2G      2C,8G 3G 6G 3C 2C,9G 2C,7G 9C 9C 10C 9C 9C 3C,9G 7G 0 0 0 0 0 CRABGRASS      6G 2G 2G 0 0 0 0 0 2G 0 5G 0 0 0 0 0 0 0 3C,5G 4G BARNYARD GRASS 9C      5C,9G 10C 10C 10C 3C,8H 2C,7G 3G 9C 4C,9H 10C 4C,9H 3C,5G 1H 9H 3H 5C,9H      4H 9C 3C,8H WILD OATS 3C,9G 2C,8G 3C,9G 2C,5G 2C,7G 2C,8G 0 0 2C,4G 0 2G      0 0 0 0 0 0 0 4C,8G 3C,6G WHEAT 3C,9G 2C,8G 9G 2C,6G 9G 9G 0 0 2C,5G 0      8G 0 0 0 0 0 0 0 9G 3C,7G CORN 4U,9C 2U,9G 5U,9C 2U,9G 10C 4U,9C 3C,7G      3C,3G 9C 5C,9G 9C 4C,9G 2C,5G 1H 2C,9G 3C,8H 3C,9G 5H 4U,9G 3C,9G      SOYBEAN 5C,8H 4C,9H 4C,9H 4C,7H 4C,9H 3C,8H 2C,8G 7H 5C,9G 4C,9G 4C,9G      3C,9G 1H 0 3C,7H 0 3C,5H 1H 5C,9G 4C,8G RICE 9C 9C 9C 4C,9G 9C 4C,9G 4G      0 7G 0 4C,9G 2G 0 0 6G 5G 5C,9G 7G 9C 9C SORGHUM 10C 5C,9G 9C 3C,9G      5C,9G 4C,9G 2C,8G 2C,6G 9C 3C,9G 5C,9G 9G 9G 3C,6G 3C,9H 4G 3C,8H 2G 9C      3C,9G CHEATGRASS 5C,9G 3C,9G 5C,9G 5C,9G 9C 4C,9G 2C,8G 7G 9C 4C,8G      5C,9G 9C 7G 0 8G 2G 7G 0 5C,9G 9G SUGAR BEETS 2C,7G 0 4C,9G 5C,9H 9C      5C,9G 9C 3C,7H 9C 10C 9C 10C 9C 3C,7G 7H 3G 3C,8H 4H 6G 3H VELVETLEAF      5C,9G 4C,8H 4C,9H 3C,8H 4C,8H 3C,5H 4C,8H 4C,7H 10C 10C 10C 9C 3C,8G 0 0      0 1C 0 4C,7H 6G GIANT FOXTAIL 9C 5C,9G 10C 5C,9G 9C 3C,9G 6G 2G 3C,8G 3G      4C,9G 6G 0 0 0 0 0 0 5C,9G 3C,7G BARLEY 4C,9G 3C,9G 4C,9G 2C,8G 3C,9G      2C,8G 2C,6G 3G 2G 0 7G 0 0 0 0 0 0 0 2G 0 PREEMERGENCE COTTON 1C,3G 0      1C,3G 2G 1C,4G 0 0 0 1C 0 9G 9G 2C,7H 3G 0 0 0 0 1C 0 MORNING GLORY 9G      2C,7G 2C,8H 2C,5G 3C,8H 2G 0 0 2C,2H 0 9G 8G 3H 0 2H 4H 0 0 3H 0      COCKLEBUR 8G 0 3C,7G -- 8H 0 0 0 2C,5G 1C 9H 9H 2C 0 0 0 0 0 1C --      NUTSEDGE 0 0 5G 0 0 0 0 0 0 0 10E 9G 5G 0 0 0 0 0 0 0 CRABGRASS 2C 0 0 0      0 0 0 0 0 0 3G 0 0 0 0 0 0 0 0 0 BARNYARD GRASS 3C,9H 0 2C,4G 0 2C,4G 0      0 0 0 0 3C,9H 5G 7H 0 0 0 0 0 0 0 WILD OATS 2C,8G 2C 2C,4G 3G 2C,7G 3G 0      0 0 0 3C,4G 0 2G 0 0 0 0 0 2C,4G 0 WHEAT 2C,9H 7G 2C,8H 6G 8H 5G 0 0 0 0      5G 0 0 0 0 0 0 0 3C,8G 0 CORN 9H 3C,8G 9H 2C,8G 9H 3C,9G 0 0 3C,4G 0      5C,9H 3C,7G 3C,6G 0 2C,6G 0 5G 0 3C,8H 0 SOYBEAN 3C,7H 2C,5G 1C,6G 4G      2C,8H 1C,3G 2G 0 5G 2C,2H 9H 6H 3H 0 0 0 0 0 3C,8H 2G RICE 10E 7G 10E      2C,7G 10H 2C,4G 2C 0 0 2G 8H 0 7G 0 0 0 5G 0 8G 0 SORGHUM 9C 3C,9H 10C      3C,9H 10C 4C,9G 0 0 3C,7G 3C,3G 9G 9H 2C,8G 3C,5G 6G 0 3C,3G 0 9H 3C,3G      CHEATGRASS 9H 2C,9H 9H 6G 9H 6G 0 0 7G 0 9H 7G 7G 0 0 0 0 0 6G 0 SUGAR      BEETS 5G 5G 5G 0 3C,7G 1C,3G 0 0 7H 2H 9H 9G 7H 0 0 0 2H 0 3H 2H      VELVETLEAF 3C,7H 0 0 0 4G 0 4G 2H 2C 2G 4C,9G 3G 0 0 0 0 0 0 0 0 GIANT      FOXTAIL 2C,8H 0 2C,5G 0 2C,5G 0 0 0 0 0 9G 0 2G 0 0 0 0 0 0 0 BARLEY 9H      7G 9G 2C,8H 4C,9G 2C,8G 0 0 0 0 3C,9G 2G 0 0 0 0 0 0 7H 0        CMPD 194 CMPD 195 CMPD 196 CMPD 197 CMPD 198* CMPD 199 CMPD 200 CMPD      201 CMPD 202 CMPD 203 CMPD 204 CMPD 205 RATE RATE = KG/HA 0.05 0.01 0.05 0      .01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01        COTTON 4C, 2C,4H 4C, 2C,9G 0 0 5H 0 0 0 0 0 3C,9G 3C, 5C,9G 5C,9G 9C      10C 9C 9H 3C,8G 3C, 4C,9H 3C,  8H  9G           8H        5G  9H MORNING      GLORY 4C, 4C,8H 9C 3C,8H 1H 0 0 0 0 0 0 0 4C,9G 4C, 10C 10C 10C 10C      4C,9G 3C, 5C,9G 3C, 4C,9G 3C,  9G             9G      8H  8G  8H      COCKLEBUR 4C, 3C,5G 5C, 4C,9H 2C,3G 0 0 0 0 0 0 0 5C,9G 4C, 10C 10C 10C      10C 5C,9G 3C, 5C,9G 3C, 4C,9H 3C,  9H  9G           9G      8G  8H  8H      NUTSEDGE 2G 0 8G 3C,5G 0 -- 0 0 0 0 0 0 0 0 3C,9G 3C,7G 9G 10C 2C,8G 8G      0 0 5G 0 CRABGRASS 0 0 0 3G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 2G 0      BARNYARD GRASS 3H 0 5H 3C,5H 0 0 0 0 0 0 0 0 2G 0 3C,9H 6H 3C, 6H 1C,2H      0 2C,8H 5H 3C,8H 2C,                  9H       7H WILD OATS 0 0 0 0 0 0      0 0 0 0 0 0 0 0 1C 0 0 0 0 0 2G 0 1C 0 WHEAT 2G 0 0 0 0 0 0 0 0 0 0 0 0      0 2G 0 2G 0 0 0 0 0 0 0 CORN 9G 7H 1C 1C 0 0 0 0 0 0 0 0 2G 0 4C,9G      3C,9H 10C 4C,9G 2C,4G 0 3G 0 0 0 SOYBEAN 8H 4H 4C, 3C,7H 0 0 0 0 0 0 0 0      3C,8G 3C, 4C,8G 3C,8H 5C, 4C,9G 3H 1H 4C,9G 3C, 4C,9G 3C,    9G       4H   9G     8G  5G RICE 7G 4G 3G 2G 4G 0 0 0 0 0 0 0 0 0 3G 0 7G 2G 0 0      6G 1C 9G 2C,                         4G SORGHUM 3C, 2G 4C, 4C,9H 0 0 0 0      0 0 0 0 3C,6G 3G 9G 4C,9G 4C, 4C,9G 3C,8G 2G 3C,7G 1C 3C,9H 3G  8H  9G                 9G CHEATGRASS 5C, 5G 2C, 8G 0 0 0 0 0 0 0 0 6G 3G 4C,9G 7G 9C      9G 6G 0 8G 5G 5C,9G 7G  9G  8G SUGAR BEETS 4C, 2C,3G 9C 5C,8H 0 0 0 0 0      0 2G 0 9C 5C, 10C 10C 10C 9C 3C,9H 4C, 4C,9G 9C 9C 3C,  8G      9G      9G    8H VELVETLEAF 1C 0 3C, 3C,3G 0 0 0 0 0 0 0 0 9C 3C, 10C      10C 10C 10C 5C,9H 3C, 4C,8H 3C, 3C,8H 3C,    7H           8H      8H  6H       5H GIANT FOXTAIL 1H 0 0 1H 0 0 0 0 0 0 0 0 0 0 3G 0 3G 2G 1C 0 2C,5G 0      3C,4G 0 BARLEY 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 2C,2G 0 0 0 0 0 0 0 0 0      PREEMERGENCE COTTON 0 0 3C, 0 0 0 0 0 0 0 0 0 2G 0 3C,6G 0 3C, 7H 6G 0      1C 0 2G 0    5G              9G MORNING GLORY 0 0 6H 0 0 0 0 0 0 0 0 0 0      0 3C,8G 2C 9G 7H 2C,2H 0 0 0 3C,6H 0 COCKLEBUR 0 0 0 2C 0 0 0 0 0 0 0 0      0 0 3C,6H 2C,6H 8H 7H 2C,2H 0 0 0 2C 6G NUTSEDGE 0 0 0 0 0 0 0 0 0 0 0 0      0 0 9G 5G 10E 10E 7G 0 0 0 0 0 CRABGRASS 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0      0 0 0 0 0 0 0 0 BARNYARD GRASS 0 0 1C 0 0 0 0 0 0 0 0 0 0 0 3C,7H 3C,2G      3C, 1H 1C 0 3G 0 3C,4G 0                  8H WILD OATS 0 0 0 0 0 0 0 0 0      0 0 0 2G 0 2G 0 3G 0 0 0 0 0 0 0 WHEAT 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0      4G 0 0 0 0 0 0 0 CORN 0 0 0 0 0 0 0 0 0 0 0 0 0 0 4C,8G 3C,5G 3C, 3C,8G      2C,3G 0 3C,5G 0 3C,7G 1C                  9G SOYBEAN 0 0 3C, 1C 0 0 0 0      0 0 0 0 0 0 2C,3H 1C,2H 4C, 3H 1C 0 1C 0 2C,2H 1H    5G              8H      RICE 0 0 2C, 0 0 0 0 0 0 0 0 0 0 0 5G 0 8G 2G 2G 0 6G 0 9H 3G    4G      SORGHUM 0 0 3C, 3G 0 0 0 0 0 0 0 0 2C,3G 0 4C,9H 3C,6G 3C, 3C,8H 2C,6G 0      3C,9H 3C, 4C,9G 3C,    7G              9H     3G  3G CHEATGRASS 0 0 7G      3G 0 0 0 0 0 0 0 0 5G 0 8G 3C,5G 9G 6G 3G 0 4G 0 8H 0 SUGAR BEETS 0 0      4C, 5G 0 0 0 0 0 0 0 0 3C,8G 0 5C,9G 3C,8G 5C, 8G 3C,8G 3H 3C,8H 2H      4C,9G 3H    8G              9G VELVETLEAF 0 0 2C 0 0 0 0 0 0 0 0 0 0 0      3C,5H 3C 3C, 3C,3G 2G 0 0 0 1C 0                  8G GIANT FOXTAIL 0 0 0      0 0 0 0 0 0 0 0 0 0 0 2G 0 2G 0 0 0 2G 0 0 0 BARLEY 0 0 0 0 0 0 0 0 0 0      0 0 0 0 2G 0 2C, 0 2G 0 0 0 2C,2G 0                  4G      *It is noted that Compound 198 was inactive at the levels tested. However      it is believed that at higher levels, herbicidal activity would be      present.

TEST B Postemergence

Two round pans (25 cm diameter by 12.5 cm deep) were filled with Sassafras sandy loam soil. One pan was planted with blackgrass, (Alopecurus myosuroides), sugar beets, nutsedge (Cyperus rotundus) tubers, rape (Brassica napus), crabgrass (Digitaria sanguinalis), sicklepod (Cassia obtusifolia), teaweed (Sida spinosa), jimsonweed (Datura stramonium), velvetleaf (Abutilon theophrasti), and giant foxtail (Seteria faberii). The other pan was planted with wheat, barley, cotton, rice, corn, soybean, wild oats (Avena fatua), cocklebur (Xanthium pensylvanicum), morningglory (Ipomoea hederacea), johnsongrass (Sorghum halepense) and barnyardgrass (Echinochloa crusgalli). The plants were grown for approximately fourteen days, then sprayed postemergence with the chemicals dissoled in a non-phytotoxic solvent.

Preemergence

Two round pans (25 cm diamater by 12.5 cm deep )were filled with Sassafras sandy loam soil. One pan was planted with blackgrass, sugar beets, nutsedge, rape, crabgrass, sicklepod, teaweed, jimsonweed, velvetleaf, and giant foxtail. The other pan was planted with wheat, barley, cotton, rice, corn, soybean, wild oats, cocklebur, morningglory, johnsongrass, and barnyardgrass. The two pans were sprayed preemergence with the chemicals dissolved in a non-phytotoxic solvent.

Treated plants and controls were maintained in the greenhouse for 28 days, then all treated plants were compared to controls and visually rated for plant response. Response ratings are based on a scale of 0 to 100 where 0=no effect, and 100=complete control. A dash (-) response means no test.

Response ratings are contained in Table B.

    TABLE B       Compound 2 Compound 3 Compound 4 Compound 5 POSTEMERGENCE Rate g/ha 62      16 16 4 4 1 .25 62 16 16 16 4 4 4 1 1 .25 .25 62 16 4 1 62 16 4 1        Corn 100 100 100 100 100 60 40 100 100 100 100 100 90 100 80 70 60 0      100 100 80 40 100 90 60 40 Wheat 100 100 100 60 100 40 0 100 100 30 70      40 0 20 0 0 0 0 100 100 40 0 70 40 0 0 Barley -- -- -- -- -- -- -- -- --      -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- Rice 100 100 100 90      70 50 30 100 100 80 100 90 60 100 50 30 30 0 100 100 60 30 100 90 30 0      Soybean 100 100 100 100 90 90 60 100 100 100 100 100 90 90 80 70 80 0      100 100 100 60 90 90 60 40 Cotton 100 100 60 70 20 40 0 100 100 100 100      100 80 100 70 40 30 0 100 90 70 30 100 90 60 30 Sugar beet 100 100 100      100 100 100 100 100 100 100 100 100 100 100 100 100 100 0 100 100 100      100 100 100 100 90 Rape 100 100 100 100 100 100 100 100 100 100 100 100      100 100 100 100 100 0 100 100 100 100 100 100 100 100 Crabgrass 100 80      100 50 60 40 0 100 90 50 70 70 30 30 50 0 30 0 100 80 50 30 70 50 40 30      Johnsongrass 100 100 100 100 90 60 40 100 100 100 100 100 70 90 70 30 30      0 100 100 70 30 100 100 80 40 Blackgrass 100 100 100 100 90 50 30 100      100 100 100 100 60 100 80 30 70 0 100 100 60 30 100 100 60 30 Barnyardgra      ss 100 100 100 100 100 60 40 100 100 100 100 100 70 100 100 30 40 0 100      100 60 30 100 100 80 40 Nutsedge 100 100 100 100 80 90 80 100 100 100      100 100 100 100 100 100 100 0 100 90 50 30 100 100 80 70 Giant Foxtail      100 100 100 90 90 50 30 100 100 80 60 60 30 30 30 0 0 0 100 90 60 30 100      80 30 0 Green Foxtail Cheatgrass Wild Oats 90 100 80 60 70 40 0 100 100      50 100 40 0 80 0 0 0 0 100 90 30 0 70 40 0 0 Wild Buckwheat Viola      Lambsquarter Cocklebur 100 100 90 70 60 30 0 100 100 90 100 100 70 90 60      60 30 0 100 90 50 30 100 100 60 30 Morningglory 100 100 90 100 70 90 60      100 100 100 100 100 100 100 100 80 70 0 100 100 80 50 100 90 80 60      Teaweed 100 100 90 70 30 40 0 100 100 60 90 80 30 60 50 0 30 0 100 80 60      40 90 70 50 30 Sicklepod 100 100 100 90 70 60 0 100 100 100 100 100 100      100 90 100 80 0 100 80 60 30 70 60 40 30 Jimsonweed 100 100 100 90 70 70      40 100 100 90 100 90 60 100 70 30 40 0 100 100 70 40 100 90 60 30      Velvetleaf 100 100 100 100 80 80 50 100 100 90 100 100 80 100 90 50 50 0      100 100 100 60 100 100 60 30        PREEMERGENCE Rate g/ha 250 62 62 16 16 4 1 250 62 62 16 16 16 4 4 1 1      250 62 16 4 250 62 16 4        Corn 100 100 100 80 90 20 0 100 100 100 70 70 100 20 40 0 0 100 100 90      60 100 100 90 30 Wheat 100 90 100 80 100 30 0 100 100 100 20 0 40 0 0 0      0 100 100 90 70 100 100 50 0 Barley -- -- -- -- -- -- -- -- -- -- -- --      -- -- -- -- -- -- -- -- -- -- -- -- -- Rice 100 100 100 100 100 90 70      100 100 100 100 100 100 100 100 90 0 100 100 100 100 100 100 100 100      Soybean 100 100 100 80 100 40 20 100 100 100 70 70 90 40 40 0 0 100 100      90 60 100 90 80 60 Cotton 100 80 100 80 80 30 0 100 100 100 70 70 100 30      0 0 0 100 90 60 30 100 80 50 30 Sugar beet 100 100 100 100 100 100 30      100 100 100 100 100 100 100 90 80 0 100 100 100 90 100 100 100 80 Rape      100 100 100 90 100 20 0 100 100 100 90 90 100 90 80 20 0 100 100 100 50      100 100 80 60 Crabgrass 100 100 100 90 90 30 0 100 90 100 60 30 80 30 0      0 0 100 90 50 30 90 70 50 30 Johnsongrass 100 100 100 100 100 90 30 100      100 100 90 70 100 80 30 50 0 100 100 100 70 100 100 100 100 Blackgrass      100 90 100 100 100 70 20 100 100 100 100 90 100 100 70 50 0 100 100 100      90 100 100 100 90 Barnyardgrass 100 100 100 90 100 80 20 100 100 100 80      50 100 30 0 0 0 100 100 100 60 100 100 90 70 Nutsedge 100 100 100 100      100 70 20 100 100 100 100 90 100 90 50 50 0 100 90 80 60 100 100 100 90      Giant Foxtail 100 100 100 90 100 80 50 100 100 100 80 30 100 50 0 0 0      100 100 100 60 100 100 90 60 Green Foxtail Cheatgrass Wild Oats 100 90      100 90 90 20 0 100 100 100 70 90 80 0 40 0 0 100 90 70 70 90 80 50 30      Wild Buckwheat Viola Lambsquarter Cocklebur 100 90 100 80 90 20 0 100      100 100 50 80 80 50 40 20 0 100 100 80 50 100 90 70 50 Morningglory 100      50 100 40 70 0 0 100 100 100 40 80 100 30 40 0 0 100 90 50 30 100 80 70      30 Teaweed 100 100 100 80 90 50 20 100 100 100 80 70 90 70 30 0 0 100 90      70 30 90 70 50 30 Sicklepod 100 90 100 80 80 60 20 100 90 100 90 50 90      80 30 20 0 100 90 60 30 90 70 50 50 Jimsonweed 100 100 100 90 90 60 20      100 100 100 100 80 100 80 30 50 0 100 90 80 50 100 90 60 30 Velvetleaf      100 100 100 100 100 60 0 100 100 100 100 80 100 90 30 60 0 100 100 80 50      100 90 60 30        Compound 8 Compound 13 Compound 14 Compound 16 Compound 20 Compound 21 C      ompound 22 Compound 23 POSTEMERGENCE Rate g/ha 62 16 4 1 62 16 4 1 16 4      1 .25 62 16 4 1 62 16 4 62 16 4 62 16 4 62 16        Corn 100 80 50 30 100 100 70 40 100 80 60 40 0 0 0 0 100 90 40 100 90      70 100 100 70 50 30 Wheat 30 0 0 0 30 0 0 0 30 0 0 0 0 0 0 0 90 60 20 0      0 0 70 20 0 40 0 Barley -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- --      -- -- -- 0 0 0 0 0 0 -- -- Rice 90 70 0 0 90 30 0 0 60 30 0 0 60 0 0 0      95 90 85 80 20 0 90 50 20 70 40 Soybean 100 80 70 0 100 100 100 70 100      100 70 60 100 70 40 0 95 90 80 100 90 50 100 100 80 100 100 Cotton 100      90 60 40 100 100 90 50 100 70 50 30 90 70 50 30 100 100 90 60 0 0 80 70      20 100 100 Sugar beet 100 100 100 90 100 100 100 100 100 100 90 70 100      100 90 70 95 90 90 90 80 0 100 90 70 100 100 Rape 100 100 100 90 100 100      100 100 100 100 90 60 100 100 90 60 100 100 100 100 90 30 100 100 70 100      100 Crabgrass 90 50 30 0 90 60 50 30 30 0 0 0 30 0 0 0 60 30 20 40 0 0      60 30 0 60 40 Johnsongrass 90 50 0 0 100 90 60 30 100 80 60 30 90 70 30      0 100 100 85 100 70 20 100 100 70 100 100 Blackgrass 100 90 30 0 100 70      40 0 70 30 0 0 70 30 0 0 100 95 85 80 60 0 100 70 50 100 70 Barnyardgrass       90 50 0 0 100 90 60 30 100 80 50 30 90 50 0 0 100 95 80 100 70 30 100      100 50 100 100 Nutsedge 100 70 70 40 100 100 90 80 90 70 50 30 90 70 60      40 100 80 60 0 0 0 0 0 0 100 100 Giant Foxtail 90 50 0 0 100 80 30 0 70      30 0 0 0 0 0 0 90 85 60 100 60 20 100 100 50 70 50 Green Foxtail                 70 20 0 100 80 50 Cheatgrass                    0 0 0 0 0 0      Wild Oats 30 0 0 0 60 30 0 0 40 0 0 0 0 0 0 0 85 70 30 0 0 0 60 20 0 40      0 Wild Buckwheat                    100 80 0 80 80 50 Viola            40 20 0 80 -- 20 Lambsquarter                    90 50 0 80 60 50      Cocklebur 100 90 50 30 100 70 50 30 100 90 60 30 90 80 50 30 100 95 85      60 0 0 100 60 20 100 100 Morningglory 100 90 60 30 100 100 100 50 90 70      50 30 90 80 60 30 100 100 90 50 0 50 70 60 20 100 80 Teaweed 100 70 30      30 100 90 60 40 90 50 30 0 70 30 30 0 90 95 90 40 20 0 70 50 20 90 70      Sicklepod 90 50 30 0 100 100 80 40 80 50 0 0 50 30 0 0 70 25 30 50 0 0      80 50 20 100 70 Jimsonweed 100 100 60 30 100 100 60 30 90 90 50 30 100      80 50 30 95 90 30 80 70 20 90 70 50 100 100 Velvetleaf 100 100 70 50 100      100 100 70 100 90 50 30 100 80 30 0 100 100 90 30 0 0 70 30 20 100      100     PREEMERGENCE Rate g/ha 250 62 16 4 250 62 16 4 62 16 4 1 250 62      16 4 250 62 16 250 62 16 250 62 16 250 62        Corn 100 90 30 0 100 90 90 20 90 70 50 30 80 50 30 0 100 95 90 90 60      20 90 80 0 70 50 Wheat 80 30 0 0 30 0 0 0 80 40 0 0 90 40 0 0 95 95 80      40 0 0 50 0 0 80 60 Barley -- -- -- -- -- -- -- -- -- -- -- -- -- -- --      -- -- -- -- 0 0 0 60 20 0 -- -- Rice 100 100 100 20 100 100 100 70 100      100 70 40 100 100 90 60 100 100 100 -- -- -- -- -- -- 100 100 Soybean      100 80 40 0 100 100 90 70 100 90 70 60 100 80 60 30 95 95 85 80 80 30 90      80 30 100 80 Cotton 100 60 20 0 100 80 80 20 80 70 50 30 90 70 50 30 95      90 80 90 20 0 90 80 20 90 70 Sugar beet 100 100 100 50 100 100 100 90      100 100 100 80 100 100 100 100 100 95 90 90 70 50 80 70 80 100 100 Rape      100 100 90 40 100 100 90 90 100 100 60 60 100 90 60 0 100 95 80 80 60 0      90 80 70 100 90 Crabgrass 80 70 40 20 90 70 50 0 90 70 50 30 90 70 50 40      90 30 10 90 0 0 70 70 20 90 70 Johnsongrass 100 90 60 20 100 100 100 60      100 80 50 30 100 80 50 30 95 95 90 100 80 0 100 90 80 100 90 Blackgrass      100 90 70 30 100 90 80 50 100 90 60 30 100 90 60 30 100 95 80 100 50 0      90 70 70 100 100 Barnyardgrass 100 90 20 0 100 100 90 60 100 70 50 0 100      80 40 0 100 95 90 100 50 0 100 90 50 100 80 Nutsedge 100 100 80 60 100      100 100 90 100 100 90 80 100 100 100 90 100 100 100 0 0 0 0 0 0 100 100      Giant Foxtail 100 90 -- 0 100 90 70 50 100 60 40 0 80 60 30 0 100 95 90      90 70 0 100 90 70 100 100 Green Foxtail                    90 90 30 100      90 50 Cheatgrass                    50 0 0 60 0 0 Wild Oats 100 90 80 0      -- -- -- -- 80 40 0 0 90 40 0 0 90 85 65 60 20 0 50 50 20 70 50 Wild      Buckwheat                    100 50 50 90 60 20 Viola      100 -- 20 90 50 30 Lambsquarter                    90 70 0 90 60 0      Cocklebur 100 80 20 0 100 70 80 20 100 90 70 50 100 80 70 30 95 90 90 30      20 0 -- 30 0 90 80 Morningglory 100 60 20 0 100 90 80 30 90 70 50 30 100      80 50 30 95 90 80 70 20 0 80 60 20 70 50 Teaweed 100 90 90 20 100 90 90      20 90 80 50 30 90 80 50 30 90 80 50 80 30 0 70 40 0 90 70 Sicklepod 100      90 30 0 100 100 80 20 90 70 50 30 90 70 50 30 90 50 10 50 0 0 70 30 0 90      70 Jimsonweed 100 100 80 30 100 100 90 50 90 70 50 30 90 70 50 30 100 90      60 60 0 0 70 30 0 100 80 Velvetleaf 100 100 60 20 100 100 90 80 90 70 50      30 90 70 50 30 100 95 70 30 0 0 60 30 0 100 80        Compound 23 Compound 24 Compound 27 Compound 28  Compound 31 Compound      32 Compound 33 POSTEMERGENCE Rate g/ha 4 1 62 16 4 1 250 62 16 4 250 62      16 62 16 4 1 62 16 4 1 62 16 4        Corn 0 0 0 0 0 0 0 0 0 0 0 0 0 100 70 50 30 80 40 0 0 80 40 30 Wheat 0      0 30 0 0 0 40 20 0 0 30 0 0 0 0 0 0 80 60 40 20 90 70 30 Barley -- -- --      -- -- -- -- -- -- --    -- -- -- -- -- -- -- -- -- -- -- Rice 0 0 30 0 0      0 90 70 50 30 50 30 0 70 30 0 0 100 70 50 30 80 70 30 Soybean 80 60 100      100 80 60 90 80 70 50 80 60 40 100 90 70 40 100 100 90 70 90 90 70      Cotton 70 40 100 90 70 40 100 90 60 30 100 70 30 80 60 30 0 100 100 100      80 90 90 50 Sugar beet 100 100 100 100 100 90 100 100 100 100 100 100      100 100 100 60 30 100 100 70 50 100 100 80 Rape 100 100 100 100 100 100      100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100      Crabgrass 30 0 30 0 0 0 70 50 30 0 50 30 0 90 70 50 30 90 70 50 30 60 30      0 Johnsongrass 80 60 100 70 50 30 100 90 70 50 90 70 50 100 100 60 30      100 100 100 80 100 100 60 Blackgrass 30 0 100 100 70 40 90 60 30 0 100      90 70 100 100 60 30 100 100 90 70 90 70 30 Barnyardgrass 80 60 80 60 30      100 90 70 50 90 60 30 100 100 70 30 100 100 100 90 100 70 50 Nutsedge 70      50 100 90 70 50 100 100 70 50 70 50 30 30 0 0 0 100 100 100 90 100 60 50      Giant Foxtail 30 0 70 30 0 0 70 50 30 0 80 60 30 100 100 70 40 100 90 70      50 90 70 50 Green Foxtail Cheatgrass Wild Oats 0 0 30 0 0 0 60 40 20 0      30 0 0 70 40 20 0 80 60 40 20 80 40 30 Wild Buckwheat Viola Lambsquarter      Cocklebur 100 100 100 100 100 90 100 90 70 50 90 70 50 90 70 50 30 100      100 100 70 100 80 60 Morningglory 60 30 100 90 70 50 90 80 70 50 100 100      70 90 70 50 30 100 100 90 70 100 100 50 Teaweed 50 30 70 50 30 0 80 60      40 20 80 60 40 80 60 30 0 100 80 60 30 80 50 30 Sicklepod 50 30 70 50 30      0 80 60 30 0 50 30 0 80 60 30 0 100 100 90 80 90 50 30 Jimsonweed 70 50      100 70 50 30 100 70 0 30 100 80 60 100 80 60 40 100 90 80 70 90 80 60      Velvetleaf 100 90 100 100 70 50 100 100 80 50 100 80 50 100 80 60 40 100      100 100 90 100 100 90        PREEMERGENCE Rate g/ha 16 4 250 62 16 4 250 62 16 4 250 62 16 4 250 62 1      6 4 250 62 16 4 250 62 16 4        Corn 30 0 30 0 0 0 0 0 0 0 0 0 0 0 90 60 0 0 90 80 70 40 40 0 0 0      Wheat 40 0 70 30 0 0 70 50 30 0 70 30 0 0 60 30 0 0 80 60 40 20 90 40 0      0 Barley -- -- -- -- -- -- -- -- -- -- 70 30 0 0 -- -- -- -- -- -- -- --      -- -- -- -- Rice 80 50 90 70 50 30 100 90 70 50 100 90 60 30 100 100 90      70 100 100 100 100 100 100 30 0 Soybean 60 40 90 70 50 30 70 50 30 0 90      60 30 0 90 70 50 30 100 80 60 40 90 60 30 0 Cotton 40 0 70 50 30 0 50 30      0 0 70 30 0 0 80 40 0 0 90 70 50 30 80 60 30 0 Sugar beet 100 80 100 100      90 80 100 90 70 50 90 70 50 30 100 90 70 50 100 100 90 70 100 80 40 0      Rape 70 50 100 90 70 50 90 70 50 30 90 70 50 30 90 70 50 20 100 90 70 50      90 70 50 30 Crabgrass 50 30 90 60 30 0 80 70 60 30 70 50 30 0 90 60 30 0      90 80 70 60 70 50 30 0 Johnsongrass 80 60 90 80 70 50 90 80 70 40 100 90      70 50 100 80 60 40 100 100 90 70 100 90 70 50 Blackgrass 80 50 90 80 70      40 90 70 50 30 90 70 50 30 100 90 70 50 90 80 70 50 90 70 30 0 Barnyardgr      ass 60 40 90 80 60 30 90 60 30 0 90 70 50 30 90 80 60 30 100 90 70 40      100 70 30 0 Nutsedge 80 60 100 80 60 40 90 70 50 30 100 70 50 30 80 60      40 20 100 90 80 70 90 70 50 30 Giant Foxtail 90 70 100 90 70 40 90 60 40      0 90 70 $0 30 100 80 60 30 100 100 80 60 100 80 50 30 Green Foxtail           90 70 50 30 Cheatgrass           60 30 0 0 Wild Oats 30 0 70 40 30      0 80 60 30 0 30 0 0 0 60 30 0 0 90 70 50 30 80 30 0 0 Wild Buckwheat            90 70 50 30 Viola           90 70 50 30 Lambsquarter           100      70 50 30 Cocklebur 70 50 90 70 50 30 80 60 40 0 90 70 50 30 90 70 50 30      90 70 50 30 90 60 30 0 Morningglory 30 0 80 60 40 20 30 0 0 0 90 60 30 0      80 60 40 20 100 90 60 30 90 60 30 0 Teaweed 50 -- 90 70 50 30 90 70 50      30     70 50 30 0 100 80 60 40 60 30 0 0 Sicklepod 40 0 90 70 40 0 90 70      40 0 40 0 0 0 80 60 40 0 100 80 40 0 90 60 30 0 JimsonWeed 60 40 90 70      50 30 90 70 50 30 90 70 50 30 90 70 50 30 90 80 70 50 90 70 50 30      Velvetleaf 60 40 90 70 50 30 90 70 50 30 90 70 50 30 90 70 50 30 90 80      70 50 80 60 40 20        Compound 34 Compound 35 Compound 36 Compound 39 Compound 40 Compound      46 Compound 53 POSTEMERGENCE Rate g/ha 62 16 4 1 62 16 4  1 62 16 4 1 62 1      6 4 1 62 16 4 1 62 16 4 1 62 16 4 1        Corn 70 30 0 0 30 0 0 0 90 70 30 0 100 100 70 30 80 20 0 0 100 80 50 0      0 0 0 0 Wheat 60 30 0 0 40 0 0 0 80 50 30 0 100 100 80 50 90 80 20 0 80      70 20 0 60 30 0 0 Barley -- -- -- -- -- -- -- -- -- -- -- -- 100 80 40 0      20 0 0 0 90 80 50 0 60 30 0 0 Rice 90 70 50 30 100 70 30 0 90 70 50 30      100 100 80 30 90 60 30 0 100 100 70 20 90 60 30 0 Soybean 90 90 80 60 90      80 60 50 100 80 60 40 100 100 90 70 100 80 80 50 100 90 80 60 100 90 80      70 Cotton 90 80 50 30 100 80 40 0 90 70 40 0 70 30 30 0 70 60 30 0 100      60 50 0 90 60 20 0 Sugar beet 100 100 70 50 100 100 100 70 100 100 100      70 100 90 40 20 70 50 0 0 100 100 60 20 100 100 100 90 Rape 100 100 100      100 100 100 100 100 0 0 0 0 100 100 100 80 100 100 70 50 100 100 90 50      100 100 100 100 Crabgrass 80 50 30 0 60 30 0 0 90 60 30 0 90 50 20 0 40      0 0 0 60 30 0 0 70 50 30 0 Johnsongrass 100 90 70 30 100 100 70 40 100      90 60 30 100 100 70 50 80 50 20 0 90 100 80 20 100 90 70 50 Blackgrass      100 70 30 0 100 80 30 0 100 100 70 30 90 100 70 60 80 50 20 0 100 90 60      0 100 90 60 30 Barnyardgrass 100 70 50 0 100 100 70 30 100 90 70 30 100      100 90 60 90 60 20 0 100 100 80 20 100 100 90 60 Nutsedge 90 70 50 30 90      70 50 30 0 0 0 0 70 80 30 0 50 0 0 0 30 -- -- 0 -- -- -- -- Giant      Foxtail 90 70 60 0 90 80 50 30 90 70 50 30 90 40 20 0 60 30 0 0 100 80      40 0 100 90 70 50 Green Foxtail             100 70 50 0 60 30 20 0 100      80 60 0 90 70 50 30 Cheatgrass             100 100 60 50 80 70 50 0 40      20 0 0 100 90 70 50 Wild Oats 70 50 30 0 50 0 0 0 90 60 30 0 100 100 90      40 100 40 0 0 90 90 30 0 30 0 0 0 Wild Buckwheat             100 90 70 0      70 0 0 0 100 100 80 0 100 90 70 50 Viola             70 80 80 30 80 --      -- -- 90 70 30 30 100 90 70 50 Lambsquarter             100 90 50 20 90      70 20 0 100 100 80 50 100 90 70 50 Cocklebur 90 70 30 0 100 90 50 30 30      0 0 0 100 100 100 30 100 90 80 0 100 70 20 0 100 90 70 50 Morningglory      90 80 60 40 100 90 50 30 100 90 70 50 100 100 90 30 100 100 70 30 100      100 80 60 100 100 90 60 Teaweed 80 50 30 0 90 60 30 0 70 50 30 0 90 50      20 0 60 50 30 0 80 60 40 0 90 70 50 30 Sicklepod 90 50 30 0 90 40 0 0 90      60 30 0 100 100 50 0 100 30 30 20 100 90 70 0 100 100 70 50 Jimsonweed      100 80 70 50 100 80 50 30 80 60 40 0 100 100 70 50 90 70 50 0 100 90 80      20 100 90 70 50 Velvetleaf 100 100 80 60 100 100 70 30 80 60 40 0 100 90      60 20 100 80 60 0 100 90 60 20 100 100 80 60        PREEMERGENCE Rate g/ha 250 62 16 4 250 62 16 4 250 62 16 4 250 62 16 4 2      50 62 16 4 250 62 16 4 250 62 16 4        Corn 60 0 0 0 30 0 0 0 70 30 0 0 100 80 70 20 80 20 0 0 90 80 0 0 0 0      0 0 Wheat 70 30 0 0 80 60 30 0 60 30 0 0 90 70 60 0 80 60 0 0 90 70 40      20 70 40 20 0 Barley -- -- -- -- -- -- -- -- -- -- -- -- 90 80 20 0 0 0      0 0 90 90 50 0 60 40 20 0 Rice 100 100 40 0 100 100 100 70 100 100 100      90 100 100 90 60 100 80 50 0 100 100 90 80 90 80 70 30 Soybean 90 50 0 0      90 80 70 30 80 40 0 0 100 100 60 60 100 50 30 0 90 80 40 0 90 80 60 30      Cotton 60 30 0 0 90 70 50 30 40 0 0 0 80 70 20 0 30 0 0 0 90 70 40 0 60      50 30 0 Sugar beet 100 90 70 50 100 100 90 70 100 90 70 50 100 100 60 20      90 80 60 0 100 90 70 50 100 90 80 70 Rape 90 70 40 0 100 90 60 30 80 60      40 0 100 100 90 20 100 90 40 0 100 100 80 50 100 90 70 50 Crabgrass 70      50 40 30 80 60 50 30 100 70 50 30 100 90 70 20 100 80 20 0 90 50 30 0 90      70 50 30 Johnsongrass 90 70 40 0 100 100 90 70 100 90 70 40 100 100 90      80 100 100 90 80 100 70 50 30 90 80 70 30 Blackgrass 100 80 40 0 100 100      90 50 100 100 80 60 100 90 90 50 100 90 70 50 90 90 50 30 100 70 50 30      Barnyardgrass 90 40 0 0 100 90 80 50 100 80 40 0 100 90 70 30 100 90 80      0 90 70 40 0 90 80 70 30 Nutsedge 90 70 50 30 100 100 70 50 70 50 30 0      100 -- -- -- -- -- 0 -- 90 70 50 30 90 80 70 50 Giant Foxtail 90 50 0 0      100 90 80 50 100 90 70 40 100 90 70 30 100 90 70 0 90 80 50 30 90 80 70      30 Green Foxtail             100 90 80 70 100 100 40 0 90 80 50 30 90 70      50 30 Cheatgrass             100 100 90 70 100 90 70 60 90 80 30 20 90      80 70 30 Wild Oats 70 30 0 0 80 60 30 0 70 40 0 0 90 90 60 20 90 30 0 0      70 60 30 0 40 20 0 0 Wild Buckwheat             100 90 80 70 100 70 60      20 100 80 60 30 90 80 70 50 Viola             100 100 90 20 90 80 20 0      100 100 100 90 100 90 70 50 Lambsquarter             100 100 90 60 100      100 80 70 100 100 70 50 90 70 50 30 Cocklebur 90 50 30 0 90 80 50 40 --      0 0 0 100 80 70 0 90 -- -- -- 40 0 0 0 90 70 50 30 Morningglory 80 50 30      0 90 80 60 30 80 60 30 0 100 90 40 0 90 70 20 0 90 80 70 50 90 80 70 60      Teaweed 80 50 30 0 90 70 40 0 90 70 50 20 100 90 60 30 90 90 50 0 90 70      50 30 90 70 50 30 Sicklepod 70 30 0 0 50 30 0 0 90 70 50 30 100 80 30 0      80 0 0 0 50 30 0 0 90 80 70 60 Jimsonweed 90 70 50 30 100 80 50 30 90 70      40 20 100 90 70 50 100 40 20 0 90 70 50 30 90 80 70 50 Velvetleaf 80 70      50 30 90 80 50 30 90 70 50 20 100 90 50 20 90 30 0 0 90 70 50 30 90 70      50 30        Compound 54 Compound 55 Compound 56 POSTEMERGENCE Rate g/ha 62 16 4 1      62 16 4 1 62 16 4 1        Corn 0 0 0 0 0 0 0 0 0 0 0 0 Wheat 80 60 40 20 90 60 30 0 40 20 0 0      Barley 60 30 0 0 70 40 0 0 20 0 0 0 Rice 90 60 30 0 90 60 30 0 80 60 30      0 Soybean 100 90 70 50 90 80 70 50 70 30 0 0 Cotton 90 70 20 0 90 60 0 0      40 0 0 0 Sugar beet 100 100 90 70 100 100 90 70 100 90 70 50 Rape 100      100 100 90 100 100 100 80 100 100 90 80 Crabgrass 60 30 0 0 80 60 40 20      50 30 0 0 Johnsongrass 100 90 70 50 100 90 70 50 90 70 50 30 Blackgrass      100 90 70 50 100 90 70 50 90 70 50 30 Barnyardgrass 100 90 70 50 100 100      70 50 90 70 50 30 Nutsedge -- -- -- -- -- -- -- -- -- -- -- -- Giant      Foxtail 90 70 50 30 90 80 70 30 90 60 30 0 Green Foxtail 90 70 50 30 90      70 50 30 90 70 50 30 Cheatgrass 100 70 50 30 100 90 70 50 90 70 50 30      Wild Oats 30 0 0 0 70 30 0 0 0 0 0 0 Wild Buckwheat 90 70 50 30 100 90      80 60 90 70 50 30 Viola 90 70 50 30 100 90 70 50 -- 70 50 30 Lambsquarter       100 90 70 50 100 90 70 50 90 70 50 30 Cocklebur 100 90 70 50 100 90 70      50 90 70 50 30 Morningglory 100 70 50 30 100 80 60 30 100 60 30 0      Teaweed 90 70 50 30 90 70 50 30 90 70 50 30 Sicklepod 100 70 50 30 100      70 50 30 70 50 30 0 Jimsonweed 100 90 70 50 90 80 60 30 90 70 50 30      Velvetleaf 100 90 70 50 100 90 70 40 100 70 50 30        PREEMERGENCE Rate g/ha 250 62 16 4 250 62 16 4 250 62 16 4        Corn 0 0 0 0 0 0 0 0 0 0 0 0 Wheat 80 50 30 0 80 40 0 0 80 40 0 0      Barley 50 30 0 0 80 30 0 0 0 0 0 0 Rice 90 70 50 30 100 70 50 30 90 80      70 40 Soybean 80 60 30 0 90 70 30 0 80 60 30 0 Cotton 80 40 0 0 90 60 30      0 70 0 0 0 Sugar beet 100 90 80 70 100 90 80 70 100 90 80 70 Rape 90 80      70 50 90 80 70 40 100 90 80 70 Crabgrass 70 50 30 0 70 50 30 0 70 50 30      0 Johnsongrass 90 70 50 30 90 80 70 50 100 90 80 60 Blackgrass 90 80 70      50 100 100 90 80 90 80 70 50 Barnyardgrass 90 80 70 40 90 80 70 40 100      80 70 50 Nutsedge 100 90 70 50 90 80 70 50 90 80 70 50 Giant Foxtail 90      80 70 40 90 80 60 30 90 80 70 40 Green Foxtail 90 80 70 50 90 80 70 50      90 80 70 50 Cheatgrass 90 80 70 50 90 80 70 40 90 80 70 50 Wild Oats 40      0 0 0 50 30 0 0 30 0 0 0 Wild Buckwheat 90 80 70 50 90 80 70 50 90 70 60      40 Viola 100 100 90 70 100 100 90 70 100 100 90 80 Lambsquarter 90 80 70      50 90 70 50 30 90 0 50 30 Cocklebur 90 70 50 30 100 70 50 30 100 70 50      30 Morningglory 90 80 70 50 100 90 60 30 90 70 50 30 Teaweed 90 70 50 30      90 70 50 30 90 70 50 30 Sicklepod 90 70 50 30 90 70 50 30 100 70 50 30      Jimsonweed 100 70 50 30 90 70 50 30 90 70 50 30 Velvetleaf 90 70 50 30      90 70 50 30 90 70 60 50

TEST C

The Corn and Sorghum Herbicide Test included the following species in both the preemergence and postemergence evaluations:

    ______________________________________                                                 SPECIES                                                                Category  Common Name  Scientific Name                                         ______________________________________                                         Crops     Corn         Zea mays                                                          Soybean      Glycine max                                                       Sorghum      Sorghum bicolor                                         Grasses   Green foxtail                                                                               Setaria viridis                                                   Giant foxtail                                                                               Setaria faberii                                                   Johnsongrass Sorghum halepense                                                 Barnyardgrass                                                                               Echinochloa crus-galli                                            Fall Panicum Panicum dichotomiflorum                                           Crabgrass    Digitaria sanguinalis                                             Nutsedge     Cyperus rotundus                                        Broadleaves                                                                              Cocklebur    Xanthium pensylvanicum                                            Morningglory Ipomoea hederacea                                                 Velvetleaf   Abutilon theophrasti                                              Jimsonweed   Datura stramonium                                                 Lambsquarters                                                                               Chenopodium album                                                 Pigweed      Amaranthus retroflexus                                            Smartweed    Polygonum persicaris                                    ______________________________________                                    

Postemergence

Postemergence plants were grown in Sassafras sandy loam soil. Corn and soybeans were grown in separate 25 cm diameter containers. Sorghum and the seven grass weed species were grown in two 18 cm diameter containers, 4 species per container. The seven broadleaf weed species were also grown in two 18 cm diameter containers, 4 species in one container, 3 species in the second container. One additional planting of corn in an 18 cm diameter container was made. The soil surface of this additional container of corn was covered with the absorbent, perlite, before spray treatment so that test chemicals would enter the plant only via the foliage. The plants were grown 10-21 days, dependent upon the species and then sprayed postemergence with the test chemicals dissolved in a non-phytotoxic solvent.

Preemergence

Preemergence plantings were grown in fertilized Tama silt loam soil. These plants are identical to those described in the postemergence section, with the exception of the corn planting having perlite covering the soil surface. These plantings were made the day of or the day before spraying the test chemicals dissolved in a non-phytotoxic solvent.

Evaluation

Treated plants and control were maintained in the greenhouse for 2 to 4 weeks. Visual planting response ratings were made on a percentage scale of 0 to 100 in comparison with a control where 0=no injury, and 100=death.

                                      TABLE C                                      __________________________________________________________________________     RATE     Compound 35          Compound 53          Compound 163                RATE GM  0004                                                                              0008                                                                              0016                                                                              0031                                                                              0062                                                                              0125                                                                              0250                                                                              0004                                                                              0008                                                                              0016                                                                              0031                                                                              0062                                                                              0125                                                                              0250                                                                              0004                                                                              0008                                                                              0016                                                                              0031               __________________________________________________________________________     POSTEMERGENCE                                                                  CORN     0  0  0  0  25 45 -- 0  0  0  0  25 45 -- 0  0  0  20                 SOYBEAN  45 70 85 100                                                                               100                                                                               100                                                                               -- 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 100                                                                               100                                                                               100                                                                               100                GREEN FXTL                                                                              45 55 70 85 95 100                                                                               -- 30 40 55 75 85 95 -- 60 80 90 100                GIANT FXTL                                                                              40 45 60 75 95 100                                                                               -- 35 50 75 90 100                                                                               100                                                                               -- 60 80 95 100                PANICUM  90 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 80 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 90 100                                                                               100                                                                               100                CRABGRASS                                                                               0  0  0  30 45 55 -- 0  0  0  30 45 60 -- 0  25 40 85                 BARNYARD-                                                                               85 95 100                                                                               100                                                                               100                                                                               100                                                                               -- 75 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 80 100                                                                               100                                                                               100                GRASS                                                                          JOHNSON- 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 95 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 100                                                                               100                                                                               100                                                                               100                GRASS                                                                          SORGHUM  100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 95 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 100                                                                               100                                                                               100                                                                               100                NUTSEDGE 30 50 85 90 100                                                                               100                                                                               -- 70 95 100                                                                               100                                                                               100                                                                               100                                                                               -- 60 75 90 100                VELVETLEAF                                                                              25 55 75 90 100                                                                               100                                                                               -- 65 95 100                                                                               100                                                                               100                                                                               100                                                                               -- 100                                                                               100                                                                               100                                                                               100                COCKLEBUR                                                                               100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 75 90 100                                                                               100                                                                               100                                                                               100                                                                               -- 0  30 60 80                 SMARTWEED                                                                               60 80 85 90 100                                                                               100                                                                               -- 55 75 90 100                                                                               100                                                                               100                                                                               -- 60 80 100                                                                               100                LAMBS-   0  30 60 75 85 100                                                                               -- 25 50 70 90 95 100                                                                               -- 65 80 100                                                                               100                QUARTER                                                                        PIGWEED  50 85 100                                                                               100                                                                               100                                                                               100                                                                               -- 70 95 100                                                                               100                                                                               100                                                                               100                                                                               -- 65 95 100                                                                               100                MORNING- 60 75 95 100                                                                               100                                                                               100                                                                               -- 60 80 90 100                                                                               100                                                                               100                                                                               -- 85 95 100                                                                               100                GLORY                                                                          JIMSONWEED                                                                              65 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- 70 95 100                                                                               100                                                                               100                                                                               100                                                                               -- 90 100                                                                               100                                                                               100                PREEMERGENCE                                                                   CORN     -- -- 0  0  0  0  35 -- -- 0  0  0  20 40 -- -- 0  0                  SOYBEAN  -- -- 0  20 30 45 65 -- -- 0  35 60 80 100                                                                               -- -- 20 30                 GREEN FXTL                                                                              -- -- 55 85 95 95 100                                                                               -- -- 35 50 70 90 95 -- -- 25 60                 GIANT FXTL                                                                              -- -- 55 85 95 100                                                                               100                                                                               -- -- 35 50 65 85 95 -- -- 20 40                 PANICUM  -- -- 80 100                                                                               100                                                                               100                                                                               100                                                                               -- -- 65 85 100                                                                               100                                                                               100                                                                               -- -- 30 70                 CRABGRASS                                                                               -- -- 0  20 25 60 70 -- -- 0  0  0  30 40 -- -- 0  25                 BARNYARD-                                                                               -- -- 85 100                                                                               100                                                                               100                                                                               100                                                                               -- -- 30 70 85 100                                                                               100                                                                               -- -- 0  35                 GRASS                                                                          JOHNSON- -- -- 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- -- 70 100                                                                               100                                                                               100                                                                               100                                                                               -- -- 40 95                 GRASS                                                                          SORGHUM  -- -- 100                                                                               100                                                                               100                                                                               100                                                                               100                                                                               -- -- 80 100                                                                               100                                                                               100                                                                               100                                                                               -- -- 70 95                 NUTSEDGE -- -- 60 95 100                                                                               100                                                                               100                                                                               -- -- 70 85 100                                                                               100                                                                               -- -- -- 60 80                 VELVETLEAF                                                                              -- -- 0  0  0  35 60 -- -- 0  0  30 45 -- -- -- 0  0                  COCKLEBUR                                                                               -- -- 0  0  0  30 65 -- -- 0  0  0  0  -- -- -- 0  0                  SMARTWEED                                                                               -- -- 0  0  30 80 100                                                                               -- -- 30 60 80 100                                                                               -- -- -- 0  35                 LAMBS-   -- -- 0  50 80 100                                                                               100                                                                               -- -- 25 60 85 100                                                                               -- -- -- 20 60                 QUARTER                                                                        PIGWEED  -- -- 0  35 70 95 100                                                                               -- -- 0  40 75 95 -- -- -- 30 70                 MORNING- -- -- 0  0  0  30 55 -- -- 0  0  25 35 -- -- -- 0  0                  GLORY                                                                          JIMSONWEED                                                                              -- -- 0  30 45 70 100                                                                               -- -- 0  30 55 80 -- -- -- 0  30                 __________________________________________________________________________     RATE     Compound 163                                                                            Compound 165          Compound 166                           RATE GM  0062                                                                              0125                                                                              0250                                                                              0004                                                                              0008                                                                              0016                                                                               0031                                                                              0062                                                                              0125                                                                              0250                                                                              0004                                                                               0008                                                                              0016                                                                              0031                                                                              0062                                                                               0125                                                                              0250               __________________________________________________________________________     POSTEMERGENCE                                                                  CORN     55 65 -- 0  20 45  85 100                                                                               -- -- 0   0  0  0  0   25 60                 SOYBEAN  100                                                                               100                                                                               -- 100                                                                               100                                                                               100 100                                                                               100                                                                               -- -- 95  100                                                                               100                                                                               100                                                                               100 100                                                                               100                GREEN FXTL                                                                              100                                                                               100                                                                               -- 25 70 75  95 95 -- -- 70  80 85 90 95  100                                                                               100                GIANT FXTL                                                                              100                                                                               100                                                                               -- 40 90 95  100                                                                               100                                                                               -- -- 70  85 95 100                                                                               100 100                                                                               100                PANICUM  100                                                                               100                                                                               -- 100                                                                               100                                                                               100 70 100                                                                               -- -- 90  95 100                                                                               100                                                                               100 100                                                                               100                CRABGRASS                                                                               100                                                                               100                                                                               -- 20 40 60  70 100                                                                               -- -- 0   0  20 40 50  65 80                 BARNYARD-                                                                               100                                                                               100                                                                               -- 100                                                                               100                                                                               100 100                                                                               100                                                                               -- -- 95  100                                                                               100                                                                               100                                                                               100 100                                                                               100                GRASS                                                                          JOHNSON- 100                                                                               100                                                                               -- 100                                                                               100                                                                               100 70 100                                                                               -- -- 100 100                                                                               100                                                                               100                                                                               100 100                                                                               100                GRASS                                                                          SORGHUM  100                                                                               100                                                                               -- 100                                                                               100                                                                               100 100                                                                               100                                                                               -- -- 100 100                                                                               100                                                                               100                                                                               100 100                                                                               100                NUTSEDGE 100                                                                               100                                                                               -- 100                                                                               100                                                                               100 100                                                                               100                                                                               -- -- 85  100                                                                               100                                                                               100                                                                               109 100                                                                               100                VELVETLEAF                                                                              100                                                                               100                                                                               -- 90 100                                                                               100 100                                                                               100                                                                               -- -- 80  90 100                                                                               100                                                                               100 100                                                                               100                COCKLEBUR                                                                               100                                                                               100                                                                               -- 25 50 80  100                                                                               100                                                                               -- -- 95  100                                                                               100                                                                               100                                                                               100 100                                                                               100                SMARTWEED                                                                               100                                                                               100                                                                               -- 65 80 90  100                                                                               100                                                                               -- -- 45  80 90 95 100 100                                                                               100                LAMBS-   100                                                                               100                                                                               -- 40 70 85  100                                                                               100                                                                               -- -- 65  65 85 95 95  100                                                                               100                QUARTER                                                                        PIGWEED  100                                                                               100                                                                               -- 95 100                                                                               100 100                                                                               100                                                                               -- -- 90  70 100                                                                               100                                                                               100 100                                                                               100                MORNING- 100                                                                               100                                                                               -- 80 95 100 100                                                                               100                                                                               -- -- 95  100                                                                               100                                                                               100                                                                               100 100                                                                               100                GLORY                                                                          JIMSONWEED                                                                              100                                                                               100                                                                               -- 80 95 100 100                                                                               100                                                                               -- -- 85  95 100                                                                               100                                                                               100 100                                                                               100                PREEMERGENCE                                                                   CORN     0  0  20 -- 0  0   0  0  15 -- --  0  0  0  0   0  45                 SOYBEAN  40 60 80 -- 20 35  60 85 100                                                                               -- --  0  0  30 50  65 70                 GREEN FXTL                                                                              75 100                                                                               100                                                                               -- 20 50  85 100                                                                               100                                                                               -- --  0  65 85 100 100                                                                               100                GIANT FXTL                                                                              70 100                                                                               100                                                                               -- 30 70  90 100                                                                               100                                                                               -- --  0  45 85 100 100                                                                               100                PANICUM  95 100                                                                               100                                                                               -- 50 85  100                                                                               100                                                                               100                                                                               -- --  20 75 100                                                                               100 100                                                                               100                CRABGRASS                                                                               55 70 100                                                                               -- 0  30  65 90 100                                                                               -- --  0  20 35 50  65 70                 BARNYARD-                                                                               65 100                                                                               100                                                                               -- 0  20  50 90 100                                                                               -- --  0  75 100                                                                               100 100                                                                               100                GRASS                                                                          JOHNSON- 100                                                                               100                                                                               100                                                                               -- 40 85  100                                                                               100                                                                               100                                                                               -- --  70 100                                                                               100                                                                               100 100                                                                               100                GRASS                                                                          SORGHUM  100                                                                               100                                                                               100                                                                               -- 40 75  100                                                                               100                                                                               100                                                                               -- --  70 100                                                                               100                                                                               100 100                                                                               100                NUTSEDGE 95 100                                                                               100                                                                               -- 30 60  80 100                                                                               100                                                                               -- --  25 85 100                                                                               100 100                                                                               100                VELVETLEAF                                                                              25 45 80 -- 0  0   25 50 85 -- --  0  0  0  35  60 80                 COCKLEBUR                                                                               30 55 70 -- 0  0   0  35 70 -- --  0  0  0  0   30 65                 SMARTWEED                                                                               60 85 100                                                                               -- 25 50  75 95 100                                                                               -- --  30 0  20 30  50 100                LAMBS-   95 100                                                                               100                                                                               -- 20 55  70 90 100                                                                               -- --  25 25 75 100 100                                                                               100                QUARTER                                                                        PIGWEED  100                                                                               100                                                                               100                                                                               -- 30 65  90 100                                                                               100                                                                               -- --  45 30 80 100 100                                                                               100                MORNING- 20 35 70 -- 0  0   20 40 85 -- --  0  0  0  20  65 75                 GLORY                                                                          JIMSONWEED                                                                              70 90 100                                                                               -- 0  0   30 70 90 -- --  0  25 50 75  95 100                __________________________________________________________________________

TEST D

Sixteen com diameter Wagner pots, equipped with a stoppered drain opening near the bottom of the side wall, were partially filled with Woodstown sandy loam. About 1500 mls of water were added to each pot to bring the water level to a point 3 cm above the soil surface. Japonica and Indica rice seedlings were hand transplanted into the pots. Also a number of barnyardgrass (Echinochloa crusgalli) seeds were added to each pot. At the same time, seedlings or tubers of the following species were transplanted into the muddy soil: water plantain (Alisma trivale), Scirpus (Scirpus mucranatus), and Cyperus (Cyperus difformis). The weed species selected for this test are of economic importance in major rice-growing areas. The chemical treatments were applied directly to the paddy water after being formulated in a non-phytotoxic solvent within hours after transplanting of two additional species: water chestnut (Eleocharis spp.) and arrowhead (Sagittaria latifolia). Shortly after treatment, the drain hole was opened to drop the water level by two cm. Water was then added to restore the water level to its original height. The following day the draining and refilling process was repeated. The pots were then maintained in the greenhouse.

Rates of application and plant response ratings made 21 days after treatment are summarized in Table D. Response ratings are based on a scale of 0 to 100 where 0=no effect and 100=complete control.

    ______________________________________                                                  Compound 188 Compound 189                                             Rate g/ha  0016    0008   0004  0016 0008  0004                                ______________________________________                                         Japonica Rice                                                                              0       0      0    15   15     0                                  Indica Rice                                                                                0       0      0    15    0     0                                  Barnyardgrass                                                                             77      22      0    95   77    30                                  Water Chestnut                                                                            82      87     85    90   85    70                                  Arrowhead  95      90     80    92   95    87                                  Scirpus    77      80     60    87   85    67                                  Cyperus    82      55     32    95   95    92                                  Water Plantain                                                                            75      75     60    85   72    67                                  ______________________________________                                     

What is claimed is:
 1. A compound of the formula: ##STR43## wherein J is ##STR44## W is O, S or NR_(X) ; R_(X) is H, OH, C₁ -C₃ alkyl, C₁ -C₃ alkoxy, allyloxy, propargyloxy, C₁ -C₃ haloalkyl, C₁ -C₃ haloalkoxy or NR_(Y) R_(Z) ;R_(Y) is H or C₁ -C₃ alkyl; R_(Z) is C₁ -C₃ alkyl; G is O, S, SO or SO₂ ; m is 0 or 1; n is 0, 1 or 2; R is H or CH₃ ; E is a single bond, CH₂ or O; Q is ##STR45## R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(a) R_(b), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, SCN, CO₂ R_(c), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio or CN; R₂ is H, C₁ -C₃ alkyl, allyl or phenyl; R₃ is H, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, CH₂ -(C₂ -C₅ alkenyl), CH₂ (C₂ -C₅ haloalkenyl), CH₂ (C₂ -C₅ alkynyl), CH₂ (C₂ -C₅ haloalkynyl), C₆ H₅ or C₁ -C₄ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, C₁ -C₂ alkylsulfinyl or C₁ -C₂ alkylsulfonyl; R₄ is H, halogen, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, C₂ -C₆ alkenyl, C₂ -C₆ haloalkenyl, C₂ -C₆ alkynyl, C₃ -C₆ haloalkynyl, C₆ H₅, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, OCH₂ CH₂ O-(C₁ -C₂ alkyl) or di(C₁ -C₃ alkyl)amino; R₅ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, allyl or propargyl; R_(a) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy; R_(b) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or R_(a) and R_(b) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --; R_(c) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl; A is ##STR46## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₃ -C₅ cycloalkyl; Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, C₁ -C₄ haloalkyl, C₂ -C₄ alkynyl, azido, cyano, ##STR47## or --N(OCH₃)CH₃ ; p is 2 or 3; L₁ and L₂ are independently O or S; R₆ is H or CH₃ ; R₇ and R₈ are independently C₁ -C₃ alkyl; Z is CH, CCH₃, CC₂ H₅, CCl or CRr; X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl; Y₄ is CH₃, OCH₃, OC₂ H₅ or Cl; and Z¹ is N;and their agriculturally suitable salts; provided that (a) when X is Cl, F, Br or I, then Z is CH and Y is OCH₃, OC₂ H₅, N(OCH₃)CH₃, NHCH₃, N(CH₃)₂ or OCF₂ H; (b) when X or Y is C₁ haloalkoxy, then Z is CH; (c) when J is J-9 and n is 0, then Q is Q-1 or Q-2; (d) when E is O, then J is J-1; (e) when W is S, then A is A-1, R is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₃ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂ or ##STR48## (f) when the total number of carbon atoms in X and Y is greater than 4, then the carbon content of R₁, R₃, R₄ and R₅ must each be less than or equal to 2; (g) X₄ and Y₄ cannot simultaneously be Cl; (h) when J is J-1 and m is 0, then n is 0; and (i) when n is 0 and m is 1, then Q is Q-1 or Q-2.
 2. A compound of claim 1 where E is a single bond.
 3. A compound of claim 1 where E is CH₂.
 4. A compound of claim 1 where E is O.
 5. A compound of claim 2 where m is 0; and W is O.
 6. A compound of claim 5 whereX is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, cyclopropyl, Cl, F, Br, I, OCF₂ H, CH₂ F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR49## OCF₂ H, SCF₂ H, OCF₂ Br, C.tbd.CH or C.tbd.CCH₃.
 7. A compound of claim 6 whereR₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; and n is
 0. 8. A compound of claim 7 whereR₃ is H, C₁ -C₃ alkyl, C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; and R₄ is H, C₁ -C₃ alkyl, C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, N(CH₃)₂, allyl, propargyl or C₁ -C₂ alkyl substituted with 1-3 atoms of F, Cl or Br.
 9. A compound of claim 8 where J is J-1.
 10. A compound of claim 9 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 11. A compound of claim 10 where Q is Q-1.
 12. A compound of claim 10 where Q is Q-2.
 13. A compound of claim 10 where Q is Q-3.
 14. A compound of claim 10 where Q is Q-4.
 15. A compound of claim 10 where Q is Q-5.
 16. A compound of claim 10 where Q is Q-6.
 17. A compound of claim 10 where Q is Q-7.
 18. A compound of claim 8 where J is J-2.
 19. A compound of claim 18 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 20. A compound of claim 19 where Q is Q-1.
 21. A compound of claim 8 where J is J-3.
 22. A compound of claim 21 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 23. A compound of claim 22 where Q is Q-1.
 24. A compound of claim 8 where J is J-4.
 25. A compound of claim 24 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 26. A compound of claim 25 where Q is Q-1.
 27. A compound of claim 8 where J is J-5.
 28. A compound of claim 27 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 29. A compound of claim 28 where Q is Q-1.
 30. A compound of claim 8 where J is J-6.
 31. A compound of claim 30 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 32. A compound of claim 31 where Q is Q-1.
 33. A compound of claim 8 where J is J-7.
 34. A compound of claim 33 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 35. A compound of claim 34 where Q is Q-1.
 36. A compound of claim 8 where J is J-8.
 37. A compound of claim 36 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 38. A compound of claim 37 where Q is Q-1.
 39. A compound of claim 37 where Q is Q-2.
 40. A compound of claim 37 where Q is Q-3.
 41. A compound of claim 37 where Q is Q-4.
 42. A compound of claim 37 where Q is Q-5.
 43. A compound of claim 37 where Q is Q-6.
 44. A compound of claim 37 where Q is Q-7.
 45. A compound of claim 8 where J is J-9.
 46. A compound of claim 45 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 47. A compound of claim 46 where Q is Q-1.
 48. A compound of claim 8 where J is J-10.
 49. A compound of claim 48 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 50. A compound of claim 49 where Q is Q-1.
 51. A compound of claim 8 where J is J-11.
 52. A compound of claim 51 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 53. A compound of claim 52 where Q is Q-1.
 54. A compound of claim 8 where J is J-12.
 55. A compound of claim 54 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 56. A compound of claim 55 where Q is Q-1.
 57. A compound of claim 8 where J is J-13.
 58. A compound of claim 57 whereA is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 59. A compound of claim 58 where Q is Q-1.
 60. A compound of claim 3 wherem is 0; n is 0; J is J-1, J-2, J-3, J-8, J-10 or J-11; W is O; R is H; R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; R₃ is H, C₁ -C₃ alkyl, CH₂ CH₂ OCH₃, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; R₄ is H or C₁ -C₃ alkyl; A is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 61. A compound of claim 4 wherem is 0; R is H; R₁ is H; R₃ is H or C₁ -C₃ alkyl; R₄ is H or C₁ -C₃ alkyl; A is A-1; Z is CH; X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 62. The compound of claim 1 which is N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-ethyl-1H-tetrazol-5-yl)benzenesulfonamide.
 63. The compound of claim 1 which is N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-methyl-6-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide.
 64. The compound of claim 1 which is N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide.
 65. The compound of claim 1 which is N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide.
 66. The compound of claim 1 which is N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-2-(-1-methyl-1H-tetrazol-5-yl)benzenesulfonamide.
 67. The compound of claim 1 which is N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole-5-sulfonamide.
 68. The compound of claim 1 which is N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl-1H-pyrazole-5-sulfonamide.
 69. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 1 and at least one of the following: surfactant, solid or liquid diluent.
 70. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 2 and at least one of the following: surfactant, solid or liquid diluent.
 71. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 3 and at least one of the following: surfactant, solid or liquid diluent.
 72. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 4 and at least one of the following: surfactant, solid or liquid diluent.
 73. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 5 and at least one of the following: surfactant, solid or liquid diluent.
 74. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 6 and at least one of the following: surfactant, solid or liquid diluent.
 75. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 62 and at least one of the following: surfactant, solid or liquid diluent.
 76. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 63 and at least one of the following: surfactant, solid or liquid diluent.
 77. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 64 and at least one of the following: surfactant, solid or liquid diluent.
 78. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 65 and at least one of the following: surfactant, solid or liquid diluent.
 79. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 66 and at least one of the following: surfactant, solid or liquid diluent.
 80. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 67 and at least one of the following: surfactant, solid or liquid diluent.
 81. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 68 and at least one of the following: surfactant, solid or liquid diluent.
 82. A composition suitable for controlling the growth of undesired vegetation in corn which comprises an effective amount of the compound of claim 62 and at least one of the following: surfactant, solid or liquid diluent.
 83. A composition suitable for controlling the growth of undesired vegetation in corn which comprises an effective amount of the compound of claim 63 and at least one of the following: surfactant, solid or liquid diluent.
 84. A composition suitable for controlling the growth of undesired vegetation in corn which comprises an effective amount of the compound of claim 64 and at least one of the following: surfactant, solid or liquid diluent.
 85. A composition suitable for controlling the growth of undesired vegetation in corn which comprises an effective amount of the compound of claim 65 and at least one of the following: surfactant, solid or liquid diluent.
 86. A composition suitable for controlling the growth of undesired vegetation in corn which comprises an effective amount of the compound of claim 66 and at least one of the following: surfactant, solid or liquid diluent.
 87. A composition suitable for controlling the growth of undesired vegetation in rice which comprises an effective amount of the compound of claim 67 and at least one of the following: surfactant, solid or liquid diluent.
 88. A composition suitable for controlling the growth of undesired vegetation in rice which comprises an effective amount of the compound of claim 68 and at least one of the following: surfactant, solid or liquid diluent.
 89. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 1. 90. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 2. 91. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 3. 92. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 4. 93. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 5. 94. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 6. 95. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 62. 96. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 63. 97. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 64. 98. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 65. 99. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 66. 100. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 67. 101. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 68. 102. A method for controlling the growth of undesired vegetation in corn which comprises applying to the corn an effective amount of the compound of claim
 62. 103. A method for controlling the growth of undesired vegetation in corn which comprises applying to the corn an effective amount of the compound of claim
 63. 104. A method for controlling the growth of undesired vegetation in corn which comprises applying to the corn an effective amount of the compound of claim
 64. 105. A method for controlling the growth of undesired vegetation in corn which comprises applying to the corn an effective amount of the compound of claim
 65. 106. A method for controlling the growth of undesired vegetation in corn which comprises applying to the corn an effective amount of the compound of claim
 66. 107. A method for controlling the growth of undesired vegetation in rice which comprises applying to the rice an effective amount of the compound of claim
 67. 108. A method for controlling the growth of undesired vegetation in rice which comprises applying to the rice an effective amount of the compound of claim
 68. 